Target Details
| UniProt AC | Q06124 |
|---|---|
| Gene Symbol | PTPN11 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00017 (SH2) PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 214
- Clinical molecules 1
- Avg pChEMBL 7.2
KEGG Pathways (21)
- Adipocytokine signaling pathway
- Axon guidance
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chronic myeloid leukemia
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Herpes simplex virus 1 infection
- IgSF CAM signaling
- Insulin resistance
- JAK-STAT signaling pathway
- Leukocyte transendothelial migration
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Pathogenic Escherichia coli infection
- Phospholipase D signaling pathway
- Proteoglycans in cancer
- Ras signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
Associated Diseases (6)
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CNWPAKCFVFDYQN
|
7.1 | IC50 | 3 | — | |
XEMDEEZOTNHZCZ
|
7.1 | IC50 | 2 | — | |
SIKKESBUGBWVRF
|
7.1 | IC50 | 3 | — | |
NQCYZSVEYSASFG
|
7.1 | IC50 | 2 | — | |
LSGOVYNHVSXFFJ
|
7.1 | IC50 | 4 | — | |
JPGLGZVWXAXTCH
|
7.1 | IC50 | 2 | — | |
QJIIXGVBODDUGN
|
7.1 | IC50 | 2 | — | |
ZNUFCVFEZWEKRQ
|
7.0 | IC50 | 2 | — | |
MCCSBHCNGJMJAW
|
7.0 | IC50 | 3 | — | |
LQDXCHQGEHUKDL
|
7.0 | IC50 | 12 | — | |
RIBDKTGIOVNZBA
|
7.0 | IC50 | 2 | — | |
CUTMOOSDQSRDHK
|
7.0 | IC50 | 2 | — | |
GSOVNVHPLHWGDA
|
7.0 | IC50 | 3 | — | |
WCBNKFWTMBJQOT
|
7.0 | IC50 | 2 | — | |
ZLEYPUJZZGTSLW
|
7.0 | IC50 | 3 | — | |
IPILYXRPIMXNGK
|
7.0 | IC50 | 3 | — | |
YCRNZPYPOFXDCB
|
7.0 | IC50 | 2 | — | |
CDVCKXMGBCDTDW
|
6.9 | IC50 | 2 | — | |
CKEXLFZOLNCINM
|
6.9 | IC50 | 2 | — | |
HWNCRAHYJRQMMV
|
6.9 | IC50 | 2 | — | |
XLKDUTBYZJONNW
|
6.9 | IC50 | 2 | — | |
ZBPQOUUAEZWTQS
|
6.9 | IC50 | 2 | — | |
SJLQMBIPYINRMF
|
6.9 | IC50 | 2 | — | |
DEVINZPHNDARNY
|
6.8 | IC50 | 2 | — | |
IEUPVYYCTFCLTF
|
6.8 | IC50 | 2 | — | |
MGGGLWKKMYVXPD
|
6.8 | IC50 | 2 | — | |
CTAYFFLEYDVMQX
|
6.8 | IC50 | 2 | — | |
FKWSHGCXJGIGPU
|
6.8 | IC50 | 2 | — | |
LJXXZVLIMZSWLE
|
6.8 | IC50 | 2 | — | |
POYNJTHRRZRCMC
|
6.8 | IC50 | 2 | — | |
BHDQDMSKLZFAOP
|
6.8 | IC50 | 2 | — | |
RGCGBFIARQENML
|
6.8 | IC50 | 3 | — | |
JCYHCBVXAFUBRD
|
6.8 | IC50 | 2 | — | |
BAPWXYXPJRISAE
|
6.7 | IC50 | 2 | — | |
QUZYGWHMIMOARM
|
6.7 | IC50 | 2 | — | |
GBRTUCQWCTVZDK
|
6.7 | IC50 | 2 | — | |
LRKKMCZEIFELNN
|
6.7 | IC50 | 2 | — | |
WILZWITYAQZYKV
|
6.7 | IC50 | 2 | — | |
CCNVAVIEHMNTEE
|
6.7 | IC50 | 2 | — | |
FNJXZHWYKAGWOU
|
6.7 | IC50 | 3 | — | |
QKNOZCPUZKQEHX
|
6.7 | IC50 | 2 | — | |
UWWTYAGOTZWMOX
|
6.7 | IC50 | 2 | — | |
RNFXSRZAAHHCDB
|
6.7 | IC50 | 2 | — | |
MFKUFVTVUGLDLG
|
6.7 | IC50 | 2 | — | |
RIBDKTGIOVNZBA
|
6.7 | IC50 | 2 | — | |
MSUDNEADKNPNRJ
|
6.7 | IC50 | 2 | — | |
ZSNQCYQABMACIK
|
6.6 | IC50 | 2 | — | |
RMZKUOVRTWVBDH
|
6.6 | IC50 | 3 | — | |
MJHCUHULQWWLSQ
|
6.5 | IC50 | 3 | — | |
ZXABOENZJMEVQC
|
6.5 | IC50 | 2 | — |