Target Details
| UniProt AC | Q07912 |
|---|---|
| Gene Symbol | TNK2 |
| Protein Name | Activated CDC42 kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09027 (GTPase_binding) PF11555 (Inhibitor_Mig-6) PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) PF14604 (SH3_9) |
Summary
- Multi-target molecules 222
- Clinical molecules 22
- Avg pChEMBL 7.46
Active Molecules (222)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FJOFREJOLJFMNF
|
8.2 | IC50 | 3 | — | |
FSFKDNPHPFINJD
|
8.2 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
ORSBXGBOZDSEJT
|
8.2 | IC50 | 3 | — | |
IYUXAJHPXXWFQO
|
8.2 | IC50 | 2 | — | |
CAQLNQYCCKYWJX
|
8.1 | Ki | 5 | Yes | |
FCMNXGJPIJFWQV
|
8.1 | IC50 | 2 | — | |
WPHKIQPVPYJNAX
|
8.1 | Ki | 81 | — | |
AMWNTQXPBJQZET
|
8.1 | IC50 | 3 | — | |
NBZFRTJWEIHFPF
|
8.1 | IC50 | 3 | — | |
OHPMDANXCFNAPB
|
8.0 | IC50 | 2 | — | |
QSDUGBPLSHIMHQ
|
8.0 | IC50 | 3 | — | |
SVYQAPDHJLXDGC
|
8.0 | IC50 | 3 | — | |
AURCLDMUVVKGCY
|
8.0 | IC50 | 3 | — | |
DPKCTDXZHPAPLS
|
8.0 | IC50 | 3 | — | |
PTHVKCSYXICMAR
|
8.0 | IC50 | 14 | — | |
USVYVEUGCBHMNU
|
8.0 | IC50 | 2 | — | |
XNSZHQUDPHATEN
|
8.0 | IC50 | 2 | — | |
SJYGJUQORXZRIJ
|
7.9 | IC50 | 3 | — | |
LZKGLICEGUTSDW
|
7.9 | IC50 | 3 | — | |
BRTHUECZMVKNMQ
|
7.9 | Ki | 31 | — | |
FACSDOITOHWERB
|
7.9 | IC50 | 2 | — | |
GDRLJBDXWDATLA
|
7.9 | IC50 | 13 | — | |
REEJHXFEIZURCB
|
7.9 | IC50 | 2 | — | |
WEFPHDYTHUNVAM
|
7.9 | IC50 | 3 | — | |
UCQAPUVIUAYEGE
|
7.9 | IC50 | 3 | — | |
GDVRVPIXWXOKQO
|
7.8 | IC50 | 10 | — | |
TWZQEBQCXWLACN
|
7.8 | IC50 | 3 | — | |
ZMRSDMLCFJDLKR
|
7.8 | IC50 | 3 | — | |
DILZMEVBCHRKIZ
|
7.8 | IC50 | 3 | — | |
DFHIKCGHCSDYRT
|
7.8 | IC50 | 2 | — | |
DIXMBHMNEHPFCX
|
7.8 | IC50 | 12 | — | |
LGLHCXISMKHLIK
|
7.8 | Kd | 3 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 213 | — | |
OXULFDKDMPHAFP
|
7.8 | IC50 | 3 | — | |
VCFDMLBPASGZTP
|
7.8 | Ki | 38 | — | |
YSWLNXFQMMFDFG
|
7.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
IIXWYSCJSQVBQM
|
7.8 | IC50 | 18 | — | |
VXYZCOCRVAQWBG
|
7.8 | IC50 | 15 | — | |
YHTSUIXFAAQWLU
|
7.8 | IC50 | 2 | — | |
ZWVLMQTXUWMUII
|
7.7 | IC50 | 9 | Yes | |
GPXBXXGIAQBQNI
|
7.7 | IC50 | 11 | — | |
CLLDBMRRUZYRLR
|
7.7 | Ki | 3 | — | |
KNRXPUFRSHTQJW
|
7.7 | IC50 | 2 | — | |
PWPDYURZGAQWPZ
|
7.7 | IC50 | 2 | — | |
QKKHXTGUTLRIAS
|
7.7 | IC50 | 4 | — | |
AQVOAZGKJLFRRO
|
7.7 | IC50 | 2 | — | |
BIMOMBRKBARWLJ
|
7.7 | IC50 | 2 | — | |
ZHOXAGNPCZTRBN
|
7.7 | Kd | 20 | — |