Target Details
| UniProt AC | Q07889 |
|---|---|
| Gene Symbol | SOS1 |
| Protein Name | Son of sevenless homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00617 (RasGEF) PF00618 (RasGEF_N) PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 766
- Clinical molecules 0
- Avg pChEMBL 8.12
KEGG Pathways (48)
- Acute myeloid leukemia
- Alcoholism
- B cell receptor signaling pathway
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Choline metabolism in cancer
- Chronic myeloid leukemia
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Estrogen signaling pathway
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gap junction
- Gastric cancer
- Glioma
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- JAK-STAT signaling pathway
- MAPK signaling pathway
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prolactin signaling pathway
- Prostate cancer
- Proteoglycans in cancer
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
- Thermogenesis
- mTOR signaling pathway
Associated Diseases (3)
Active Molecules (766)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVSQQYYKYZLOBJ
|
8.5 | IC50 | 2 | — | |
YZLQQBQMEPAKOK
|
8.5 | IC50 | 2 | — | |
YZSGRZKAZJBVMH
|
8.5 | IC50 | 2 | — | |
ZIMSKVCOCJHPKL
|
8.5 | IC50 | 2 | — | |
INNCCXSGHDHCIX
|
8.5 | IC50 | 2 | — | |
ACNIGGXNBAGWAL
|
8.5 | IC50 | 2 | — | |
ALKBXXQEXQYHTE
|
8.5 | IC50 | 2 | — | |
CWXWRDKIANATGM
|
8.5 | Kd | 2 | — | |
JESLNXDJBCYBBK
|
8.5 | IC50 | 2 | — | |
VQQQDOFXWFHFFS
|
8.4 | IC50 | 2 | — | |
KRRQLEVIPFKSQQ
|
8.4 | IC50 | 2 | — | |
NXUXDOAOHBPRPQ
|
8.4 | IC50 | 2 | — | |
AMJPASDPTHFZEA
|
8.4 | Kd | 2 | — | |
FHNTVNJVRBRJNA
|
8.4 | IC50 | 2 | — | |
FHYUPAHDRNXBQT
|
8.4 | IC50 | 2 | — | |
FNCBEVUDTZYUJD
|
8.4 | IC50 | 2 | — | |
FOMRDGOGXWHHPF
|
8.4 | IC50 | 2 | — | |
FRJGHWCMERVQNX
|
8.4 | IC50 | 2 | — | |
GPVOHUGMEQFZAX
|
8.4 | IC50 | 2 | — | |
GSIYKERYWYJMIC
|
8.4 | IC50 | 2 | — | |
HDMYPMZLPCHKHK
|
8.4 | IC50 | 2 | — | |
HNVFYUAXKGDPJY
|
8.4 | IC50 | 2 | — | |
HOWMCJREBXFBJM
|
8.4 | IC50 | 2 | — | |
IBUDGJIEMFVDDJ
|
8.4 | IC50 | 2 | — | |
KJXDYWKYMITBKG
|
8.4 | IC50 | 2 | — | |
KPCHQBHOEVTDBB
|
8.4 | IC50 | 2 | — | |
LQSDQSCCYWXGNW
|
8.4 | IC50 | 2 | — | |
NCAVQQNNPWZUEZ
|
8.4 | IC50 | 2 | — | |
NXZGIEBGFDSHKM
|
8.4 | IC50 | 2 | — | |
PFXGGGUFVBVCGD
|
8.4 | IC50 | 2 | — | |
PRLBGKOQFVUAPC
|
8.4 | IC50 | 2 | — | |
SFOBNFTWEMNFEH
|
8.4 | IC50 | 2 | — | |
SQRRKLYAIUOFDH
|
8.4 | IC50 | 2 | — | |
SVVNXAJLFMJMJA
|
8.4 | IC50 | 2 | — | |
UOWZLEGGMBTOCO
|
8.4 | IC50 | 2 | — | |
VRYFRNUPBQYDAQ
|
8.4 | IC50 | 2 | — | |
WKDDDYCTFFFIOR
|
8.4 | IC50 | 2 | — | |
WSXVXASFVIUABY
|
8.4 | IC50 | 2 | — | |
XAUKQADSCJLOPS
|
8.4 | IC50 | 2 | — | |
XDWYDGMJVUZRHA
|
8.4 | IC50 | 2 | — | |
XHKJENSQDYMNJN
|
8.4 | IC50 | 2 | — | |
XIOJXVPOGOHKBM
|
8.4 | IC50 | 2 | — | |
XWBGXHFUUDQMRY
|
8.4 | IC50 | 2 | — | |
YPSNSQLMXKKCLN
|
8.4 | IC50 | 2 | — | |
ZNRNWQQVBXCLRX
|
8.4 | IC50 | 2 | — | |
ZOIFVYFBAFEMST
|
8.4 | IC50 | 2 | — | |
LRHZAWQNSKBZFA
|
8.4 | IC50 | 2 | — | |
HLRZUCSGYSFJQJ
|
8.4 | IC50 | 2 | — | |
VBJCXRRBKBYGTG
|
8.3 | IC50 | 2 | — | |
WASPCBWBJXQVDJ
|
8.3 | Kd | 2 | — |