Target Details
| UniProt AC | Q06124 |
|---|---|
| Gene Symbol | PTPN11 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00017 (SH2) PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 214
- Clinical molecules 1
- Avg pChEMBL 7.2
KEGG Pathways (21)
- Adipocytokine signaling pathway
- Axon guidance
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chronic myeloid leukemia
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Herpes simplex virus 1 infection
- IgSF CAM signaling
- Insulin resistance
- JAK-STAT signaling pathway
- Leukocyte transendothelial migration
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Pathogenic Escherichia coli infection
- Phospholipase D signaling pathway
- Proteoglycans in cancer
- Ras signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
Associated Diseases (6)
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VNPAVLDSIONFMU
|
6.1 | IC50 | 2 | — | |
PIIJGIPNQPGCJA
|
6.1 | IC50 | 2 | — | |
CPGHULPHYSDBNR
|
6.1 | IC50 | 2 | — | |
YSWVIGJDOZEAPY
|
6.1 | IC50 | 2 | — | |
IIZRLNOBXIGZFR
|
6.0 | IC50 | 3 | — | |
MLQBNUCBCXWMME
|
6.0 | IC50 | 2 | — | |
YMDXJDQSJVLAPR
|
6.0 | IC50 | 2 | — | |
AQNQKVLAOFOLOO
|
6.0 | IC50 | 2 | — | |
HZYUNIMXNROZHD
|
6.0 | IC50 | 2 | — | |
SXLQVLBGTXXABW
|
6.0 | IC50 | 2 | — | |
UCVNJKUCRRXAMU
|
6.0 | IC50 | 2 | — | |
ZIWJTYIFLVSYBO
|
6.0 | IC50 | 2 | — | |
ACZCNRCVPUGLCW
|
6.0 | IC50 | 2 | — | |
LWULRPYIMPIYQD
|
6.0 | IC50 | 2 | — |