Target Details
| UniProt AC | Q07889 |
|---|---|
| Gene Symbol | SOS1 |
| Protein Name | Son of sevenless homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00617 (RasGEF) PF00618 (RasGEF_N) PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 766
- Clinical molecules 0
- Avg pChEMBL 8.12
KEGG Pathways (48)
- Acute myeloid leukemia
- Alcoholism
- B cell receptor signaling pathway
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Choline metabolism in cancer
- Chronic myeloid leukemia
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Estrogen signaling pathway
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gap junction
- Gastric cancer
- Glioma
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- JAK-STAT signaling pathway
- MAPK signaling pathway
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prolactin signaling pathway
- Prostate cancer
- Proteoglycans in cancer
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
- Thermogenesis
- mTOR signaling pathway
Associated Diseases (3)
Active Molecules (766)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OCEXUDSXGGCFOS
|
8.6 | IC50 | 2 | — | |
RSPVPSCYTHCDDW
|
8.6 | IC50 | 2 | — | |
CSMXSTFEQJRFJB
|
8.6 | IC50 | 2 | — | |
HKMMDGCMFRMCTQ
|
8.6 | IC50 | 2 | — | |
OJAZNZNRLFBVEV
|
8.6 | IC50 | 2 | — | |
POJLABBZRFQKHP
|
8.6 | IC50 | 2 | — | |
TVJCBPMURLWQQQ
|
8.6 | IC50 | 2 | — | |
YBDSRLUXKOTGRW
|
8.6 | IC50 | 2 | — | |
YPXMSOODCRETLP
|
8.6 | IC50 | 2 | — | |
CECUHSUUFDBRNE
|
8.5 | IC50 | 2 | — | |
CNZVROLTTYQZCO
|
8.5 | IC50 | 2 | — | |
CPEJDIYHZXLMJL
|
8.5 | IC50 | 2 | — | |
CTWHCQOSGTUDTI
|
8.5 | IC50 | 2 | — | |
DFXYJVTZPXGTKU
|
8.5 | IC50 | 2 | — | |
GJRKVDBUKDWBRM
|
8.5 | IC50 | 2 | — | |
GRFGEXVYYJKXPK
|
8.5 | IC50 | 2 | — | |
HORHVFVJWRHQID
|
8.5 | IC50 | 2 | — | |
HSFCTTCKKBNWLI
|
8.5 | IC50 | 2 | — | |
IJELKIMNCCSKKG
|
8.5 | IC50 | 2 | — | |
JGAYIHIFGNIEAN
|
8.5 | IC50 | 2 | — | |
JJTCEMCNXITBQK
|
8.5 | IC50 | 2 | — | |
JRCWKCYVDQCETC
|
8.5 | IC50 | 2 | — | |
KVMGOGUJOBTQKJ
|
8.5 | IC50 | 2 | — | |
KWPMDODRFACSFM
|
8.5 | IC50 | 2 | — | |
LAXAYIVRADCESX
|
8.5 | IC50 | 2 | — | |
LQAYWPGINPYXTE
|
8.5 | IC50 | 2 | — | |
LTINNJDDPBZKGA
|
8.5 | Kd | 2 | — | |
MQLHOXHYDKDBPX
|
8.5 | IC50 | 2 | — | |
NPAKABRGRUPLNZ
|
8.5 | Kd | 2 | — | |
NXJNVANYUDNXMJ
|
8.5 | IC50 | 2 | — | |
OAENWTVDYYRWNW
|
8.5 | IC50 | 2 | — | |
OFKDAUIZYWMMLO
|
8.5 | IC50 | 2 | — | |
OHOLRBJMYCLZRA
|
8.5 | IC50 | 2 | — | |
OPQNXQCZVZVYPZ
|
8.5 | IC50 | 2 | — | |
OXIGZAOWYOKHSH
|
8.5 | IC50 | 2 | — | |
PAAVVYUMFVJLBV
|
8.5 | IC50 | 2 | — | |
PIZOZWTXVFXEEL
|
8.5 | IC50 | 2 | — | |
QDHCSNMFEDWAKH
|
8.5 | Kd | 2 | — | |
QFFBMTWOIWAMIX
|
8.5 | IC50 | 2 | — | |
RDIDJQIMCDBIGJ
|
8.5 | IC50 | 2 | — | |
UBXUFHLYDGKITG
|
8.5 | IC50 | 2 | — | |
USMFBWGAPMHVGN
|
8.5 | Kd | 2 | — | |
VGMNONGKEKVCEM
|
8.5 | IC50 | 2 | — | |
VPLCGSAAJJRSQW
|
8.5 | IC50 | 2 | — | |
VSESPOILRXPQEM
|
8.5 | IC50 | 2 | — | |
VUGHUHODOMWWDI
|
8.5 | IC50 | 2 | — | |
XWUVXZLOVONISO
|
8.5 | Kd | 2 | — | |
XZCGBNGXGZJFCN
|
8.5 | IC50 | 2 | — | |
YEUAJBKCOKIMCY
|
8.5 | IC50 | 2 | — | |
YJTUSRMMESLSMY
|
8.5 | IC50 | 2 | — |