Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CGZJWCJQOOVDSV
|
6.5 | IC50 | 3 | Yes | |
RYJIUYPHHDCWNM
|
6.5 | IC50 | 2 | — | |
SLGVPUQAGYTPGZ
|
6.5 | IC50 | 3 | Yes | |
AWDORCFLUJZUQS
|
6.5 | Ki | 22 | — | |
DPRGOXVMSNDADU
|
6.5 | Ki | 16 | — | |
FLEAYYMORDPWAJ
|
6.5 | Ki | 90 | — | |
JXMYIDZREHNPDO
|
6.5 | Ki | 19 | — | |
LOOCBXNRYHTANC
|
6.5 | IC50 | 2 | — | |
LRZYYIZFBXFSJB
|
6.5 | Ki | 69 | — | |
MASJMHFQMYAPJR
|
6.5 | Ki | 41 | — | |
PHDOQFYDQFLEMJ
|
6.5 | IC50 | 3 | Yes | |
QQWUGDVOUVUTOY
|
6.5 | Ki | 231 | Yes | |
SNQKPKFVSANKFP
|
6.5 | IC50 | 6 | — | |
TVIALAOHRQNPOI
|
6.5 | IC50 | 12 | Yes | |
USHMNZBDAOGLMB
|
6.5 | Ki | 26 | — | |
XMFUGSRATNLPRM
|
6.5 | Ki | 19 | — | |
XYZNKCSDQRKAFR
|
6.5 | Ki | 53 | — | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
LNLLTZUEPWPAPX
|
6.5 | IC50 | 3 | Yes | |
MGQDMSJZRRHMFT
|
6.5 | IC50 | 6 | — | |
MGQDMSJZRRHMFT
|
6.5 | IC50 | 6 | — | |
HCDKPFLBNVCSDB
|
6.5 | IC50 | 5 | — | |
HCDKPFLBNVCSDB
|
6.5 | IC50 | 5 | — | |
NJADSZALPMCYLV
|
6.5 | IC50 | 3 | Yes | |
RMRAGHHDUPBIJZ
|
6.5 | Ki | 2 | — | |
XEAWPTQREKCGSA
|
6.5 | IC50 | 3 | Yes | |
DMTWTBBJQAQFID
|
6.5 | IC50 | 3 | Yes | |
HPCPUHOULFPBCQ
|
6.5 | IC50 | 12 | Yes | |
JDZXLEPJWLCESI
|
6.5 | IC50 | 12 | Yes | |
JSBPEIYUYLNLLN
|
6.5 | IC50 | 3 | Yes | |
KPDRLZMGHJWHQC
|
6.5 | IC50 | 3 | Yes | |
RHBWAFDCVFMIFK
|
6.5 | IC50 | 12 | Yes | |
SFDFKLDQKSPRHB
|
6.5 | IC50 | 15 | Yes | |
BJLOBSMGZUMYOP
|
6.5 | IC50 | 8 | — | |
MCQPMCDEXWCMDM
|
6.5 | Ki | 2 | — | |
QYEKPILGAVXHQH
|
6.4 | IC50 | 2 | — | |
QYEKPILGAVXHQH
|
6.4 | IC50 | 5 | — | |
RPLXVENRWORMRX
|
6.4 | IC50 | 12 | Yes | |
AJFLRCLZEMUXCH
|
6.4 | IC50 | 4 | — | |
LBDSTAIEEDAXPE
|
6.4 | IC50 | 3 | Yes | |
VKLQFIYLAKBNIW
|
6.4 | IC50 | 3 | Yes | |
GCWARPTUQCJUSX
|
6.4 | IC50 | 3 | Yes | |
NGEJXMPZKYWYCI
|
6.4 | IC50 | 3 | Yes | |
GHCPXYAHSHXFSC
|
6.4 | IC50 | 3 | Yes | |
KEBDGBLZUWTDQL
|
6.4 | IC50 | 3 | Yes | |
MQFYZWYYZGTHAN
|
6.4 | IC50 | 14 | — | |
NCMIECXUNJAKKP
|
6.4 | IC50 | 4 | — | |
UDPITYZQIVOTOD
|
6.4 | IC50 | 3 | Yes | |
WQSBBBAQXNAUEM
|
6.4 | Ki | 2 | — | |
HCJOTKSJPHFVJC
|
6.4 | IC50 | 6 | — |