Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
7.4 | IC50 | 49 | Yes | |
JPINQKLMVKTGTL
|
7.4 | IC50 | 3 | Yes | |
JVSULVHQOCWQHQ
|
7.4 | IC50 | 3 | Yes | |
NTUVEMUMVHHACY
|
7.4 | IC50 | 12 | Yes | |
ZPKBYERIJJCKAI
|
7.4 | IC50 | 3 | Yes | |
KADSBMDSVAYXRE
|
7.4 | IC50 | 3 | Yes | |
OXPLGRNOXPCLEB
|
7.4 | IC50 | 3 | Yes | |
USYSUTGHQKSLCI
|
7.4 | IC50 | 3 | Yes | |
IIRWNGPLJQXWFJ
|
7.4 | Kd | 21 | — | |
SPKAGPPMKYJUPF
|
7.4 | IC50 | 3 | Yes | |
WNDOFCPEDZYDPL
|
7.4 | IC50 | 10 | — | |
CLENZPTUQALSKC
|
7.3 | IC50 | 3 | Yes | |
GFLGIZVUCFIBRB
|
7.3 | IC50 | 3 | Yes | |
KOZFSFOOLUUIGY
|
7.3 | IC50 | 88 | Yes | |
LBDMJMNVJZNONC
|
7.3 | IC50 | 3 | Yes | |
OLTHFAIHFDAJGG
|
7.3 | IC50 | 5 | Yes | |
WKZTVBCDQYBGBO
|
7.3 | IC50 | 16 | Yes | |
KRXPQEKAJKYQGS
|
7.3 | Ki | 5 | — | |
QEPARSUKSLKMMO
|
7.3 | IC50 | 7 | Yes | |
LUDKZCXHZJRUAZ
|
7.3 | Ki | 5 | — | |
CLQHLBAJBOQPRR
|
7.3 | IC50 | 3 | — | |
CSCOHEYTBLBQMG
|
7.3 | IC50 | 7 | Yes | |
GWJHMRBQEUHFOC
|
7.3 | Ki | 42 | — | |
JNXDDALKPXMKQB
|
7.3 | IC50 | 3 | Yes | |
KSITVHDHIJKJBG
|
7.3 | IC50 | 3 | — | |
KSITVHDHIJKJBG
|
7.3 | IC50 | 6 | — | |
MDHNNGDJYHAYKJ
|
7.3 | IC50 | 12 | Yes | |
NNVINYYJNCKGRA
|
7.3 | IC50 | 4 | — | |
SSMSJTVEHMWTFZ
|
7.3 | IC50 | 6 | — | |
SSMSJTVEHMWTFZ
|
7.3 | IC50 | 6 | — | |
TUJUZVJICDSNLY
|
7.3 | Ki | 19 | — | |
ULGQQNXZFKHRIL
|
7.3 | IC50 | 3 | — | |
XDTAJQIDTGQFQG
|
7.3 | IC50 | 3 | — | |
LTGPAFCQBMWTBC
|
7.3 | IC50 | 5 | Yes | |
TWDPQJRHLMLPRP
|
7.3 | IC50 | 3 | Yes | |
YSWBUBWIVNTGAC
|
7.3 | IC50 | 4 | Yes | |
CYRPAUWSHGGREB
|
7.3 | Ki | 8 | Yes | |
QYTBMLLWBZLPMF
|
7.3 | IC50 | 6 | — | |
TUKOILYAIRACKC
|
7.3 | IC50 | 7 | Yes | |
UJBAYCIQPBHHBB
|
7.3 | IC50 | 3 | Yes | |
VNPLXDZLURAZHZ
|
7.3 | IC50 | 5 | — | |
KGPGFQWBCSZGEL
|
7.3 | Kd | 59 | Yes | |
VLEXKLPWUMHBQI
|
7.3 | IC50 | 3 | Yes | |
CLAXUCQFRATVEQ
|
7.2 | IC50 | 3 | Yes | |
HFSXGAKDODZJBV
|
7.2 | IC50 | 3 | Yes | |
NKWSAYGUIMPROA
|
7.2 | IC50 | 10 | — | |
DEAHYBLYNUJAIJ
|
7.2 | IC50 | 3 | Yes | |
ITOPVUHELOTFOX
|
7.2 | IC50 | 3 | Yes | |
PDSONWYECZHBAE
|
7.2 | Ki | 3 | — | |
CEMBEUHBOHDWPN
|
7.2 | IC50 | 4 | — |