Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YOSWNJPQIDFLAM
|
6.9 | Ki | 3 | — | |
GTWLYEVXNCSGBU
|
6.9 | IC50 | 3 | Yes | |
KEUYDWVTHJQHIH
|
6.9 | IC50 | 3 | Yes | |
KEUYDWVTHJQHIH
|
6.9 | IC50 | 3 | Yes | |
NDPCMXFATSKLHE
|
6.9 | IC50 | 3 | Yes | |
PDSONWYECZHBAE
|
6.9 | Ki | 2 | — | |
VBWJOMJNVZBWBF
|
6.9 | IC50 | 3 | Yes | |
XHHYVFRQYUOODP
|
6.9 | IC50 | 3 | Yes | |
XPKKUXKJOCVNEJ
|
6.9 | IC50 | 3 | Yes | |
DVMQYKHCZLPSAP
|
6.9 | IC50 | 5 | — | |
BMGQWWVMWDBQGC
|
6.9 | IC50 | 91 | Yes | |
JZTOUVBEZONDKA
|
6.9 | Ki | 80 | — | |
OGJTZCZJWZSZBT
|
6.9 | IC50 | 12 | Yes | |
OUJZYQBEFNDJQN
|
6.9 | Ki | 71 | — | |
TVEREFRWBLRPPJ
|
6.9 | Ki | 15 | — | |
ZCXXFPLQFFRMPN
|
6.9 | Ki | 12 | — | |
BSSIEJNTKGYHRD
|
6.9 | Ki | 2 | — | |
CZYUVYJLWVYZNM
|
6.9 | Ki | 2 | — | |
DWKWEQIKOVHMQW
|
6.9 | IC50 | 3 | — | |
IYKCWOIZNVHUMI
|
6.9 | Ki | 5 | Yes | |
KDIRIFZBLUSLJU
|
6.9 | Ki | 5 | — | |
LPIJVXOQOOJCRR
|
6.9 | IC50 | 3 | Yes | |
UOHOMVNTUXAPFC
|
6.9 | IC50 | 3 | Yes | |
VWHZWDRIMLETBG
|
6.9 | IC50 | 12 | Yes | |
ZZARJEJPLRJJQO
|
6.9 | IC50 | 3 | Yes | |
JKLDSNMMVPQIRH
|
6.9 | Ki | 2 | — | |
WVLMGPVSSPPHSJ
|
6.9 | Ki | 2 | — | |
FDCMEPRGSNNHNX
|
6.9 | Ki | 4 | — | |
WUWJDRGPTHRZQB
|
6.9 | IC50 | 3 | Yes | |
DDVKURVSLBGSOS
|
6.8 | IC50 | 3 | Yes | |
DRCBMJUPXHWGMN
|
6.8 | IC50 | 15 | Yes | |
IJYPXTWDRNLKMU
|
6.8 | IC50 | 3 | Yes | |
SDZRYLPROGBZMB
|
6.8 | IC50 | 8 | — | |
WXEYWIXOJDRUIB
|
6.8 | IC50 | 3 | Yes | |
FAQJIZKBJRQPIA
|
6.8 | IC50 | 3 | Yes | |
MVQGUYKZTHVOEH
|
6.8 | Ki | 8 | Yes | |
FNLZNOBAYWDBFQ
|
6.8 | Ki | 2 | — | |
JWVXPOMGWPAEAJ
|
6.8 | IC50 | 10 | Yes | |
PXONMVAMARNSJO
|
6.8 | Ki | 4 | — | |
QNULKTUETCUJKC
|
6.8 | IC50 | 14 | Yes | |
QXQGSOMQKZFIRY
|
6.8 | IC50 | 10 | — | |
SWZXKBUPFISEFY
|
6.8 | IC50 | 3 | Yes | |
UYICUHDKBPIZCB
|
6.8 | IC50 | 3 | Yes | |
YUZANCJQMKLODH
|
6.8 | IC50 | 3 | Yes | |
ASDRIDGWWRNUHE
|
6.8 | IC50 | 3 | Yes | |
CZIVUSJISIAXJB
|
6.8 | IC50 | 18 | — | |
CGIUQTLYFGDGTD
|
6.8 | IC50 | 4 | — | |
DWTNLZZEPSCAIH
|
6.8 | Ki | 25 | — | |
FXQWJULRETZHHW
|
6.8 | Ki | 14 | — | |
NLJJDZMBYLCWHR
|
6.8 | IC50 | 2 | — |