Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MCQPMCDEXWCMDM
|
6.1 | Ki | 2 | — | |
RLJSCSODGXVAEX
|
6.1 | IC50 | 3 | Yes | |
TWCARTFPHQNBPF
|
6.1 | Ki | 16 | — | |
UTFXYGYVDDLJER
|
6.1 | Ki | 36 | — | |
UUMNMGQJQBYDMR
|
6.1 | IC50 | 2 | — | |
UZWDCWONPYILKI
|
6.1 | Kd | 47 | — | |
WSXYBDKZFNJOTP
|
6.1 | IC50 | 12 | Yes | |
ZRQXCQXWTLVASO
|
6.1 | Ki | 36 | — | |
MRBNLCLXWRXFJX
|
6.1 | IC50 | 15 | — | |
JPOSFPUHBHRUAX
|
6.1 | IC50 | 40 | Yes | |
UVUMDKAWNBACHR
|
6.1 | IC50 | 3 | Yes | |
ADVDNJCNXOTAHZ
|
6.1 | IC50 | 2 | — | |
DIZACSOTRSXCHC
|
6.1 | IC50 | 4 | — | |
QEQRMPXQCBZMSU
|
6.1 | IC50 | 3 | Yes | |
GHRBXKFGXPOEGA
|
6.0 | IC50 | 12 | Yes | |
NLJJDZMBYLCWHR
|
6.0 | IC50 | 2 | — | |
ONMFJTSDBZIFTK
|
6.0 | Ki | 2 | — | |
IAYGCINLNONXHY
|
6.0 | Kd | 50 | — | |
PQUHKNDRTYATRD
|
6.0 | IC50 | 3 | Yes | |
SGHXFHRRWFLILP
|
6.0 | IC50 | 8 | — | |
UNULBQHMZBESJQ
|
6.0 | IC50 | 4 | — | |
GZHZMFFLSDMMTQ
|
6.0 | IC50 | 2 | — | |
XCOCBCMPDCQQRX
|
6.0 | Ki | 2 | — | |
AYCPARAPKDAOEN
|
6.0 | Kd | 73 | — | |
KQUBTSBQLPIFSM
|
6.0 | IC50 | 5 | — | |
UHVOJNPWRWKQSP
|
6.0 | IC50 | 3 | Yes | |
GAEKZIARZJRZTM
|
6.0 | IC50 | 3 | — | |
GPKQGYSDQQIJLW
|
6.0 | Ki | 19 | — | |
GVMDVMPNOAVKJR
|
6.0 | Ki | 26 | Yes | |
GXFGHUNNGNQSMQ
|
6.0 | Ki | 19 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LWSORTKUYSYDMP
|
6.0 | IC50 | 12 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MHHTXOIOMYDUOQ
|
6.0 | Ki | 4 | — | |
NKANXQFJJICGDU
|
6.0 | IC50 | 35 | Yes | |
UQFRSHRWRKYNDE
|
6.0 | Ki | 17 | Yes | |
UUCJUCRTIKZRFG
|
6.0 | IC50 | 12 | Yes | |
VAMDLIMJLAPZGX
|
6.0 | Ki | 10 | — | |
VXBAJLGYBMTJCY
|
6.0 | Kd | 34 | Yes | |
WZOQKGRFRIFIEB
|
6.0 | IC50 | 3 | — | |
YKYRQCWLYUTVIE
|
6.0 | Ki | 16 | — |