Target Details
| UniProt AC | Q07889 |
|---|---|
| Gene Symbol | SOS1 |
| Protein Name | Son of sevenless homolog 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00617 (RasGEF) PF00618 (RasGEF_N) PF00621 (RhoGEF) PF22697 (SOS1_NGEF_PH) |
Summary
- Multi-target molecules 766
- Clinical molecules 0
- Avg pChEMBL 8.12
KEGG Pathways (48)
- Acute myeloid leukemia
- Alcoholism
- B cell receptor signaling pathway
- Breast cancer
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Choline metabolism in cancer
- Chronic myeloid leukemia
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Estrogen signaling pathway
- Fc epsilon RI signaling pathway
- Focal adhesion
- FoxO signaling pathway
- Gap junction
- Gastric cancer
- Glioma
- GnRH signaling pathway
- Growth hormone synthesis, secretion and action
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- JAK-STAT signaling pathway
- MAPK signaling pathway
- MicroRNAs in cancer
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prolactin signaling pathway
- Prostate cancer
- Proteoglycans in cancer
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Relaxin signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
- Thermogenesis
- mTOR signaling pathway
Associated Diseases (3)
Active Molecules (766)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LVXZSEGYCAIVFJ
|
7.9 | IC50 | 2 | — | |
MLMCEKGXKQSHLV
|
7.9 | IC50 | 2 | — | |
OPWSDOPRIRMMJL
|
7.9 | IC50 | 2 | — | |
POZGXECZBAYTIO
|
7.9 | Kd | 2 | — | |
SZFSFOIJHVKHDW
|
7.9 | IC50 | 2 | — | |
WOJDVMNKWBVECE
|
7.9 | IC50 | 2 | — | |
WQLRMMJDBZMQBG
|
7.9 | IC50 | 2 | — | |
XLCXNTXRPJRWRW
|
7.9 | IC50 | 2 | — | |
YEUMTULSGFNZHE
|
7.9 | IC50 | 2 | — | |
ZGPXGUPCJXHCGG
|
7.9 | IC50 | 2 | — | |
ARWFFXGRORNNNM
|
7.9 | IC50 | 2 | — | |
DOQLEUCLDNIOLK
|
7.9 | Kd | 2 | — | |
AMJPASDPTHFZEA
|
7.9 | Kd | 2 | — | |
ATAONWOPYHSDPU
|
7.9 | Kd | 2 | — | |
BSXKMLXPDHSEMN
|
7.9 | IC50 | 2 | — | |
CKBASITYRGBUED
|
7.9 | IC50 | 2 | — | |
FELOZWGBLKXDTI
|
7.9 | Kd | 2 | — | |
GPWBQBGVBKHNHI
|
7.9 | Kd | 2 | — | |
HDWBMTGSYRWLBC
|
7.9 | IC50 | 2 | — | |
HENSSECZGIFNLJ
|
7.9 | IC50 | 2 | — | |
HLRZUCSGYSFJQJ
|
7.9 | IC50 | 2 | — | |
JKFNRQAYTHLNLD
|
7.9 | IC50 | 2 | — | |
LIMYCUZQDBBHMZ
|
7.9 | IC50 | 2 | — | |
MMWORYFMOALMCV
|
7.9 | IC50 | 2 | — | |
MUUYFRSBNMFFTH
|
7.9 | IC50 | 2 | — | |
NHBDZIVLGPMXJY
|
7.9 | IC50 | 2 | — | |
QZBNZZWAPHPHNF
|
7.9 | IC50 | 2 | — | |
RCRCRSRUXXJNEG
|
7.9 | IC50 | 2 | — | |
RPDJLOLIEXXEJU
|
7.9 | IC50 | 2 | — | |
MFHBJGXWJWBFAM
|
7.9 | Kd | 2 | — | |
SXJFIJVXCQMDQK
|
7.9 | IC50 | 2 | — | |
HQRZAUXRRCRFEJ
|
7.9 | IC50 | 2 | — | |
ZVRJLGIVSIILRA
|
7.9 | IC50 | 2 | — | |
KILRSBNGOIDKAX
|
7.9 | IC50 | 2 | — | |
RSEWFMXCMHFDMS
|
7.9 | IC50 | 2 | — | |
AKXCPLJSAXYOGM
|
7.8 | IC50 | 2 | — | |
MYOMQNUICMUCPA
|
7.8 | IC50 | 2 | — | |
QJKBYBALCLEPGU
|
7.8 | IC50 | 2 | — | |
STATWBMSNVVOBM
|
7.8 | IC50 | 2 | — | |
VPEADMOUKUEMFK
|
7.8 | Kd | 2 | — | |
WKOUTBPOTLMIOM
|
7.8 | IC50 | 2 | — | |
XUWFDNOAJZOILL
|
7.8 | IC50 | 2 | — | |
OJKWQOQTOTXMEL
|
7.8 | IC50 | 2 | — | |
QUANGCDVTQSWAW
|
7.8 | IC50 | 2 | — | |
VLKMHSRFELLNSM
|
7.8 | IC50 | 2 | — | |
BSCTWHRUSVFZKE
|
7.8 | Kd | 2 | — | |
FHUPYSDNLIRUTO
|
7.8 | IC50 | 2 | — | |
GEHNCGXAFODUMD
|
7.8 | IC50 | 2 | — | |
IPRJZYPTRGEBHP
|
7.8 | IC50 | 2 | — | |
JTGAKPQYAUSICP
|
7.8 | Kd | 2 | — |