Target Details
| UniProt AC | Q06124 |
|---|---|
| Gene Symbol | PTPN11 |
| Protein Name | Tyrosine-protein phosphatase non-receptor type 11 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00017 (SH2) PF00102 (Y_phosphatase) |
Summary
- Multi-target molecules 214
- Clinical molecules 1
- Avg pChEMBL 7.2
KEGG Pathways (21)
- Adipocytokine signaling pathway
- Axon guidance
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chronic myeloid leukemia
- Efferocytosis
- Epithelial cell signaling in Helicobacter pylori infection
- Herpes simplex virus 1 infection
- IgSF CAM signaling
- Insulin resistance
- JAK-STAT signaling pathway
- Leukocyte transendothelial migration
- Natural killer cell mediated cytotoxicity
- Neurotrophin signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Pathogenic Escherichia coli infection
- Phospholipase D signaling pathway
- Proteoglycans in cancer
- Ras signaling pathway
- Renal cell carcinoma
- T cell receptor signaling pathway
Associated Diseases (6)
Active Molecules (214)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QZVSNMBRLYUYQI
|
9.0 | IC50 | 2 | — | |
WRHXPUBAPLIIDL
|
9.0 | IC50 | 2 | — | |
IKUYEYLZXGGCRD
|
8.8 | IC50 | 3 | — | |
OKLKDPLBWBNFAN
|
8.7 | IC50 | 2 | — | |
PGMVMBOOWXFMHK
|
8.6 | IC50 | 2 | — | |
AOEKGRJBTLUHAE
|
8.6 | IC50 | 2 | — | |
BDJJZYXDJQVPIV
|
8.5 | IC50 | 2 | — | |
GAXRSLAUXVLRCM
|
8.5 | IC50 | 2 | — | |
IPUGYWBSZWTMTM
|
8.5 | IC50 | 2 | — | |
XVLBIZWRRODPHP
|
8.5 | IC50 | 2 | — | |
JXFVWCLYSJQTHY
|
8.5 | IC50 | 2 | — | |
YQNLXVRRERHINB
|
8.5 | IC50 | 2 | — | |
BQSWGKBMQOWIJV
|
8.4 | IC50 | 2 | — | |
BQSWGKBMQOWIJV
|
8.4 | IC50 | 2 | — | |
PAKOJENWJZRWER
|
8.4 | IC50 | 2 | — | |
AYKLDGZOGDEWOB
|
8.4 | IC50 | 2 | — | |
CHLHMGGBVMLLOD
|
8.4 | IC50 | 2 | — | |
IHIKNAQWTTVBFU
|
8.4 | IC50 | 2 | — | |
JBTYRLRPDPSWAY
|
8.4 | IC50 | 2 | — | |
AOEKGRJBTLUHAE
|
8.4 | IC50 | 2 | — | |
YQNLXVRRERHINB
|
8.4 | IC50 | 2 | — | |
ZDEBEWQYXJZQRS
|
8.4 | IC50 | 12 | — | |
DADBALWTMMVAKC
|
8.3 | IC50 | 12 | — | |
WFRALCQQPKDCIU
|
8.3 | IC50 | 2 | — | |
CVCSGWXUXZEZBE
|
8.3 | IC50 | 2 | — | |
QCNFQPYDUXRNEN
|
8.3 | IC50 | 2 | — | |
ZNGLHHGXOQHVRP
|
8.3 | IC50 | 2 | — | |
ZVBSVBHUEYAOGL
|
8.3 | IC50 | 2 | — | |
GJJQUHQSJVEHNN
|
8.3 | IC50 | 2 | — | |
APBRCMWEQMUMHX
|
8.2 | IC50 | 12 | — | |
GHBLKRGJLJRKBB
|
8.2 | IC50 | 2 | — | |
ARCKFDMKZIEWRQ
|
8.2 | IC50 | 2 | — | |
GZTRITRCVPNXCC
|
8.2 | IC50 | 2 | — | |
LJZPRAULMDMOHN
|
8.2 | IC50 | 2 | — | |
BDJJZYXDJQVPIV
|
8.2 | IC50 | 2 | — | |
FIDXYKFRGLNFAF
|
8.2 | IC50 | 2 | — | |
GPMCVSXTDRZSLO
|
8.2 | IC50 | 2 | — | |
NYPXMXPABWAYNI
|
8.2 | IC50 | 2 | — | |
QQGWBWWGXPNCEH
|
8.2 | IC50 | 2 | — | |
WRYBCDHGKKPMKW
|
8.2 | IC50 | 2 | — | |
OPEZBSGNVCPIIK
|
8.2 | IC50 | 2 | — | |
SXLOCFFGRYJKJH
|
8.2 | IC50 | 2 | — | |
JJTYMCPMKUFMGA
|
8.1 | IC50 | 2 | — | |
HNONCNSCKGVMAR
|
8.1 | IC50 | 2 | — | |
AZCZIDVDHVGBES
|
8.1 | IC50 | 2 | — | |
GPMCVSXTDRZSLO
|
8.1 | IC50 | 2 | — | |
IGSGJEYNZCLOAG
|
8.1 | IC50 | 2 | — | |
JZIVZJLOIQOPCM
|
8.1 | IC50 | 2 | — | |
NNHSFUJHEDZYGF
|
8.1 | IC50 | 2 | — | |
OIBRHNUGJRDNJV
|
8.1 | IC50 | 2 | — |