Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDXNZQYZADSNCP
|
8.0 | IC50 | 12 | Yes | |
DSXXEELGXBCYNQ
|
8.0 | IC50 | 28 | Yes | |
FFKRSNGYONHGEV
|
8.0 | IC50 | 12 | Yes | |
FWEDWNSLCBHVQT
|
8.0 | IC50 | 5 | — | |
MKCCHIFQLCHEBR
|
8.0 | IC50 | 3 | Yes | |
OPQUGNXQOSDRMT
|
8.0 | IC50 | 12 | Yes | |
PGWBJRRPIUVOAD
|
8.0 | IC50 | 12 | Yes | |
QZIHHXYMIRLTTO
|
8.0 | IC50 | 3 | Yes | |
XSRHBCYNCKAFKS
|
8.0 | Ki | 45 | — | |
CPXHOALOZNWMML
|
8.0 | Ki | 3 | — | |
LUZOFMGZMUZSSK
|
8.0 | Ki | 8 | Yes | |
WUJFWMRQXPIJIN
|
8.0 | IC50 | 3 | Yes | |
XYUFCXJZFZPEJD
|
8.0 | IC50 | 9 | — | |
XUTMONHBGYHWES
|
7.9 | Ki | 5 | — | |
BGMFLWUQWMTTSW
|
7.9 | IC50 | 8 | — | |
FHISAROGPSYNME
|
7.9 | Ki | 10 | — | |
HSZCSAUAGLABDS
|
7.9 | Ki | 5 | — | |
QNKCGRSWHZOKEA
|
7.9 | IC50 | 3 | — | |
STEGBXHZVWLLAP
|
7.9 | IC50 | 6 | — | |
WOFBHAKTZOZODW
|
7.9 | IC50 | 6 | — | |
HOTMBRBDTHIOMH
|
7.9 | IC50 | 3 | Yes | |
NXSJMRCTGYTSTK
|
7.9 | Kd | 200 | — | |
PBCZSGKMGDDXIJ
|
7.9 | IC50 | 14 | Yes | |
RSTWARDIGORXQU
|
7.9 | Ki | 7 | Yes | |
GPGZMTPPOHCJRE
|
7.8 | IC50 | 16 | Yes | |
SMZYTCQRZVNFFJ
|
7.8 | IC50 | 16 | Yes | |
YTAXZQBKZAMFER
|
7.8 | IC50 | 3 | Yes | |
DNZGKSANTHABGF
|
7.8 | IC50 | 3 | Yes | |
MVPSDKPPZLPMBB
|
7.8 | Ki | 7 | Yes | |
ZMHXVAQNZDUNOG
|
7.8 | IC50 | 6 | — | |
JKERAVGYQRGKNA
|
7.8 | Ki | 2 | — | |
BUCGAQTZOOCIRW
|
7.8 | IC50 | 5 | Yes | |
CLRFYTGANQZOBS
|
7.8 | Ki | 41 | — | |
CXSQMXRQOZZFLD
|
7.8 | IC50 | 18 | — | |
GHPFQRTVUDXWCC
|
7.8 | Ki | 35 | — | |
GXRHJQDLOAPBIK
|
7.8 | IC50 | 3 | Yes | |
HXWARSZQGAFXJM
|
7.8 | Ki | 7 | — | |
MLGGUGPIWDHBAI
|
7.8 | IC50 | 10 | — | |
MLGGUGPIWDHBAI
|
7.8 | Ki | 33 | — | |
XEHZTUCPROUDNJ
|
7.8 | IC50 | 3 | Yes | |
XYKVGXVSUAFNLB
|
7.8 | IC50 | 3 | Yes | |
ZCBUQCWBWNUWSU
|
7.8 | Kd | 59 | — | |
DZIUPOCVDSYPSY
|
7.8 | IC50 | 8 | Yes | |
JOSDGPURRZWOOC
|
7.8 | Ki | 2 | — | |
OQICVMYHDNIADM
|
7.8 | IC50 | 6 | — | |
FXGHOAZJQNLNFD
|
7.8 | IC50 | 13 | Yes | |
CIVFNZIOXQANAM
|
7.8 | IC50 | 5 | — | |
DNZGKSANTHABGF
|
7.7 | IC50 | 3 | Yes | |
GMQQMSKNSNVPOW
|
7.7 | IC50 | 9 | Yes | |
ICQQDVZUHPTFPS
|
7.7 | IC50 | 3 | Yes |