Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXZAPNVTOAXLTD
|
6.3 | Ki | 3 | — | |
DBENCPRFMOMLTO
|
6.3 | Ki | 2 | — | |
NEGCBIBMPAHBIM
|
6.3 | IC50 | 12 | Yes | |
BAQFZMFDZMQJAM
|
6.2 | IC50 | 12 | Yes | |
TXBFOGDMTCNBBT
|
6.2 | IC50 | 12 | Yes | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 82 | Yes | |
HSRYETVWRVWJQQ
|
6.2 | IC50 | 6 | — | |
JXGKWKHETDHDCC
|
6.2 | Ki | 5 | — | |
OLYSKMGKJANIPC
|
6.2 | Ki | 2 | — | |
QHLWNCNFYOUHJB
|
6.2 | IC50 | 2 | — | |
QQKKPWJFHBFCTH
|
6.2 | IC50 | 10 | Yes | |
TWUWFRLZDWDJLT
|
6.2 | Ki | 10 | Yes | |
ZUKHVOLIPVGCHQ
|
6.2 | Ki | 10 | Yes | |
FNTXTLNLTQPVBJ
|
6.2 | IC50 | 6 | — | |
JBXKODTZBBUAQG
|
6.2 | IC50 | 3 | Yes | |
DKXHSOUZPMHNIZ
|
6.2 | Ki | 51 | Yes | |
FONINLXADYUZFI
|
6.2 | Ki | 25 | — | |
HLXIFVDYTGEUJV
|
6.2 | IC50 | 15 | Yes | |
LWBSSNRDDDFHSH
|
6.2 | Ki | 9 | — | |
MBRVCJRFWYHVHE
|
6.2 | Ki | 9 | — | |
NKGLJTITEFZKAN
|
6.2 | Ki | 35 | — | |
NRSGWEVTVGZDFC
|
6.2 | Ki | 50 | — | |
QMMMGQKKOKYDMN
|
6.2 | Ki | 5 | — | |
SGHXFHRRWFLILP
|
6.2 | Ki | 29 | — | |
ZZKAMKCYEYGTEB
|
6.2 | IC50 | 4 | — | |
AKBBEKGAHSYAKD
|
6.2 | IC50 | 2 | — | |
KPJDEGAKXAUVAC
|
6.2 | Ki | 15 | Yes | |
SBTUVVZTMJEJMZ
|
6.2 | IC50 | 3 | Yes | |
BGVKOUSMQGMSDY
|
6.2 | IC50 | 4 | — | |
CWFIQHQECWPWQG
|
6.2 | IC50 | 16 | Yes | |
JRKIWLCZVXSNKH
|
6.2 | IC50 | 2 | — | |
LOLIGEKXJXAKFQ
|
6.2 | IC50 | 3 | Yes | |
ORNADCNXUPZOQN
|
6.2 | IC50 | 15 | — | |
DAGKXAWMGQZKFD
|
6.2 | IC50 | 4 | — | |
AFICENYJQYURCA
|
6.1 | Ki | 2 | — | |
OPMCPILSGDNUOY
|
6.1 | IC50 | 3 | Yes | |
AXTAPYRUEKNRBA
|
6.1 | IC50 | 24 | — | |
BGLHPPIIHCSAHO
|
6.1 | IC50 | 3 | Yes | |
KVPCAWMJGFMDHN
|
6.1 | IC50 | 3 | Yes | |
AUQFRAINFQCKDW
|
6.1 | IC50 | 2 | — | |
CFBADDSSFSYJPF
|
6.1 | Ki | 23 | — | |
CLGKERUQODCNJI
|
6.1 | IC50 | 3 | Yes | |
DFMCXVONDDGQIY
|
6.1 | Ki | 66 | — | |
GDYZFFBMSBDTAA
|
6.1 | Ki | 60 | — | |
GPDVHOTUPZYYBA
|
6.1 | IC50 | 2 | Yes | |
HOBMVEVXDIOMDM
|
6.1 | Ki | 18 | — | |
IYOZTVGMEWJPKR
|
6.1 | Ki | 10 | — | |
JJJSCYSPSKBQAX
|
6.1 | Ki | 34 | — | |
KCKXYZOBGBJZEG
|
6.1 | Ki | 36 | — |