Target Details
| UniProt AC | Q06124 |
|---|---|
| Gene Symbol | PTPN11 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00017 (SH2) PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 214
- Clinical molecules 1
- Avg pChEMBL 7.2
KEGG Pathways (21)
- Adipocytokine signaling pathway
- Axon guidance
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chronic myeloid leukemia
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Herpes simplex virus 1 infection
- IgSF CAM signaling
- Insulin resistance
- JAK-STAT signaling pathway
- Leukocyte transendothelial migration
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Pathogenic Escherichia coli infection
- Phospholipase D signaling pathway
- Proteoglycans in cancer
- Ras signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
Associated Diseases (6)
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MAUDHCQAMRNUAG
|
8.1 | IC50 | 3 | — | |
VOHJNJREZGGBHF
|
8.1 | IC50 | 2 | — | |
WUANGOCWSCYKOJ
|
8.1 | IC50 | 2 | — | |
PVRKROKBYOCJNE
|
8.0 | IC50 | 2 | — | |
AZCZIDVDHVGBES
|
8.0 | IC50 | 2 | — | |
IGSGJEYNZCLOAG
|
8.0 | IC50 | 2 | — | |
MFAPJVDHXWVGIU
|
8.0 | IC50 | 2 | — | |
WMXJUWADUGXUIO
|
8.0 | IC50 | 2 | — | |
MFAPJVDHXWVGIU
|
8.0 | IC50 | 2 | — | |
RCRWPBKEEYEBDV
|
8.0 | IC50 | 2 | — | |
APCVETMNHFLTTE
|
7.9 | IC50 | 2 | — | |
JNXHZAMNUTXZFA
|
7.9 | IC50 | 2 | — | |
FQXAGRFLFFENPB
|
7.9 | IC50 | 2 | — | |
VXXRNTLTIAEVNE
|
7.9 | IC50 | 2 | — | |
JNXHZAMNUTXZFA
|
7.8 | IC50 | 2 | — | |
AKZKUGUQZMUCJC
|
7.8 | IC50 | 2 | — | |
QOIJTELOSKKPNI
|
7.8 | IC50 | 3 | — | |
UYHZBRZIVCBSMC
|
7.8 | IC50 | 12 | — | |
VKQWFSBYDFOYLI
|
7.7 | IC50 | 2 | — | |
CJJLAWVMRURPRM
|
7.7 | IC50 | 12 | — | |
JZIVZJLOIQOPCM
|
7.7 | IC50 | 2 | — | |
NGJFCIYVFFUILZ
|
7.6 | IC50 | 2 | — | |
LCDKHVMBHOTRTK
|
7.6 | IC50 | 3 | — | |
AJNXRYLTABACFI
|
7.5 | IC50 | 2 | — | |
XNIYTWAJXXHCLG
|
7.5 | IC50 | 3 | — | |
AWCUGJTVKPBYHS
|
7.5 | IC50 | 2 | — | |
CQHDXEWKDCKMHF
|
7.5 | IC50 | 6 | — | |
FCVULWLGEGJWIH
|
7.5 | IC50 | 3 | — | |
XETBCFSFVAVHSU
|
7.5 | IC50 | 3 | — | |
LKXGJCAIIDCTPQ
|
7.5 | IC50 | 3 | — | |
UFDJDSLGPDGBBZ
|
7.5 | IC50 | 2 | — | |
YPLHAXDRIIJALD
|
7.5 | IC50 | 3 | — | |
BWQAQACZKDLJAW
|
7.4 | IC50 | 3 | — | |
FBFPWPVDVUHEKP
|
7.4 | IC50 | 2 | — | |
RFYWVDVFMZNBBB
|
7.4 | IC50 | 3 | — | |
PVBNSTQJFPASQY
|
7.4 | IC50 | 2 | — | |
JTSYRPMZSWPUHL
|
7.4 | IC50 | 2 | — | |
CLVKLHYQSCMHQX
|
7.3 | IC50 | 3 | — | |
XSVLQUPXLDCENB
|
7.3 | IC50 | 3 | — | |
AMADCPJVPLUGQO
|
7.3 | IC50 | 2 | — | |
KOFLHKSEIMZJFM
|
7.3 | IC50 | 2 | — | |
URLQCJFKEIJEMW
|
7.3 | IC50 | 3 | — | |
ZJCWKDUZVMTXRX
|
7.2 | IC50 | 3 | — | |
BBHOXURWAZHPOP
|
7.2 | IC50 | 3 | — | |
GYFNRQGETQTKEM
|
7.2 | IC50 | 3 | — | |
LANVDWAEBRQKDI
|
7.2 | IC50 | 3 | — | |
FZVDMPMSYYNXLJ
|
7.2 | IC50 | 3 | — | |
HZNWRFAFSDEIMQ
|
7.2 | IC50 | 3 | — | |
COZSKBGMNPMNET
|
7.2 | IC50 | 3 | — | |
YGUFCDOEKKVKJK
|
7.2 | IC50 | 4 | — |