Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HHLKZSJXDAZIGG
|
6.4 | IC50 | 10 | Yes | |
IPKHSYHXXAIZDD
|
6.4 | Ki | 18 | — | |
JQGRMZUVGWRDIV
|
6.4 | IC50 | 6 | — | |
QAJPIJHWTGPUNZ
|
6.4 | Ki | 37 | — | |
RELJBNLDXPSLLS
|
6.4 | IC50 | 6 | — | |
VYXIZKJRRNWQAK
|
6.4 | IC50 | 6 | — | |
YCFZRTPAYLSXMM
|
6.4 | IC50 | 2 | — | |
YGEACCLUBSGMMJ
|
6.4 | Ki | 16 | — | |
AGFZKGRTVAVKSP
|
6.4 | IC50 | 2 | — | |
DOCCMHSNEKDEOV
|
6.4 | IC50 | 3 | Yes | |
JJFJVIQFBDEVSN
|
6.4 | IC50 | 4 | Yes | |
OBEJTRHPRSRHSZ
|
6.4 | Ki | 2 | — | |
WMWXMWABKUQJNC
|
6.4 | IC50 | 3 | — | |
KAJXOWFGKYKMMZ
|
6.4 | IC50 | 26 | Yes | |
MMBXHOMWDHTANV
|
6.4 | IC50 | 3 | Yes | |
NFRKACJUZYOBMM
|
6.4 | Ki | 5 | Yes | |
TZLVNGQSHBVJDQ
|
6.4 | IC50 | 3 | Yes | |
XYUFCXJZFZPEJD
|
6.4 | IC50 | 5 | — | |
XYUFCXJZFZPEJD
|
6.4 | IC50 | 4 | — | |
XEAWPTQREKCGSA
|
6.4 | IC50 | 3 | Yes | |
HAWYDMHDXJUGRR
|
6.3 | IC50 | 3 | Yes | |
RQFQHXQYIYDKMC
|
6.3 | IC50 | 3 | Yes | |
SONJXLIPDOXRGA
|
6.3 | IC50 | 3 | Yes | |
WRHOONMCSKWHRY
|
6.3 | IC50 | 2 | — | |
ZFNQOYBHHLGQDV
|
6.3 | IC50 | 12 | Yes | |
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
CPRVBHBRBVVLHL
|
6.3 | IC50 | 11 | — | |
PXRPXQKBRGMQJJ
|
6.3 | Ki | 2 | — | |
XYUYSDBKGVJSKN
|
6.3 | IC50 | 5 | — | |
AOBLBPWPSKBHSI
|
6.3 | Ki | 55 | — | |
ATBAETXFFCOZOY
|
6.3 | IC50 | 39 | — | |
CCRCRSXDKXZDGK
|
6.3 | IC50 | 12 | Yes | |
HNXJWWRRSGDVIW
|
6.3 | Ki | 13 | — | |
JRKIWLCZVXSNKH
|
6.3 | IC50 | 2 | — | |
QQVBBJUQEBYOFD
|
6.3 | IC50 | 3 | Yes | |
RFVBRKXQYUDGIO
|
6.3 | Ki | 23 | — | |
RRGJUOHIDUNWCQ
|
6.3 | IC50 | 2 | — | |
SBFPHSVZEXSHTL
|
6.3 | Ki | 62 | — | |
VBNPWXWJZJNXEY
|
6.3 | Ki | 18 | Yes | |
VDRCTDRTPPONJY
|
6.3 | IC50 | 2 | — | |
WNMXOXGXHRHBLO
|
6.3 | Ki | 4 | — | |
WZBMMJKAHHOXRG
|
6.3 | Ki | 16 | — | |
XOIXULDEDZVLBV
|
6.3 | IC50 | 2 | — | |
YROCVAOLJXRFKK
|
6.3 | IC50 | 3 | Yes | |
ZKZXNDJNWUTGDK
|
6.3 | Ki | 14 | — | |
NZTPJNIILSLMRH
|
6.3 | IC50 | 7 | — | |
JSPAUBUYPPZXSG
|
6.3 | Ki | 17 | Yes | |
ORNADCNXUPZOQN
|
6.3 | IC50 | 15 | — | |
QQTVBLADGKPBRJ
|
6.3 | Ki | 2 | — | |
ZBGSOGNHNSNOLN
|
6.3 | Ki | 2 | — |