Target Details
| UniProt AC | Q06187 |
|---|---|
| Gene Symbol | BTK |
| Protein Name | Tyrosine-protein kinase BTK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,619
- Clinical molecules 27
- Avg pChEMBL 7.81
KEGG Pathways (7)
Associated Diseases (3)
Active Molecules (1,619)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YMFKLMVUBGVUPG
|
9.3 | IC50 | 2 | — | |
YMFKLMVUBGVUPG
|
9.3 | IC50 | 2 | — | |
FHNCSRKSWPZETL
|
9.3 | IC50 | 4 | — | |
MNDLPZPZVIEBFF
|
9.3 | IC50 | 4 | — | |
OXOMWFOJARKFIY
|
9.3 | IC50 | 4 | — | |
RJARQSDFMBQVEH
|
9.3 | IC50 | 4 | — | |
ZKYNGODFNLAFMZ
|
9.3 | IC50 | 2 | — | |
LCYSSHSIKSARGO
|
9.3 | IC50 | 19 | — | |
MNUZXSBABPJWOR
|
9.3 | IC50 | 2 | — | |
PZWSKESWDIFAFK
|
9.3 | IC50 | 9 | — | |
SRSQULBCTWSVKL
|
9.3 | IC50 | 15 | — | |
UNSFWPUQRXYWKE
|
9.3 | IC50 | 4 | — | |
ZUXIOCJCONDJBE
|
9.3 | IC50 | 4 | — | |
BEKXRKQECXXKGJ
|
9.3 | IC50 | 2 | — | |
JHUWBOAVDAIILQ
|
9.3 | IC50 | 2 | — | |
UBWXSCATULGCSA
|
9.3 | IC50 | 4 | — | |
IRBVGTPPFBYDKX
|
9.3 | IC50 | 9 | — | |
LZOYRTMQLOFTSF
|
9.2 | IC50 | 4 | — | |
MBTQEKOQTVSXTJ
|
9.2 | IC50 | 2 | — | |
AVNRKIYQTBXHEU
|
9.2 | IC50 | 2 | — | |
CQYOCHGVYYCAJH
|
9.2 | IC50 | 4 | — | |
PKGJEJSOPQZJNR
|
9.2 | IC50 | 2 | — | |
RXBBNYOZZYEKJZ
|
9.2 | IC50 | 4 | — | |
RLAPDPXPNISUNN
|
9.2 | IC50 | 2 | — | |
VMDYPRANJKKHLD
|
9.2 | IC50 | 2 | — | |
CATGYHXLDRQPGZ
|
9.2 | IC50 | 3 | — | |
FUZSHLVNKZZEKR
|
9.2 | IC50 | 16 | — | |
KOQJXUXLQGQJDF
|
9.2 | IC50 | 4 | — | |
NBNBOYCGFBMTJH
|
9.2 | IC50 | 2 | — | |
UKCXKMIKWBUVSF
|
9.2 | IC50 | 2 | — | |
ZTQVREOZSGAIKH
|
9.2 | IC50 | 2 | — | |
QRYWETQFXDSLKP
|
9.2 | IC50 | 4 | — | |
YEQGARBJDLREPV
|
9.2 | IC50 | 4 | — | |
MSOXGTBOMYQLRK
|
9.2 | IC50 | 4 | — | |
ROUNLVFMMJKGCE
|
9.2 | IC50 | 2 | — | |
VAHPHFUKSVSWLN
|
9.2 | IC50 | 2 | — | |
WPFZWTKQXNTKQJ
|
9.2 | IC50 | 4 | — | |
ZXGCNNKDPNECIS
|
9.2 | IC50 | 4 | — | |
GFXJEHXKSRGUJJ
|
9.2 | IC50 | 4 | — | |
NHMAKMLWAUSTMS
|
9.2 | IC50 | 4 | — | |
BIRLBQULISTSMZ
|
9.2 | IC50 | 4 | — | |
DYOZBZNVCJZQTG
|
9.2 | IC50 | 2 | — | |
PFZFZZIBHZGYGR
|
9.2 | IC50 | 4 | — | |
QNNJMWIVIVLSHC
|
9.2 | IC50 | 4 | — | |
MWNASUNUUFWMNK
|
9.2 | IC50 | 3 | — | |
SJYAVQZFEBVYGJ
|
9.2 | IC50 | 4 | — | |
CLKNHJDZJCCLAZ
|
9.2 | IC50 | 4 | — | |
NJQKXLPNGPRPBX
|
9.2 | IC50 | 2 | — | |
OILCFDXBRQHLMC
|
9.2 | IC50 | 2 | — | |
ABBSDUKZIMPCRZ
|
9.2 | IC50 | 2 | — |