Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IFLKFPIAJMOXTG
|
7.6 | IC50 | 3 | Yes | |
ZBGKNKIERAXNKR
|
7.6 | IC50 | 3 | Yes | |
GDEWTWLRSSWVEX
|
7.5 | IC50 | 3 | Yes | |
KJYFFRNQSIBKHB
|
7.5 | IC50 | 3 | Yes | |
KPCVAMMFCPIUIU
|
7.5 | IC50 | 12 | Yes | |
IFPLUMSPGLKAOT
|
7.5 | IC50 | 3 | Yes | |
KAJIDAUQCMSGGN
|
7.5 | IC50 | 3 | Yes | |
RDFXBYJUHGEYHA
|
7.5 | IC50 | 9 | Yes | |
COHIPYSTFCKVTM
|
7.5 | Ki | 2 | — | |
FLWBAZOREVFEAD
|
7.5 | IC50 | 3 | Yes | |
JOOTZGPUMCZHLH
|
7.5 | IC50 | 5 | — | |
JOOTZGPUMCZHLH
|
7.5 | IC50 | 5 | — | |
NNVINYYJNCKGRA
|
7.5 | IC50 | 5 | — | |
TXVBBLNFLUZGIT
|
7.5 | IC50 | 6 | — | |
USEYXZSHZLLAJS
|
7.5 | IC50 | 6 | — | |
WOFBHAKTZOZODW
|
7.5 | IC50 | 6 | — | |
XXDWSQPJTJZKSJ
|
7.5 | IC50 | 12 | Yes | |
ZZSBPGIGIUFJRA
|
7.5 | IC50 | 15 | Yes | |
BGFPMEIULZPARM
|
7.5 | Ki | 3 | — | |
FELQRVDTGNDOSI
|
7.5 | IC50 | 15 | Yes | |
GVSRILDMSGVJTR
|
7.5 | IC50 | 7 | — | |
MVMGNWUSDKNEKN
|
7.5 | IC50 | 5 | — | |
MYOUXQLHWTWXON
|
7.5 | IC50 | 16 | Yes | |
OBGSXFHKYFQXJY
|
7.5 | IC50 | 2 | — | |
XYUFCXJZFZPEJD
|
7.5 | IC50 | 6 | — | |
ZYTFPHRVOZXPGZ
|
7.5 | Ki | 30 | — | |
QMGUOJYZJKLOLH
|
7.5 | IC50 | 21 | Yes | |
BSPJFZBMQCBCCJ
|
7.5 | IC50 | 3 | Yes | |
FOPORVBLOTVXEK
|
7.5 | Ki | 5 | — | |
LRHWSAFUUBKSML
|
7.5 | Ki | 5 | — | |
YDZJEODKNRAYMA
|
7.5 | IC50 | 12 | Yes | |
JTVBXQAYBIJXRP
|
7.5 | Kd | 20 | — | |
MMFFLYVAVCPQHO
|
7.5 | IC50 | 3 | Yes | |
YAHQEFRFUBPDAT
|
7.5 | IC50 | 3 | Yes | |
DKOCZDDCSUQYTF
|
7.5 | IC50 | 5 | — | |
ZYUGNHPOVKADFZ
|
7.5 | IC50 | 11 | — | |
AWKZERSILQVXCP
|
7.4 | IC50 | 3 | Yes | |
DAQIKFLEHCFYPH
|
7.4 | IC50 | 3 | Yes | |
HPBJQOWLAKYNDM
|
7.4 | IC50 | 15 | Yes | |
MMVHNEPFDQHBTM
|
7.4 | IC50 | 5 | Yes | |
XWKJUHBICAMYNW
|
7.4 | Ki | 6 | — | |
AMSOPBXQXSAAAC
|
7.4 | IC50 | 12 | Yes | |
PBCZSGKMGDDXIJ
|
7.4 | IC50 | 68 | Yes | |
LPIHDMXDUPXXEU
|
7.4 | IC50 | 6 | — | |
IVGCXWIFBNPPBW
|
7.4 | IC50 | 6 | — | |
KJGUOQMSLKZPAT
|
7.4 | IC50 | 17 | Yes | |
PQWWKDOKHDWZBH
|
7.4 | IC50 | 6 | — | |
SIXGXRZCYDCNFL
|
7.4 | IC50 | 4 | — | |
YPJJSXBVVGPFHA
|
7.4 | Ki | 18 | — | |
ZKROVQCECIHHES
|
7.4 | IC50 | 3 | Yes |