Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXZFDXZCJALHRF
|
7.2 | IC50 | 6 | — | |
IDMUMGBXJGYJTD
|
7.2 | Ki | 3 | — | |
ALLMHFJXFWBPDH
|
7.2 | IC50 | 3 | Yes | |
JHSOAROIYKSHKX
|
7.2 | IC50 | 3 | Yes | |
LCLDOTQNYVMPRQ
|
7.2 | IC50 | 3 | Yes | |
NMRUWPRCOQSHGH
|
7.2 | IC50 | 3 | Yes | |
WALDOGJQTYJBFG
|
7.2 | IC50 | 3 | Yes | |
XXIWRTOLXWAEJC
|
7.2 | IC50 | 13 | Yes | |
BVCPWHHJIAYYTM
|
7.2 | IC50 | 3 | Yes | |
FUMCKNCUEAQHCV
|
7.2 | Ki | 103 | — | |
JRVSFZKYQCETAH
|
7.2 | Ki | 19 | — | |
PFCUZXCHLYIMTJ
|
7.2 | Ki | 18 | — | |
TUBBFDZWFNUZLH
|
7.2 | IC50 | 12 | Yes | |
VLUGUCDUHZVABE
|
7.2 | IC50 | 6 | — | |
KRMLZRDHQHQPJW
|
7.2 | IC50 | 5 | Yes | |
NRUVICOXXLOXCB
|
7.2 | IC50 | 13 | Yes | |
ASUGUQWIHMTFJL
|
7.2 | Kd | 18 | — | |
MGLBGUZLARZAOR
|
7.2 | IC50 | 4 | — | |
MWKQDYOZWRAWMS
|
7.2 | IC50 | 3 | Yes | |
MXZMNMJBRPSOOG
|
7.2 | IC50 | 3 | Yes | |
PBWBADGNVJJHFC
|
7.2 | IC50 | 3 | Yes | |
RVIJQMOQZFCSHL
|
7.2 | Ki | 8 | Yes | |
MEAHLUNWZGONEH
|
7.2 | IC50 | 3 | Yes | |
MGMNDPRNDCWSMZ
|
7.2 | IC50 | 12 | Yes | |
PJGVITFBPVCDNT
|
7.2 | IC50 | 3 | Yes | |
HHLNVCKLKSYSJN
|
7.1 | IC50 | 3 | Yes | |
JSBPEIYUYLNLLN
|
7.1 | IC50 | 3 | Yes | |
FQUIZYRWNTVYLN
|
7.1 | IC50 | 3 | Yes | |
GRENHRYHWHSBLM
|
7.1 | IC50 | 12 | Yes | |
OFAWVNTWBAYIQM
|
7.1 | IC50 | 3 | Yes | |
MOJGUBLPDOMBJL
|
7.1 | IC50 | 3 | Yes | |
VEMLCWMDXJGJLI
|
7.1 | Ki | 8 | Yes | |
DKZYXHCYPUVGAF
|
7.1 | Kd | 112 | — | |
GLHNMQILKIFCNS
|
7.1 | Ki | 3 | — | |
HOWICUYRWBCICG
|
7.1 | IC50 | 6 | — | |
LGCKGDRUTNACTA
|
7.1 | IC50 | 11 | — | |
NXOILRDXHDPZAY
|
7.1 | IC50 | 2 | — | |
OFPFIAWWDTYSBZ
|
7.1 | Ki | 15 | Yes | |
OWRXHGAFWZFFCW
|
7.1 | Ki | 113 | — | |
RHLRPKGACJKWPF
|
7.1 | IC50 | 12 | Yes | |
GGQAEINRBKFRGZ
|
7.1 | IC50 | 15 | Yes | |
GZRXZIIXJPGKRW
|
7.1 | Ki | 2 | — | |
HAYBNIARWRGYIC
|
7.1 | IC50 | 3 | Yes | |
JWTNYYVEXFBGQI
|
7.1 | IC50 | 3 | Yes | |
MVYBDSJHHWQUEP
|
7.1 | IC50 | 4 | Yes | |
PEDXJGLVPJEZIK
|
7.1 | IC50 | 3 | Yes | |
NHDDTLMPCVOXFH
|
7.1 | IC50 | 16 | Yes | |
OBVZNBSDRAGXLG
|
7.1 | IC50 | 3 | Yes | |
FUOBGQKXJPZPSV
|
7.1 | IC50 | 3 | Yes | |
OHQBRPBJOMAGLO
|
7.1 | IC50 | 3 | Yes |