Target Details
| UniProt AC | Q07912 |
|---|---|
| Gene Symbol | TNK2 |
| Protein Name | Activated CDC42 kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09027 (GTPase_binding) PF11555 (Inhibitor_Mig-6) PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) PF14604 (SH3_9) |
Summary
- Multi-target molecules 222
- Clinical molecules 22
- Avg pChEMBL 7.46
Active Molecules (222)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XKFTZKGMDDZMJI
|
7.0 | Ki | 56 | — | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 91 | Yes | |
ZMWKUKIYVSUWAS
|
6.9 | IC50 | 4 | — | |
ADLPKFFMGIJZIM
|
6.9 | Ki | 44 | — | |
HFNKQEVNSGCOJV
|
6.9 | Ki | 18 | — | |
OGNYUTNQZVRGMN
|
6.9 | Ki | 16 | Yes | |
VNDWQCSOSCCWIP
|
6.9 | Ki | 39 | Yes | |
HMYOERVFCVBIDK
|
6.8 | IC50 | 2 | — | |
VRQMAABPASPXMW
|
6.8 | Kd | 10 | — | |
XLSPYLMTRXPYKY
|
6.8 | IC50 | 13 | — | |
WLKGPIPZNVLVAM
|
6.8 | IC50 | 4 | — | |
UQNNJYLAPYGZBD
|
6.8 | Ki | 28 | — | |
PBCZSGKMGDDXIJ
|
6.8 | Kd | 68 | Yes | |
JPVQIIJQJZQGID
|
6.8 | IC50 | 4 | — | |
YHVHYWYQEFELOW
|
6.8 | IC50 | 44 | — | |
VERWOWGGCGHDQE
|
6.8 | IC50 | 23 | — | |
KNNAWFQMISAWMQ
|
6.7 | IC50 | 4 | — | |
PTILEOLOGGMFCS
|
6.7 | IC50 | 2 | — | |
RSRIBZZUPWIEDF
|
6.7 | IC50 | 2 | — | |
KJMURTHIPWRIMC
|
6.7 | IC50 | 7 | — | |
CXQHYVUVSFXTMY
|
6.7 | Kd | 154 | — | |
FFCFHBVSGILIJY
|
6.7 | Ki | 17 | — | |
KFHMLBXBRCITHF
|
6.7 | IC50 | 2 | — | |
SEJGTFPOEJWEGG
|
6.7 | Kd | 149 | — | |
CSGQVNMSRKWUSH
|
6.7 | Kd | 21 | — | |
GNLAGGCSJGJECE
|
6.6 | Ki | 19 | Yes | |
SHPFDGWALWEPGS
|
6.6 | Kd | 35 | — | |
ZGDYBJXDIXVTLV
|
6.6 | Ki | 54 | — | |
FCHNDUSRWAGJES
|
6.6 | IC50 | 2 | — | |
MIMOHMCANSGXIG
|
6.6 | IC50 | 15 | — | |
WKDACQVEJIVHMZ
|
6.5 | Kd | 46 | — | |
SBWCIJOOABLPME
|
6.5 | Ki | 13 | — | |
TVLFEDKEAOXRCZ
|
6.5 | Ki | 22 | — | |
VSVWQTDDGQSGHP
|
6.5 | Ki | 51 | — | |
PNGBKTYRDRRBHW
|
6.5 | IC50 | 2 | — | |
JNXJKTXDSPWNRP
|
6.4 | Ki | 30 | — | |
KTEIFNKAUNYNJU
|
6.4 | Ki | 48 | — | |
NVRXTLZYXZNATH
|
6.4 | Ki | 47 | Yes | |
QUIQCYFSBGOBKE
|
6.4 | IC50 | 4 | — | |
LCVIRAZGMYMNNT
|
6.3 | Kd | 20 | — | |
LKCNOGUUCKOMBY
|
6.3 | Ki | 3 | — | |
WQFGNANQTYLQBP
|
6.3 | Ki | 16 | — | |
PDOQBOJDRPLBQU
|
6.3 | Kd | 21 | — | |
UJBJWYNPUOLFIZ
|
6.2 | IC50 | 49 | — | |
NYNZQNWKBKUAII
|
6.2 | IC50 | 4 | — | |
PQXQJSMNKNNINY
|
6.2 | IC50 | 2 | — | |
AEYLJTAIDDIOBA
|
6.2 | Ki | 53 | — | |
UIRCQOKSJDLYBB
|
6.2 | Ki | 50 | — | |
DDTPGANIPBKTNU
|
6.2 | IC50 | 8 | — |