Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OOPMDKIRVTXOPT
|
6.8 | IC50 | 11 | — | |
QEWSTOOMTBAUAG
|
6.8 | Ki | 17 | — | |
RKUKAACYUCUJEE
|
6.8 | Ki | 58 | — | |
VYIMDEHSEMUAKI
|
6.8 | IC50 | 3 | Yes | |
ZKHDDJKHTPLPOQ
|
6.8 | Ki | 62 | — | |
JCHWETQOLSPUBV
|
6.8 | IC50 | 14 | — | |
QGLALYPAHULRIM
|
6.8 | IC50 | 3 | Yes | |
WUXPTIWFTBYPCX
|
6.8 | Ki | 5 | Yes | |
ZEYTZKVCOZMUKL
|
6.8 | IC50 | 5 | — | |
JHKZENPNLYAVCT
|
6.8 | IC50 | 15 | Yes | |
OQSTWXKHTZWKLD
|
6.8 | IC50 | 15 | Yes | |
RSTWARDIGORXQU
|
6.8 | Ki | 5 | Yes | |
JTJAWKUSBMOQSN
|
6.7 | Ki | 5 | — | |
KRSQMQFKFCQXKG
|
6.7 | IC50 | 3 | Yes | |
MPKJLCGWZCOAHC
|
6.7 | IC50 | 3 | Yes | |
XJYBZBREOWBYIA
|
6.7 | IC50 | 3 | Yes | |
XRZURBBBXNHUNO
|
6.7 | IC50 | 7 | Yes | |
DQYBRTASHMYDJG
|
6.7 | IC50 | 13 | Yes | |
LGSHHKIOBFPSEK
|
6.7 | IC50 | 12 | Yes | |
OGFRRHMGGJQLRU
|
6.7 | IC50 | 3 | Yes | |
BOJKFRKNLSCGHY
|
6.7 | Ki | 10 | Yes | |
NOYZSLBPRMUTQD
|
6.7 | IC50 | 3 | Yes | |
NWNXQPGNDJISRZ
|
6.7 | IC50 | 2 | — | |
ORUUEFDGYYTXAF
|
6.7 | Ki | 26 | — | |
OSNSLFCSJAHEKW
|
6.7 | IC50 | 3 | Yes | |
RTQPLZRMXYMSIQ
|
6.7 | IC50 | 3 | Yes | |
SHENEEFOURUIBP
|
6.7 | Ki | 29 | — | |
TWUWFRLZDWDJLT
|
6.7 | Ki | 10 | Yes | |
UJYYVUFESIJSEY
|
6.7 | IC50 | 3 | Yes | |
VWVYILCFSYNJHF
|
6.7 | IC50 | 49 | — | |
XPHWIERLJBFPFV
|
6.7 | Ki | 69 | — | |
XTCHBPCWJUSYFA
|
6.7 | IC50 | 5 | Yes | |
YTCNCUIPQVXVOR
|
6.7 | IC50 | 2 | — | |
NTXWXFSAJRMWNA
|
6.7 | IC50 | 15 | — | |
RAOJISQDGOOXTK
|
6.7 | IC50 | 14 | Yes | |
DVHIIOLZYZNPJG
|
6.7 | IC50 | 3 | Yes | |
OCPILGAGUGFNJE
|
6.7 | IC50 | 6 | Yes | |
GDZULWKNFKCRJP
|
6.7 | IC50 | 7 | — | |
KHGDEZDNICAMOO
|
6.7 | IC50 | 6 | — | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
GZJKVFKNTQXSQM
|
6.7 | IC50 | 12 | Yes | |
IDVIOLNZWSXZGL
|
6.7 | Ki | 5 | Yes | |
JMRDOCPDIXFWLY
|
6.7 | IC50 | 3 | Yes | |
LBRQDCWYCRVFAG
|
6.7 | IC50 | 4 | — | |
QRBLWZIADYBYNA
|
6.7 | IC50 | 5 | — | |
ZMNWXCJLFBVMEJ
|
6.7 | IC50 | 3 | — | |
ZZNLNGDYKWBALR
|
6.7 | Ki | 2 | — | |
LGZGODIORQOSNB
|
6.7 | IC50 | 5 | — | |
LYJKMVFAIXOQLE
|
6.7 | IC50 | 9 | — | |
PWTCCMJTPHCGMS
|
6.7 | Ki | 3 | — |