Target Details
| UniProt AC | Q07912 |
|---|---|
| Gene Symbol | TNK2 |
| Protein Name | Activated CDC42 kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09027 (GTPase_binding) PF11555 (Inhibitor_Mig-6) PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) PF14604 (SH3_9) |
Summary
- Multi-target molecules 222
- Clinical molecules 22
- Avg pChEMBL 7.46
Active Molecules (222)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PESNFBOGJFKUMG
|
7.6 | IC50 | 2 | — | |
JJBNBDJXYZZFBC
|
7.6 | IC50 | 3 | — | |
XNFHHOXCDUAYSR
|
7.6 | IC50 | 5 | — | |
IFRQDJZBFXKVOQ
|
7.6 | IC50 | 2 | — | |
LBVKEEFIPBQIMD
|
7.6 | Ki | 27 | — | |
LJKJYKWDLJUZHA
|
7.6 | Ki | 24 | — | |
SZNYUUZOQHNEKB
|
7.6 | IC50 | 7 | — | |
VPOWOPVCLUEIIA
|
7.6 | IC50 | 2 | — | |
FZPWJZCQBCBZKE
|
7.6 | IC50 | 2 | — | |
GGGQYLRXTXDJRN
|
7.6 | IC50 | 2 | — | |
DKNACWKOKCXDEJ
|
7.6 | IC50 | 2 | — | |
VAARYSWULJUGST
|
7.6 | Kd | 119 | Yes | |
GWFZRGVIOWEPRA
|
7.5 | IC50 | 2 | — | |
OHBDADSLOSGAHB
|
7.5 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
7.5 | Ki | 66 | — | |
MOHYPRXHKRXDSE
|
7.5 | IC50 | 8 | — | |
GXLCEYYXBWDRJO
|
7.5 | IC50 | 3 | — | |
NEIVLVMGHRRCDM
|
7.5 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — | |
UEEVERDPEVIFBH
|
7.4 | IC50 | 2 | — | |
JWXZQEPPXRGVKZ
|
7.4 | IC50 | 3 | — | |
IOSKHROQBBQEOB
|
7.4 | IC50 | 2 | — | |
GPJRGBLZCBBYMB
|
7.4 | IC50 | 2 | — | |
FJABJYQHNWUFPP
|
7.4 | IC50 | 2 | — | |
PIMBZWQACDWQJV
|
7.4 | IC50 | 2 | — | |
UYJNQQDJUOUFQJ
|
7.4 | Ki | 68 | — | |
LAJAFFLJAJMYLK
|
7.4 | IC50 | 17 | — | |
OSVUGUHRKMMBSE
|
7.4 | Kd | 170 | — | |
KOMGSVVWXUEBNT
|
7.3 | IC50 | 3 | — | |
HMVDGWSYIBOKRV
|
7.3 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.2 | Kd | 64 | Yes | |
FCMKRDBRBZALAL
|
7.2 | IC50 | 2 | — | |
RGNHKJWHFIPHIM
|
7.2 | Ki | 66 | — | |
RYYNGWLOYLRZLK
|
7.2 | Ki | 104 | — | |
JOOXLOJCABQBSG
|
7.2 | Kd | 139 | — | |
UEVFMGJBRLJVKO
|
7.2 | IC50 | 3 | — | |
HAYYBYPASCDWEQ
|
7.2 | IC50 | 47 | — | |
DUYJMQONPNNFPI
|
7.2 | IC50 | 11 | — | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
ALKJNCZNEOTEMP
|
7.1 | Kd | 55 | — | |
SSVDSZIWJBBCNN
|
7.1 | IC50 | 4 | Yes | |
PROLIXHVRCJEFH
|
7.1 | Ki | 46 | — | |
WYNDNQIGGGWABE
|
7.1 | IC50 | 4 | — | |
SXBGVYYYZFBEKG
|
7.1 | IC50 | 2 | — | |
BDRDZIHCMNAENW
|
7.1 | IC50 | 2 | — | |
YKMSWECJITXGJA
|
7.0 | IC50 | 2 | — | |
KNRKFYBCACDGCC
|
7.0 | IC50 | 2 | — | |
DMZTWOCJNVKCBW
|
7.0 | IC50 | 6 | Yes | |
SWTRMCZKDHCOOZ
|
7.0 | IC50 | 2 | — | |
HZPACYSNLOCDLW
|
7.0 | Ki | 48 | — |