Target Details
| UniProt AC | Q06278 |
|---|---|
| Gene Symbol | AOX1 |
| Protein Name | Aldehyde oxidase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01315 (Ald_Xan_dh_C) PF03450 (CO_deh_flav_C) PF00941 (FAD_binding_5) PF00111 (Fer2) PF01799 (Fer2_2) PF02738 (MoCoBD_1) PF20256 (MoCoBD_2) |
Summary
- Multi-target molecules 7
- Clinical molecules 4
- Avg pChEMBL 6.98
KEGG Pathways (9)
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GZUITABIAKMVPG
|
8.8 | Ki | 22 | Yes | |
RGCVKNLCSQQDEP
|
7.5 | IC50 | 16 | — | |
VOXZDWNPVJITMN
|
7.1 | IC50 | 8 | — | |
TZBJGXHYKVUXJN
|
6.5 | IC50 | 12 | Yes | |
BFPYWIDHMRZLRN
|
6.4 | IC50 | 10 | — | |
RGLYKWWBQGJZGM
|
6.3 | IC50 | 8 | Yes | |
ZPEIMTDSQAKGNT
|
6.2 | IC50 | 35 | Yes |