Target Details
| UniProt AC | Q07889 |
|---|---|
| Gene Symbol | SOS1 |
| Protein Name | Son of sevenless homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00617 (RasGEF) PF00618 (RasGEF_N) PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 766
- Clinical molecules 0
- Avg pChEMBL 8.12
KEGG Pathways (48)
- Acute myeloid leukemia
- Alcoholism
- B cell receptor signaling pathway
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Choline metabolism in cancer
- Chronic myeloid leukemia
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Estrogen signaling pathway
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gap junction
- Gastric cancer
- Glioma
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- JAK-STAT signaling pathway
- MAPK signaling pathway
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prolactin signaling pathway
- Prostate cancer
- Proteoglycans in cancer
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
- Thermogenesis
- mTOR signaling pathway
Associated Diseases (3)
Active Molecules (766)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GHGDXGIBYAFMJZ
|
8.8 | IC50 | 2 | — | |
IAZGWTRECHWLPL
|
8.8 | IC50 | 2 | — | |
LBTUDOHVURPDGN
|
8.8 | IC50 | 2 | — | |
NCLOBZVMMQYFSX
|
8.8 | IC50 | 2 | — | |
NSMSPIWWMSZJJZ
|
8.8 | IC50 | 2 | — | |
ONKIFAGLVVECAM
|
8.8 | IC50 | 2 | — | |
ONZZIAUUSXABMR
|
8.8 | IC50 | 2 | — | |
QUQACOALGFSPEZ
|
8.8 | IC50 | 2 | — | |
RFGJVVZPNHJTRE
|
8.8 | IC50 | 2 | — | |
SGDPSOKNGBLBJZ
|
8.8 | IC50 | 2 | — | |
SOYNBRLHXZQDLA
|
8.8 | IC50 | 2 | — | |
VEXRXMWZGLSCPC
|
8.8 | IC50 | 2 | — | |
HRTWETMBLURISK
|
8.8 | IC50 | 2 | — | |
AAERNVBNVNZFKK
|
8.7 | IC50 | 2 | — | |
AFONTOFZLGSFJN
|
8.7 | IC50 | 2 | — | |
ANIPNHZWVMYJLY
|
8.7 | IC50 | 2 | — | |
BEUZFLDAEOFGNM
|
8.7 | IC50 | 2 | — | |
BGRKBJVMTURZBQ
|
8.7 | IC50 | 2 | — | |
BKDXPAAVRWPDPX
|
8.7 | IC50 | 2 | — | |
BUIOJFPVYMAXFD
|
8.7 | IC50 | 2 | — | |
CDEMFJBHKSTJBV
|
8.7 | IC50 | 2 | — | |
CMCXWVBCHOAIEX
|
8.7 | IC50 | 2 | — | |
CPDOGCGQQAAZIW
|
8.7 | IC50 | 2 | — | |
CPDOGCGQQAAZIW
|
8.7 | IC50 | 2 | — | |
CSSFWSFGMVJSAN
|
8.7 | IC50 | 2 | — | |
CXWDWXDMNLGZBW
|
8.7 | IC50 | 2 | — | |
DCFCUOGLXHAKCW
|
8.7 | IC50 | 2 | — | |
FGZLNWASTZPNLC
|
8.7 | IC50 | 2 | — | |
FTWZLBLTONBYHH
|
8.7 | IC50 | 2 | — | |
FYUQBUWDBFQWEV
|
8.7 | IC50 | 2 | — | |
GBCFKGCLSSSUMK
|
8.7 | IC50 | 2 | — | |
GERUSBHCFZPWDM
|
8.7 | IC50 | 2 | — | |
GFONDRQIDTUGNO
|
8.7 | IC50 | 2 | — | |
GFONDRQIDTUGNO
|
8.7 | IC50 | 2 | — | |
HCQLBVFQRDJJBA
|
8.7 | IC50 | 2 | — | |
HYIYVIBSZMQMHM
|
8.7 | IC50 | 2 | — | |
IQXLYQBMEPTZEO
|
8.7 | IC50 | 2 | — | |
IWBBYVKTABCSRE
|
8.7 | IC50 | 2 | — | |
JBIBZGLAWQVJLO
|
8.7 | IC50 | 2 | — | |
JFUYUTORRPOVER
|
8.7 | IC50 | 2 | — | |
JHRQFZCYSGOWTE
|
8.7 | IC50 | 2 | — | |
JIZCHNWVSOZUFN
|
8.7 | IC50 | 2 | — | |
KLHILMPJQMZZJF
|
8.7 | IC50 | 2 | — | |
KVGPKGSJVMLXCH
|
8.7 | IC50 | 2 | — | |
KVPAUWKFPNGRSX
|
8.7 | IC50 | 2 | — | |
KXMGCCQLOUJEHK
|
8.7 | IC50 | 2 | — | |
KZGHGHDFVIZCGE
|
8.7 | IC50 | 2 | — | |
LECCRWPQHHHXEG
|
8.7 | Kd | 2 | — | |
LGRWFIKZGOVIHT
|
8.7 | IC50 | 2 | — | |
LWDVYKMOIBCPGL
|
8.7 | IC50 | 2 | — |