Target Details
| UniProt AC | Q07889 |
|---|---|
| Gene Symbol | SOS1 |
| Protein Name | Son of sevenless homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00617 (RasGEF) PF00618 (RasGEF_N) PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 766
- Clinical molecules 0
- Avg pChEMBL 8.12
KEGG Pathways (48)
- Acute myeloid leukemia
- Alcoholism
- B cell receptor signaling pathway
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Choline metabolism in cancer
- Chronic myeloid leukemia
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Estrogen signaling pathway
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gap junction
- Gastric cancer
- Glioma
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- JAK-STAT signaling pathway
- MAPK signaling pathway
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prolactin signaling pathway
- Prostate cancer
- Proteoglycans in cancer
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
- Thermogenesis
- mTOR signaling pathway
Associated Diseases (3)
Active Molecules (766)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OSWCMMCAVFTCGC
|
8.2 | IC50 | 2 | — | |
OTMRVBJWLVHJRM
|
8.2 | IC50 | 2 | — | |
QGLOQVAVWPSGHC
|
8.2 | IC50 | 2 | — | |
RMNFJVXZIPSSOK
|
8.2 | IC50 | 2 | — | |
RNHIVUSKTFSCIP
|
8.2 | IC50 | 2 | — | |
UOTULNIUFKCFLM
|
8.2 | Kd | 2 | — | |
UPGJJZISRBTWIN
|
8.2 | IC50 | 2 | — | |
UPPJSQLSZZMFNI
|
8.2 | IC50 | 2 | — | |
UUYULGJWPNXBGF
|
8.2 | IC50 | 2 | — | |
VMNMFAMIABBFQC
|
8.2 | IC50 | 2 | — | |
VQMPMEMPTDGWLT
|
8.2 | IC50 | 2 | — | |
VYVNAHNGENYHPP
|
8.2 | IC50 | 2 | — | |
XTIJSWBXVSEYPU
|
8.2 | IC50 | 2 | — | |
YKPJANMSGCSQFF
|
8.2 | IC50 | 2 | — | |
ZWDJXGMYAKFYGQ
|
8.2 | IC50 | 2 | — | |
ISRQTEUZJGHSGH
|
8.2 | IC50 | 2 | — | |
RSEWFMXCMHFDMS
|
8.2 | IC50 | 2 | — | |
PEXUVLCXACJAGY
|
8.2 | IC50 | 2 | — | |
BUFOCMAFUZPDHU
|
8.2 | IC50 | 2 | — | |
HZCDDUMYOSCMEQ
|
8.2 | Kd | 2 | — | |
ISDZPRLWPGBJIB
|
8.2 | IC50 | 2 | — | |
BCSZTRLTTXRNLL
|
8.2 | IC50 | 2 | — | |
BCTYHPPAFUEFCP
|
8.2 | IC50 | 2 | — | |
BCTYHPPAFUEFCP
|
8.2 | IC50 | 2 | — | |
CKAMBYUZKWQCKJ
|
8.2 | IC50 | 2 | — | |
CRSGWJXJQPUQLH
|
8.2 | IC50 | 2 | — | |
FMORUOSRPGLYNK
|
8.2 | Kd | 2 | — | |
FRPITCBVFZSSRV
|
8.2 | IC50 | 2 | — | |
IFWWCAXIGLYBCF
|
8.2 | IC50 | 2 | — | |
IGSHOKJBHODTOI
|
8.2 | IC50 | 2 | — | |
IHDBFLWRENURNH
|
8.2 | IC50 | 2 | — | |
IIGDOSIRBAMELH
|
8.2 | IC50 | 2 | — | |
IOOYTXLGBJLPLO
|
8.2 | IC50 | 2 | — | |
IUZDRIVOGKPURG
|
8.2 | Kd | 2 | — | |
OAWXSVRKCSVVLS
|
8.2 | IC50 | 2 | — | |
PBPYBHPRAQXQCB
|
8.2 | Kd | 2 | — | |
PSZWQWGFXMXQLQ
|
8.2 | IC50 | 2 | — | |
PXKAELQVWYOADZ
|
8.2 | IC50 | 2 | — | |
RFOZVBBBQXEUFS
|
8.2 | IC50 | 2 | — | |
SEJYEYDGHUWBEN
|
8.2 | IC50 | 2 | — | |
SHJPDYSLZPVWNH
|
8.2 | IC50 | 2 | — | |
TWVQBTCNHBHZAV
|
8.2 | IC50 | 2 | — | |
UFEBIPUVEJHURX
|
8.2 | IC50 | 2 | — | |
VKXOZRXFOLMYTB
|
8.2 | IC50 | 2 | — | |
YPSONZJHQZOMBF
|
8.2 | IC50 | 2 | — | |
ZLIYCWXQQAHPJC
|
8.2 | IC50 | 2 | — | |
HYZAOVIBHSDAHI
|
8.1 | IC50 | 2 | — | |
PAJFXVZZBJNSHN
|
8.1 | IC50 | 2 | — | |
PGQDMPGFHCCYAL
|
8.1 | IC50 | 2 | — | |
IGXFSCUDQOSJQK
|
8.1 | IC50 | 2 | — |