Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PGBOLFMQGRFIRL
|
8.4 | Ki | 5 | — | |
CKJRKRPDNLRZPQ
|
8.4 | IC50 | 6 | — | |
CKJRKRPDNLRZPQ
|
8.4 | IC50 | 7 | — | |
QJVMNACFDUTHPM
|
8.4 | IC50 | 6 | — | |
DHUPFOOXPODTRC
|
8.4 | IC50 | 3 | Yes | |
CVCIQKJLZNEUAZ
|
8.4 | IC50 | 7 | Yes | |
FCVHMDURXUOCFY
|
8.3 | IC50 | 6 | — | |
FCVHMDURXUOCFY
|
8.3 | IC50 | 7 | — | |
MKPSMRQVGPTYRL
|
8.3 | IC50 | 5 | — | |
MKPSMRQVGPTYRL
|
8.3 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
8.3 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
8.3 | IC50 | 7 | — | |
WOFBHAKTZOZODW
|
8.3 | IC50 | 6 | — | |
YIZRPXUMLQCIMQ
|
8.3 | IC50 | 9 | — | |
YIZRPXUMLQCIMQ
|
8.3 | IC50 | 7 | — | |
YIZRPXUMLQCIMQ
|
8.3 | IC50 | 9 | — | |
YIZRPXUMLQCIMQ
|
8.3 | IC50 | 6 | — | |
YOVNFNXUCOWYSG
|
8.3 | Ki | 33 | Yes | |
YRTMRGPNXUUDTD
|
8.3 | IC50 | 5 | — | |
ZDISSWUDAVTQSK
|
8.3 | IC50 | 3 | Yes | |
OWLWQUHZHTVSAN
|
8.2 | IC50 | 6 | — | |
SZJIXBKHTOPEKG
|
8.2 | IC50 | 6 | Yes | |
BPNNZZBLGSVSAA
|
8.2 | IC50 | 6 | — | |
BPNNZZBLGSVSAA
|
8.2 | IC50 | 7 | — | |
OWJIKBAZUBPKGN
|
8.2 | IC50 | 6 | — | |
OWJIKBAZUBPKGN
|
8.2 | IC50 | 7 | — | |
AQGHYUYFBXMRBC
|
8.2 | IC50 | 6 | — | |
QZCYXWFWSDBJGL
|
8.2 | Ki | 8 | Yes | |
SAYMBMAHSBYKKR
|
8.2 | IC50 | 12 | Yes | |
YRYJOPMCJLSMNU
|
8.2 | IC50 | 6 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
ZQBULZYTDGUSSK
|
8.2 | Ki | 3 | Yes | |
XXJXHXJWQSCNPX
|
8.2 | IC50 | 7 | — | |
IDSZLHFEKAUIOL
|
8.1 | IC50 | 7 | Yes | |
WQEXBJWFPAMSGJ
|
8.1 | Ki | 8 | Yes | |
BPNUQXPIQBZCMR
|
8.1 | Ki | 60 | — | |
NDIUYMHNCUTVGE
|
8.1 | Ki | 25 | — | |
UAQJVFADAYIBGC
|
8.1 | Ki | 23 | — | |
XFWUTMHVDGPWLH
|
8.1 | Ki | 75 | — | |
XUDDPIKSCLCQKJ
|
8.1 | IC50 | 3 | Yes | |
YUJAAMQBNNAQRP
|
8.1 | IC50 | 6 | — | |
SNIZLDGVUOKDEA
|
8.1 | IC50 | 3 | Yes | |
UHIFMIXIMAHXIB
|
8.1 | IC50 | 6 | — | |
BQJRUJTZSGYBEZ
|
8.1 | Kd | 13 | Yes | |
POTTVLREWUNNRO
|
8.1 | IC50 | 17 | Yes | |
VDBJPTBJJMQNOW
|
8.0 | IC50 | 6 | — | |
PQWWKDOKHDWZBH
|
8.0 | IC50 | 6 | — | |
PQWWKDOKHDWZBH
|
8.0 | IC50 | 6 | — | |
MCIAOHYVDXDCLF
|
8.0 | Ki | 8 | Yes | |
SJLWKRZGICWCDL
|
8.0 | IC50 | 3 | Yes |