Target Details
| UniProt AC | Q06418 |
|---|---|
| Gene Symbol | TYRO3 |
| Protein Name | Tyrosine-protein kinase receptor TYRO3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF07679 (I-set) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 938
- Clinical molecules 16
- Avg pChEMBL 6.96
KEGG Pathways (2)
Active Molecules (938)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZSPYZKJALVPWOV
|
7.3 | IC50 | 2 | — | |
ZVGRBNITRNLZNZ
|
7.3 | IC50 | 2 | — | |
ZYCWFLSNKRWWQH
|
7.3 | IC50 | 2 | — | |
AGYRCBTVZCTMOP
|
7.2 | IC50 | 3 | — | |
IKENQUDOTQBCJH
|
7.2 | Kd | 18 | — | |
JJXRAZVLEQHSOL
|
7.2 | IC50 | 4 | — | |
VEFDEIILCRXHNC
|
7.2 | IC50 | 4 | — | |
WQIPRNUEYVQWKW
|
7.2 | IC50 | 2 | — | |
KAAPXWSYROPAEL
|
7.2 | IC50 | 4 | — | |
ORJFNGOUYHBFPE
|
7.2 | IC50 | 4 | — | |
FEXRSRXFBIRFMY
|
7.2 | IC50 | 4 | — | |
UBPYILGKFZZVDX
|
7.2 | Kd | 130 | Yes | |
WQLWLOMHWYQNFN
|
7.2 | IC50 | 4 | — | |
WZSUDZDKYJWJPS
|
7.2 | IC50 | 4 | — | |
HQMSWMADUGUYFF
|
7.2 | IC50 | 4 | — | |
UEIRKXUBXCSHJE
|
7.2 | Ki | 19 | — | |
WPHKIQPVPYJNAX
|
7.2 | Ki | 81 | — | |
GFIIPWSSHMVXHK
|
7.2 | IC50 | 4 | — | |
FXPKSABYJKCHOV
|
7.2 | IC50 | 4 | — | |
UEMPFKOYBHCUIG
|
7.2 | IC50 | 4 | — | |
ICAQVATUJCMIBT
|
7.2 | IC50 | 4 | — | |
NLXWFBBYANWXPR
|
7.2 | IC50 | 4 | — | |
JHLDSSUQVZCRDO
|
7.2 | IC50 | 3 | — | |
YWILRIPPYUJHMX
|
7.2 | IC50 | 4 | — | |
VWCZORWQNKCYGE
|
7.1 | IC50 | 17 | — | |
APPUYFNVFFWYFM
|
7.1 | IC50 | 4 | — | |
GPXJRVLKUZJOES
|
7.1 | IC50 | 3 | — | |
JZBDNDJNPAVSSE
|
7.1 | IC50 | 3 | — | |
MAIZEWVIGRBICN
|
7.1 | IC50 | 4 | — | |
RADSRRYRWZKEEW
|
7.1 | IC50 | 4 | — | |
MQWWFFUKPGKZQF
|
7.1 | IC50 | 3 | — | |
MXSXJVUUCUTMAN
|
7.1 | IC50 | 3 | — | |
VKBFHTIUXUCYRQ
|
7.1 | Ki | 66 | — | |
JGIUBJWBTUOQHP
|
7.1 | IC50 | 4 | — | |
JNYMZWUOQWXOII
|
7.1 | IC50 | 3 | — | |
PWOIRDUWFWWFMT
|
7.1 | IC50 | 4 | — | |
HTMNAROLUQALML
|
7.1 | IC50 | 4 | — | |
MXFGPNMMPZLQTR
|
7.1 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
7.1 | Kd | 147 | Yes | |
MIYIUVBGBPRNLG
|
7.1 | IC50 | 4 | — | |
WVXNSAVVKYZVOE
|
7.1 | IC50 | 92 | — | |
YVAPXKWBCBCTDS
|
7.1 | IC50 | 3 | — | |
YYTVUKVXIKXZNG
|
7.0 | IC50 | 4 | — | |
DGRCFAYRKDYEMX
|
7.0 | IC50 | 7 | — | |
XYASHXPUZJDWIO
|
7.0 | IC50 | 7 | — | |
BBJHTTNJKZUZCD
|
7.0 | IC50 | 4 | — | |
BONBXBPLENOTTM
|
7.0 | IC50 | 3 | — | |
KJLMCBXHAQXCDZ
|
7.0 | IC50 | 4 | — | |
UHTHHESEBZOYNR
|
7.0 | Kd | 66 | Yes | |
VPDVHIDCAMWQER
|
7.0 | IC50 | 4 | — |