Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
COCXXLGXRJTCQZ
|
6.6 | IC50 | 6 | — | |
MZNUNTIEUOYNNT
|
6.6 | IC50 | 12 | Yes | |
OXEOHAXVZADDOC
|
6.6 | IC50 | 12 | Yes | |
YSVVBGPTTSJYPA
|
6.6 | IC50 | 12 | Yes | |
GLBDOEWDGNREFF
|
6.6 | IC50 | 3 | Yes | |
IELYDRFCDPGZGF
|
6.6 | Ki | 6 | — | |
SUMGTNPLBQXBDN
|
6.6 | IC50 | 3 | Yes | |
UIARLYUEJFELEN
|
6.6 | Kd | 289 | Yes | |
VCVVTOKATIJIQL
|
6.6 | Ki | 2 | — | |
WGNCBVWINIDEOT
|
6.6 | IC50 | 3 | Yes | |
YOSAIRCVRQVWFK
|
6.6 | IC50 | 3 | Yes | |
DEUHHHBUOZFXCN
|
6.6 | IC50 | 3 | Yes | |
DNPFEENAAKLCMC
|
6.6 | IC50 | 6 | — | |
GIVLJYSTNKNCGZ
|
6.6 | IC50 | 4 | — | |
GLKZLGGCNUQEAN
|
6.6 | IC50 | 3 | Yes | |
KAKGFGCTONHQJW
|
6.6 | Ki | 25 | — | |
KOZFSFOOLUUIGY
|
6.6 | IC50 | 26 | — | |
MVJMMLFMPWITEJ
|
6.6 | Ki | 110 | — | |
ORSMLITYQOYOSE
|
6.6 | IC50 | 2 | — | |
RCKVYOXLMHAPMO
|
6.6 | IC50 | 3 | Yes | |
RWYIXXFPIXIFNJ
|
6.6 | IC50 | 3 | — | |
SSZFVGXDYBMVDD
|
6.6 | IC50 | 12 | Yes | |
UDFDIIVNIYWXDM
|
6.6 | Ki | 74 | — | |
UZHPHLWTNWZGRX
|
6.6 | IC50 | 3 | Yes | |
XOVPCPRZRHQFBI
|
6.6 | Ki | 15 | — | |
XSDJOIOVIMPMHD
|
6.6 | Ki | 44 | — | |
YRTMRGPNXUUDTD
|
6.6 | IC50 | 2 | — | |
ZYTAPJWMMBTUHH
|
6.6 | IC50 | 4 | Yes | |
CQBKEYNDDXJYNG
|
6.6 | Ki | 2 | — | |
DZBJTZXFZCERBJ
|
6.6 | Ki | 3 | — | |
PBCZSGKMGDDXIJ
|
6.6 | IC50 | 12 | Yes | |
LAOIBIIMKUINJL
|
6.6 | IC50 | 12 | Yes | |
QPOFNLCOWXWKRN
|
6.6 | IC50 | 3 | Yes | |
IXOVKVHWGKDXKQ
|
6.6 | IC50 | 12 | Yes | |
WQSCDMQTCWOCID
|
6.6 | IC50 | 2 | — | |
ZQTCWRKVJWJCMV
|
6.6 | IC50 | 3 | Yes | |
BRZYOTMFHLERHD
|
6.5 | Ki | 17 | Yes | |
DETMXRBVADAKAO
|
6.5 | IC50 | 3 | — | |
ZEGIXAPFKAAIOT
|
6.5 | IC50 | 3 | Yes | |
BNAXHIOTDMDOLF
|
6.5 | IC50 | 6 | — | |
NEBLJCMPKZILIG
|
6.5 | IC50 | 3 | Yes | |
ORVUCMUEXPKXML
|
6.5 | IC50 | 3 | — | |
WZFQFSZXBRORHS
|
6.5 | IC50 | 5 | — | |
ARKNUCQRPYIUMU
|
6.5 | IC50 | 6 | — | |
FDIBZBJWWAQEFA
|
6.5 | IC50 | 3 | Yes | |
FPSGCBWWRUZTIV
|
6.5 | IC50 | 3 | Yes | |
HODOOWOVFQSXBB
|
6.5 | IC50 | 6 | — | |
PEHFMYWGWHPKOC
|
6.5 | IC50 | 3 | — | |
QHZHJSWWHXUNNZ
|
6.5 | IC50 | 2 | — | |
XNKIVXYFRPYKHO
|
6.5 | IC50 | 12 | Yes |