Target Details
| UniProt AC | Q07912 |
|---|---|
| Gene Symbol | TNK2 |
| Protein Name | Activated CDC42 kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09027 (GTPase_binding) PF11555 (Inhibitor_Mig-6) PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) PF14604 (SH3_9) |
Summary
- Multi-target molecules 222
- Clinical molecules 22
- Avg pChEMBL 7.46
Active Molecules (222)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IHWDTUMEQRTNBN
|
9.6 | Ki | 2 | — | |
NPJLFKUSWFFZLW
|
9.5 | IC50 | 2 | — | |
RSZFCUWJGDNCGK
|
9.0 | IC50 | 3 | — | |
CYXPHNZJEDAZDD
|
9.0 | IC50 | 2 | — | |
IFPPYSWJNWHOLQ
|
8.9 | Ki | 52 | Yes | |
JQJGYBASPJXNIJ
|
8.9 | IC50 | 3 | — | |
IXNZYKNOAINDTN
|
8.9 | IC50 | 3 | — | |
XUFWBGKENCGHSD
|
8.9 | IC50 | 3 | — | |
OCLDJPYPPFDDNO
|
8.9 | IC50 | 3 | — | |
GRPXLKXGJAGYSD
|
8.8 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.8 | Ki | 118 | — | |
DBLBOZLZPCJKAH
|
8.8 | IC50 | 3 | — | |
OUERNEXEYTUWRZ
|
8.8 | IC50 | 3 | — | |
PZYRHYWULWFGBG
|
8.8 | IC50 | 3 | — | |
ZJLXSIPWULUCRJ
|
8.8 | IC50 | 5 | — | |
UOAHTPZUUUBPBK
|
8.7 | IC50 | 3 | — | |
CVLCVUYBIPUQBG
|
8.7 | IC50 | 3 | — | |
DRPXVULWOOOZDV
|
8.7 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
8.7 | Kd | 231 | Yes | |
WQVZBZQCVBIXLT
|
8.7 | IC50 | 3 | — | |
NJQTWWNECKEAQJ
|
8.7 | IC50 | 3 | — | |
RAPGQTWOPCNSEJ
|
8.7 | IC50 | 3 | — | |
OTDIMNJLKVGGOB
|
8.6 | IC50 | 3 | — | |
RLKUZCOFKFUEHH
|
8.6 | IC50 | 3 | — | |
ONEIDYKHPRMDQO
|
8.6 | IC50 | 3 | — | |
QAJSMIVRRQDYBG
|
8.6 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
8.6 | IC50 | 130 | Yes | |
UWIOUEAALWYOMW
|
8.6 | IC50 | 3 | — | |
DVBFHLPDOMIKKR
|
8.6 | IC50 | 3 | — | |
XFINPBQKFDIRJH
|
8.5 | IC50 | 3 | — | |
JQGBWSRCIMCMTI
|
8.5 | IC50 | 2 | — | |
PITKHMJQSBHPED
|
8.5 | IC50 | 3 | — | |
CBRIZHZYFLCPAP
|
8.5 | IC50 | 3 | — | |
NZDMYHLPDHCLGC
|
8.5 | IC50 | 3 | — | |
SOASXIFPFLUWRH
|
8.5 | IC50 | 3 | — | |
QWQRHMZFZSWUOD
|
8.4 | IC50 | 3 | — | |
CINNRILLZCDNOZ
|
8.4 | IC50 | 3 | — | |
VAOQBNBDBKHNQY
|
8.4 | IC50 | 3 | — | |
OWRXHGAFWZFFCW
|
8.4 | Ki | 113 | — | |
CDELRUCHGDJWNM
|
8.4 | IC50 | 3 | — | |
INRRUWSEBDJLPW
|
8.4 | IC50 | 3 | — | |
CCWTWPIDXUGAKX
|
8.3 | IC50 | 3 | — | |
WPSFTNDXYZENJA
|
8.3 | IC50 | 3 | — | |
CVTFVYCHNGODLR
|
8.3 | IC50 | 3 | — | |
FBIGNDFZRCUSDQ
|
8.3 | IC50 | 3 | — | |
MGGBYMDAPCCKCT
|
8.3 | IC50 | 23 | — | |
ZBNZXTGUTAYRHI
|
8.2 | Kd | 102 | Yes | |
BJKWAQGXAVDGLG
|
8.2 | IC50 | 2 | — | |
WPTNASIDXWQCDG
|
8.2 | IC50 | 3 | — | |
MWLJLVHPVHBVDL
|
8.2 | IC50 | 3 | — |