Target Details
| UniProt AC | Q07002 |
|---|---|
| Gene Symbol | CDK18 |
| Protein Name | Cyclin-dependent kinase 18 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 15
- Clinical molecules 4
- Avg pChEMBL 6.83
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OVPNQJVDAFNBDN
|
7.8 | Kd | 44 | Yes | |
JRNJNYBQQYBCLE
|
7.7 | Kd | 40 | Yes | |
OUSFTKFNBAZUKL
|
7.4 | Kd | 58 | Yes | |
ODPGGGTTYSGTGO
|
7.3 | Kd | 153 | — | |
AYCPARAPKDAOEN
|
7.2 | Kd | 73 | — | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
RPGZQOOZHIEPJW
|
7.0 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.0 | Kd | 18 | — | |
CXQHYVUVSFXTMY
|
6.6 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.6 | Kd | 149 | — | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 213 | — | |
XZXHXSATPCNXJR
|
6.3 | Kd | 165 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |