Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTBKLEUJZBEEEQ
|
7.7 | IC50 | 3 | Yes | |
PCMKNGBJTSLXPM
|
7.7 | IC50 | 3 | Yes | |
SDEAUNNPTULCST
|
7.7 | Ki | 3 | — | |
UWDSNDOLVCLEJW
|
7.7 | Ki | 8 | Yes | |
VREDQQFDKBEALJ
|
7.7 | IC50 | 5 | — | |
ZRTHIYZKVPIBMW
|
7.7 | IC50 | 3 | Yes | |
LUZOFMGZMUZSSK
|
7.7 | Ki | 3 | — | |
AZIMEXGKUWHPQV
|
7.7 | IC50 | 12 | Yes | |
BPNNZZBLGSVSAA
|
7.7 | IC50 | 6 | — | |
BPNNZZBLGSVSAA
|
7.7 | IC50 | 7 | — | |
BSFNGHCTZDCQBF
|
7.7 | Ki | 93 | — | |
CKJRKRPDNLRZPQ
|
7.7 | IC50 | 6 | — | |
CKJRKRPDNLRZPQ
|
7.7 | IC50 | 7 | — | |
DKHPQQRGPHOKBV
|
7.7 | IC50 | 3 | — | |
FSBMWCWKNXQVMP
|
7.7 | IC50 | 12 | Yes | |
GQCWIZZVARXZGR
|
7.7 | IC50 | 6 | — | |
GQCWIZZVARXZGR
|
7.7 | IC50 | 6 | — | |
HDYPWSDXJZTYPP
|
7.7 | IC50 | 3 | Yes | |
NIUBYBAPAVVDMG
|
7.7 | IC50 | 6 | — | |
NIUBYBAPAVVDMG
|
7.7 | IC50 | 6 | — | |
OBRQLJITIRIMLQ
|
7.7 | IC50 | 11 | — | |
OVJZHEDXGAPGDA
|
7.7 | IC50 | 5 | — | |
UVZVWLFSZNPMBS
|
7.7 | Ki | 17 | — | |
VVHIKEQUOUROGD
|
7.7 | Ki | 3 | — | |
YUKJJLKBBAFYNN
|
7.7 | IC50 | 12 | Yes | |
ZOGSVRRXRLSQNC
|
7.7 | IC50 | 6 | — | |
IPEXHQGMTHOKQV
|
7.7 | Kd | 12 | — | |
IWPNPNGPAZFVCZ
|
7.7 | IC50 | 3 | Yes | |
POTTVLREWUNNRO
|
7.7 | IC50 | 3 | — | |
AJWYNSXOWAWFRT
|
7.7 | IC50 | 3 | Yes | |
FDFNBRWULOMEEQ
|
7.7 | Ki | 3 | — | |
MODWLWDUUDGOEB
|
7.7 | IC50 | 5 | Yes | |
BJNQKVADRDIKFO
|
7.6 | Ki | 6 | Yes | |
XYUFCXJZFZPEJD
|
7.6 | IC50 | 9 | — | |
XYUFCXJZFZPEJD
|
7.6 | IC50 | 23 | Yes | |
WEAXGDQVWHPARP
|
7.6 | Ki | 2 | — | |
GQKHMFJDTFXZNM
|
7.6 | IC50 | 5 | Yes | |
JMBOYLIMLIXSDW
|
7.6 | IC50 | 3 | Yes | |
YQYBJEBDZCPCSM
|
7.6 | IC50 | 5 | — | |
BOJKFRKNLSCGHY
|
7.6 | Ki | 3 | — | |
ATTAVUMAVKBGLW
|
7.6 | IC50 | 3 | Yes | |
AXRCEOKUDYDWLF
|
7.6 | Kd | 31 | — | |
AZEVIHVCFXQWCI
|
7.6 | IC50 | 3 | Yes | |
GQDKNFXTRUBAEB
|
7.6 | IC50 | 3 | Yes | |
IWZNOWDHBWUZLK
|
7.6 | IC50 | 3 | Yes | |
UWFSHWFUBYEFAT
|
7.6 | IC50 | 6 | — | |
VGNKOJURPOHWJF
|
7.6 | Ki | 21 | — | |
KAJIDAUQCMSGGN
|
7.6 | IC50 | 8 | Yes | |
BPNUQXPIQBZCMR
|
7.6 | Kd | 83 | Yes | |
HFPUIOYUZROFHG
|
7.6 | IC50 | 6 | — |