Target Details
| UniProt AC | Q07889 |
|---|---|
| Gene Symbol | SOS1 |
| Protein Name | Son of sevenless homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00617 (RasGEF) PF00618 (RasGEF_N) PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 766
- Clinical molecules 0
- Avg pChEMBL 8.12
KEGG Pathways (48)
- Acute myeloid leukemia
- Alcoholism
- B cell receptor signaling pathway
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Choline metabolism in cancer
- Chronic myeloid leukemia
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Estrogen signaling pathway
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gap junction
- Gastric cancer
- Glioma
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- JAK-STAT signaling pathway
- MAPK signaling pathway
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prolactin signaling pathway
- Prostate cancer
- Proteoglycans in cancer
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
- Thermogenesis
- mTOR signaling pathway
Associated Diseases (3)
Active Molecules (766)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MOMAMGKWTZLCAU
|
8.1 | IC50 | 2 | — | |
DMNIDOMEYCRERJ
|
8.1 | IC50 | 2 | — | |
HQHMWIQHZFTBKR
|
8.1 | IC50 | 2 | — | |
IUPOREKKZPGXSB
|
8.1 | IC50 | 2 | — | |
LECCRWPQHHHXEG
|
8.1 | Kd | 2 | — | |
LPHCLPWKMGJBNW
|
8.1 | Kd | 2 | — | |
LSHAFPJTIGEDAX
|
8.1 | IC50 | 2 | — | |
LUKKJFYKNFEPFN
|
8.1 | IC50 | 2 | — | |
MSNZQZZNHYNTPM
|
8.1 | IC50 | 2 | — | |
MVNCRRMRZYSLCY
|
8.1 | IC50 | 2 | — | |
QBSMNOSDQQLYHO
|
8.1 | IC50 | 2 | — | |
QLZCREPUWVDVHA
|
8.1 | IC50 | 2 | — | |
RRYXLEUQMGWADQ
|
8.1 | Kd | 2 | — | |
RVDRLOFLZMAVBK
|
8.1 | Kd | 2 | — | |
URUBHTZQWCSUEV
|
8.1 | IC50 | 2 | — | |
USMFBWGAPMHVGN
|
8.1 | Kd | 2 | — | |
WTWLSKFEVQIZPA
|
8.1 | IC50 | 2 | — | |
XDXFVTLDOBJHDT
|
8.1 | IC50 | 2 | — | |
YAUPEDUOPVBUJQ
|
8.1 | Kd | 2 | — | |
ZBFAZPBBZRKBNE
|
8.1 | Kd | 2 | — | |
ZLGDRFGKFHUPTB
|
8.1 | IC50 | 2 | — | |
DTVYAWHQQPAKGA
|
8.1 | Kd | 2 | — | |
VGLWPCBCFZPMQZ
|
8.1 | Kd | 2 | — | |
KKFFOOWORPUAJB
|
8.1 | IC50 | 2 | — | |
DJESUWUXSVTYRR
|
8.1 | IC50 | 2 | — | |
KVNAVABONRFGHA
|
8.1 | IC50 | 2 | — | |
ONDHAZVEHVKYBQ
|
8.1 | IC50 | 2 | — | |
PYLGLCLYBWAHJY
|
8.1 | Kd | 2 | — | |
SSBLSQBAYIUCDQ
|
8.1 | IC50 | 2 | — | |
KXODPSQLBUFDCE
|
8.1 | IC50 | 2 | — | |
RSEWFMXCMHFDMS
|
8.1 | IC50 | 2 | — | |
STSSGPBVWJDERO
|
8.1 | Kd | 2 | — | |
UVNQICXVXBBWBT
|
8.1 | IC50 | 2 | — | |
AKUAKPHLDHMFDX
|
8.1 | IC50 | 2 | — | |
ARMUZAKSBNFJME
|
8.1 | Kd | 2 | — | |
AUBYCSKNJWSVFD
|
8.1 | IC50 | 2 | — | |
AWRAQZZUQMLMMB
|
8.1 | IC50 | 2 | — | |
BZVKJAWBMYKQLU
|
8.1 | IC50 | 2 | — | |
CMSYJDFFDZBJTR
|
8.1 | IC50 | 2 | — | |
FMORUOSRPGLYNK
|
8.1 | Kd | 2 | — | |
IGWYEWFTIGJUQM
|
8.1 | IC50 | 2 | — | |
IUZDRIVOGKPURG
|
8.1 | Kd | 2 | — | |
JMJBAHZUQNQSGI
|
8.1 | IC50 | 2 | — | |
LGIUONROHUVWNX
|
8.1 | Kd | 2 | — | |
LYQVHQDNXIBVDN
|
8.1 | Kd | 2 | — | |
MDEUMDPWTVDPGV
|
8.1 | IC50 | 2 | — | |
MPVFMKBXBRSUAA
|
8.1 | IC50 | 2 | — | |
QXIMKFJETXWZKS
|
8.1 | IC50 | 2 | — | |
RLRRQDYPUVUPOP
|
8.1 | Kd | 2 | — | |
ROVMEWOBLJKPAY
|
8.1 | IC50 | 2 | — |