Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKWRGMLRFOFLFQ
|
7.1 | IC50 | 3 | Yes | |
VMRZSNDAPJYPND
|
7.1 | IC50 | 3 | Yes | |
WPSBCJTXGDVGAZ
|
7.1 | IC50 | 5 | — | |
AGJAPEBQOOHERM
|
7.1 | IC50 | 4 | Yes | |
CNXKJMKQJSETCG
|
7.1 | Ki | 3 | — | |
AZHZQWZIQCSEHF
|
7.0 | IC50 | 3 | Yes | |
FYHDYXSOJZTOJN
|
7.0 | IC50 | 3 | — | |
FYHDYXSOJZTOJN
|
7.0 | IC50 | 4 | — | |
JKLDSNMMVPQIRH
|
7.0 | Ki | 2 | — | |
MDRQBBNTQCZOBR
|
7.0 | IC50 | 6 | — | |
MDRQBBNTQCZOBR
|
7.0 | IC50 | 6 | — | |
TXKSMXUHBNRXFZ
|
7.0 | IC50 | 2 | — | |
VBBJIIXIIXRQOK
|
7.0 | IC50 | 3 | — | |
VBBJIIXIIXRQOK
|
7.0 | IC50 | 3 | — | |
ZLGMCAODGHZKDH
|
7.0 | IC50 | 2 | — | |
BLYAGPCWZUKSNN
|
7.0 | IC50 | 6 | — | |
DLMIREIQJNSNMF
|
7.0 | Ki | 3 | — | |
OYPYXQXNEBSSGB
|
7.0 | Ki | 8 | Yes | |
JTUGJZFQRMCZQW
|
7.0 | IC50 | 3 | Yes | |
KIAJUGUFTMKTNB
|
7.0 | IC50 | 3 | Yes | |
NSFGGHWNWJTVMO
|
7.0 | IC50 | 5 | — | |
SXDPQGRNHSLZPC
|
7.0 | IC50 | 18 | — | |
UZHOUJWDVUELSD
|
7.0 | IC50 | 3 | Yes | |
XOTNYFMXYDWFEU
|
7.0 | IC50 | 3 | Yes | |
DNYURFSSJKXPTF
|
7.0 | IC50 | 3 | Yes | |
GJIHZDZOVHMYJS
|
7.0 | IC50 | 3 | Yes | |
HETWGNHMXYNQPB
|
7.0 | IC50 | 2 | — | |
MQCCJEYZKWZQHU
|
7.0 | IC50 | 15 | Yes | |
YSVVBGPTTSJYPA
|
7.0 | IC50 | 13 | Yes | |
QMYFYCSCELQGHP
|
7.0 | IC50 | 7 | Yes | |
ZQKCTEOSJBBWBB
|
7.0 | IC50 | 3 | Yes | |
KLTAXINXABHYMC
|
7.0 | IC50 | 5 | — | |
LOCWELCIOZHZHE
|
7.0 | Ki | 11 | — | |
PEZLAFKDOMGSEL
|
7.0 | IC50 | 4 | — | |
PEZLAFKDOMGSEL
|
7.0 | IC50 | 4 | — | |
PFAZIMNYEBJHOA
|
7.0 | IC50 | 12 | Yes | |
QMNJRUYPIVXCAT
|
7.0 | IC50 | 3 | Yes | |
RZHAEOSLBJVDFX
|
7.0 | IC50 | 5 | — | |
XRFOMFNAMTYCFF
|
7.0 | IC50 | 12 | Yes | |
YUAWUNMKPARPJD
|
7.0 | IC50 | 14 | Yes | |
ZRTWUBWXIGHVET
|
7.0 | Ki | 10 | — | |
JHLONFVVTLRHIZ
|
7.0 | IC50 | 4 | — | |
DQGXZJOMYLWAKM
|
7.0 | IC50 | 3 | Yes | |
KXRUTZLUYFIXDZ
|
7.0 | IC50 | 3 | Yes | |
MGQDMSJZRRHMFT
|
7.0 | IC50 | 6 | — | |
NIAJEEMQNUPFJB
|
7.0 | IC50 | 3 | Yes | |
REVNTLJVVFYWNE
|
7.0 | IC50 | 3 | Yes | |
MJVOZZPYOLLRCY
|
7.0 | Ki | 2 | — | |
BTFQHCKJTLZZRE
|
6.9 | IC50 | 3 | Yes | |
KOZFSFOOLUUIGY
|
6.9 | IC50 | 15 | Yes |