Target Details
| UniProt AC | Q05655 |
|---|---|
| Gene Symbol | PRKCD |
| Protein Name | Protein kinase C delta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 742
- Clinical molecules 341
- Avg pChEMBL 7.15
KEGG Pathways (17)
- AGE-RAGE signaling pathway in diabetic complications
- Autophagy - animal
- C-type lectin receptor signaling pathway
- Chemical carcinogenesis - reactive oxygen species
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Estrogen signaling pathway
- Fc gamma R-mediated phagocytosis
- GnRH signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NOD-like receptor signaling pathway
- Neurotrophin signaling pathway
- Prion disease
- Shigellosis
- Type II diabetes mellitus
- Vascular smooth muscle contraction
Associated Diseases (1)
Active Molecules (742)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WTXAWDOYPWWUJL
|
10.1 | IC50 | 11 | — | |
FANQQVWXAKUWNI
|
10.0 | IC50 | 6 | — | |
MWKSRKSEWLRPBL
|
9.9 | Kd | 1075 | — | |
SSXCVTWCXHGTLK
|
9.9 | IC50 | 11 | — | |
KTGVSZYYHHRRGW
|
9.8 | IC50 | 11 | — | |
PUIKISPVMMUIMT
|
9.8 | Ki | 4 | — | |
VIESIZQAHOPEBR
|
9.8 | IC50 | 11 | — | |
NVYBXIDWOJVGQI
|
9.8 | IC50 | 11 | — | |
DSQFKUKVDCXORL
|
9.8 | Kd | 4 | — | |
APVOCXHEVZBCGS
|
9.7 | IC50 | 11 | — | |
FCYKUTUWVZTVAK
|
9.7 | Kd | 4 | — | |
DHTLXMRCLSUJPP
|
9.7 | IC50 | 11 | — | |
XSJFPSCYMJFDNI
|
9.5 | Ki | 7 | — | |
BQJRUJTZSGYBEZ
|
9.5 | Kd | 4 | — | |
VVRRZOFLLJAMIK
|
9.4 | IC50 | 11 | — | |
WAKGEHXTOOFEAE
|
9.4 | IC50 | 27 | — | |
MJQUEDHRCUIRLF
|
9.4 | Ki | 4 | — | |
DASVAQCTVIQROX
|
9.3 | Ki | 8 | Yes | |
JAMGGIDPOXFRAM
|
9.2 | Ki | 3 | — | |
UZCZCOMLMMSRLY
|
9.2 | IC50 | 6 | — | |
SUQYTYOVPXAUGB
|
9.1 | Ki | 3 | — | |
PHEDXBVPIONUQT
|
9.1 | Ki | 6 | Yes | |
SUQYTYOVPXAUGB
|
9.1 | Ki | 5 | — | |
IRGJDPZJEUYSKS
|
9.1 | IC50 | 7 | — | |
IRGJDPZJEUYSKS
|
9.1 | IC50 | 9 | — | |
IRGJDPZJEUYSKS
|
9.1 | IC50 | 6 | — | |
XKEOGEXDEKIDNA
|
9.1 | Ki | 3 | — | |
IRGJDPZJEUYSKS
|
9.0 | IC50 | 9 | — | |
URLJNGHIJZMXTK
|
9.0 | IC50 | 6 | — | |
XKEOGEXDEKIDNA
|
8.9 | Ki | 2 | — | |
ZOLWRJUQMXEKEO
|
8.9 | IC50 | 6 | — | |
OAVGBZOFDPFGPJ
|
8.9 | IC50 | 42 | Yes | |
REAZZDPREXHWNV
|
8.9 | Ki | 7 | — | |
QZVQSVZEEJEZSI
|
8.8 | Kd | 5 | — | |
HKSZLNNOFSGOKW
|
8.8 | Kd | 213 | — | |
NVSJOASGKCGXBZ
|
8.8 | IC50 | 16 | Yes | |
KMFOKKGKNMQAAN
|
8.7 | IC50 | 6 | — | |
QYBVZIIWBRIXMX
|
8.7 | IC50 | 12 | Yes | |
JZLFYMHIISZQCZ
|
8.7 | IC50 | 12 | Yes | |
RHJPBGWFGOAEID
|
8.7 | Ki | 8 | Yes | |
COOZRRUJSWPFHC
|
8.6 | IC50 | 3 | Yes | |
ZRYGSUWUNVQPFR
|
8.6 | IC50 | 6 | — | |
JHFLXYPDFJHPMX
|
8.6 | IC50 | 6 | — | |
OSVUGUHRKMMBSE
|
8.5 | Kd | 170 | — | |
ADMFLILDQJSEIK
|
8.5 | Ki | 72 | — | |
SWKUTOXEFLDOID
|
8.5 | Ki | 7 | — | |
UYBWOWHCXDBQRO
|
8.5 | IC50 | 6 | — | |
LPMWTDXPUOFZOV
|
8.5 | Ki | 7 | — | |
BDJSJCPWFZBQRA
|
8.5 | IC50 | 3 | Yes | |
CKCJAVJYEBDBEI
|
8.4 | Ki | 5 | — |