Target Details
| UniProt AC | Q05586 |
|---|---|
| Gene Symbol | GRIN1 |
| Protein Name | Glutamate receptor ionotropic, NMDA 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd) |
Summary
- Multi-target molecules 1,847
- Clinical molecules 2
- Avg pChEMBL 7.16
KEGG Pathways (19)
- Alcoholism
- Alzheimer disease
- Amphetamine addiction
- Amyotrophic lateral sclerosis
- Calcium signaling pathway
- Circadian entrainment
- Cocaine addiction
- Glutamatergic synapse
- Huntington disease
- Long-term potentiation
- Neuroactive ligand signaling
- Neuroactive ligand-receptor interaction
- Nicotine addiction
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Rap1 signaling pathway
- Ras signaling pathway
- Spinocerebellar ataxia
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (1,847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RCFQXVRTWUCEGF
|
7.9 | IC50 | 2 | — | |
UYNVMODNBIQBMV
|
7.9 | Ki | 12 | — | |
UZLQVSWICMHFOQ
|
7.9 | IC50 | 3 | — | |
XEZVPMCTUXYBQL
|
7.9 | IC50 | 3 | — | |
XGMDOIBDLYIGIR
|
7.9 | IC50 | 3 | — | |
MCPJEMSOWLNCCI
|
7.9 | IC50 | 2 | — | |
HGKAMARNFGKMLC
|
7.9 | IC50 | 2 | — | |
CUSFQDKHTGPAEB
|
7.8 | IC50 | 2 | — | |
HNYWSFRUDMHCJT
|
7.8 | IC50 | 3 | — | |
IBSHDUNQNHANES
|
7.8 | IC50 | 3 | — | |
JMIBTAQRPASKGS
|
7.8 | IC50 | 3 | — | |
LJPJRZZUZDMNHH
|
7.8 | IC50 | 2 | — | |
NBTCGYOJFCFXGC
|
7.8 | IC50 | 2 | — | |
PGHYKQGKLVXRFZ
|
7.8 | IC50 | 3 | — | |
QRWURIWWBKIGEH
|
7.8 | IC50 | 2 | — | |
RFMQELXSBUQROF
|
7.8 | IC50 | 2 | — | |
SBVYALDFQLTXPI
|
7.8 | IC50 | 3 | — | |
SLPAKDNQDFFJCF
|
7.8 | IC50 | 2 | — | |
ZHUXYMPPTHTCHT
|
7.8 | IC50 | 2 | — | |
ODCZSTMLJZVPMX
|
7.8 | IC50 | 2 | — | |
VMKGPIAHOBGSSJ
|
7.8 | IC50 | 2 | — | |
AXSCBNILWSGNQN
|
7.8 | IC50 | 3 | — | |
CQFDLBOEYHMIAO
|
7.8 | Ki | 7 | — | |
FXLVJUCJNSRRFS
|
7.8 | IC50 | 3 | — | |
GPZGIZRHGMSOFF
|
7.8 | IC50 | 2 | — | |
KNCORNNLLGPEEH
|
7.8 | IC50 | 2 | — | |
LEYPOMSTRVKGIO
|
7.8 | IC50 | 7 | — | |
MSRCCIJEUIUHKR
|
7.8 | IC50 | 2 | — | |
OVFADTJTEQNGRZ
|
7.8 | IC50 | 7 | — | |
PJELBWFBQFHVSN
|
7.8 | IC50 | 2 | — | |
PJRNVVYBYALHKB
|
7.8 | IC50 | 3 | — | |
QMYPDBMXMVHSTP
|
7.8 | IC50 | 3 | — | |
RNXMXSRYMNNORX
|
7.8 | IC50 | 2 | — | |
SAZWVXBHDXTTOA
|
7.8 | IC50 | 3 | — | |
ZGUFFXXBYKKICV
|
7.8 | IC50 | 3 | — | |
ZHDYEFOQPVKNEZ
|
7.8 | IC50 | 3 | — | |
ZRXUGWAQKKELFJ
|
7.8 | IC50 | 2 | — | |
ZZPOEZQWQQSOPW
|
7.8 | IC50 | 3 | — | |
AIQNIVLEFCDLOO
|
7.8 | IC50 | 3 | — | |
BRIPWIYBYCGTDM
|
7.8 | IC50 | 2 | — | |
BZQOGTTUTCCEIL
|
7.8 | IC50 | 3 | — | |
CWZJNVCLWRLJKV
|
7.8 | IC50 | 3 | — | |
DAUFBMVIIOKPFE
|
7.8 | IC50 | 2 | — | |
DYSFGTXMTFAFKK
|
7.8 | IC50 | 2 | — | |
FIYVYXKRDLLHTR
|
7.8 | IC50 | 2 | — | |
FMIAMQMNCXUHOE
|
7.8 | IC50 | 2 | — | |
HYZSDJJKDDEBRH
|
7.8 | IC50 | 3 | — | |
JXZDZNLIRKIPAG
|
7.8 | IC50 | 2 | — | |
LYTXTYPRIVRMHZ
|
7.8 | IC50 | 3 | — | |
SFVMMVWLGJROOM
|
7.8 | IC50 | 2 | — |