Target Details
| UniProt AC | Q05586 |
|---|---|
| Gene Symbol | GRIN1 |
| Protein Name | Glutamate receptor ionotropic, NMDA 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd) |
Summary
- Multi-target molecules 1,847
- Clinical molecules 2
- Avg pChEMBL 7.16
KEGG Pathways (19)
- Alcoholism
- Alzheimer disease
- Amphetamine addiction
- Amyotrophic lateral sclerosis
- Calcium signaling pathway
- Circadian entrainment
- Cocaine addiction
- Glutamatergic synapse
- Huntington disease
- Long-term potentiation
- Neuroactive ligand signaling
- Neuroactive ligand-receptor interaction
- Nicotine addiction
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Rap1 signaling pathway
- Ras signaling pathway
- Spinocerebellar ataxia
- cAMP signaling pathway
Associated Diseases (4)
Active Molecules (1,847)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XDOXQXVOQXBFEG
|
7.5 | IC50 | 3 | — | |
YTMYFHIXMXDDNC
|
7.5 | IC50 | 2 | — | |
MTBDNFJHIYJQJD
|
7.5 | IC50 | 2 | — | |
BDABGOLMYNHHTR
|
7.5 | IC50 | 7 | — | |
BZHNUBPUQWUDLK
|
7.5 | IC50 | 2 | — | |
CNQACROBXLOAOB
|
7.5 | IC50 | 2 | — | |
DTJFCMYFTQGQAV
|
7.5 | IC50 | 3 | — | |
FHGNVNGHYFDYNH
|
7.5 | IC50 | 2 | — | |
HIOJOKNCHBKSBH
|
7.5 | IC50 | 3 | — | |
IUTOHTCSZQLSEN
|
7.5 | IC50 | 3 | — | |
MVCXAPXDPCEJBN
|
7.5 | IC50 | 7 | — | |
NBVHNWXCUNZLAP
|
7.5 | IC50 | 2 | — | |
VWWCKJOBBMOFOB
|
7.5 | IC50 | 2 | — | |
WFCPRJXUOBJBNG
|
7.5 | IC50 | 2 | — | |
WSGRCCGHPXUJIX
|
7.5 | IC50 | 3 | — | |
YHSHZMVEPTTZEN
|
7.5 | IC50 | 2 | — | |
YRPXHEMBLZZKBZ
|
7.5 | IC50 | 2 | — | |
YSCWZYSSEFCNCE
|
7.5 | IC50 | 2 | — | |
ZFGYWAIHASVNRY
|
7.5 | IC50 | 2 | — | |
ZSCMNYOQZCYEIP
|
7.5 | IC50 | 2 | — | |
APXQQZMKKRAENC
|
7.5 | IC50 | 2 | — | |
FIBOTTIKYQQTKD
|
7.5 | IC50 | 2 | — | |
IIIXWSDMSFNCGD
|
7.5 | IC50 | 3 | — | |
LBJFZUMTQRTTFK
|
7.5 | IC50 | 2 | — | |
MTSDPZHXQKADDH
|
7.5 | IC50 | 2 | — | |
NFUVQXNWLIOKHO
|
7.5 | IC50 | 2 | — | |
OFDCWBLZQJRQNC
|
7.5 | IC50 | 3 | — | |
QENHDVWRWPITTM
|
7.5 | Ki | 2 | — | |
QKKOJQJQMMUNJU
|
7.5 | IC50 | 2 | — | |
SJXVVZZGIHEHIJ
|
7.5 | IC50 | 2 | — | |
SUUUWZXPEXVKGX
|
7.5 | IC50 | 7 | — | |
UCYXHLIEZUUIJU
|
7.5 | IC50 | 2 | — | |
YNRIRGBEDNUPFT
|
7.5 | IC50 | 3 | — | |
ZBDDVAPOFCENEY
|
7.5 | IC50 | 2 | — | |
BIAIXZOAJTVRMZ
|
7.5 | IC50 | 3 | — | |
BQQAHRHHVVWUHO
|
7.5 | IC50 | 3 | — | |
HZVBRPJHCZVDIS
|
7.5 | IC50 | 2 | — | |
LTXJHGWRFQTURD
|
7.5 | IC50 | 2 | — | |
UOGUAODRHCJVGQ
|
7.5 | Ki | 2 | — | |
WFWPOGDKKNYHRY
|
7.5 | IC50 | 3 | — | |
CCHANKFDJCNRBT
|
7.5 | IC50 | 7 | — | |
FGFCASMMJUWFQC
|
7.5 | IC50 | 2 | — | |
FMYAQBNTFWSMBU
|
7.5 | IC50 | 3 | — | |
HEHKSPSHGQTIPU
|
7.5 | IC50 | 2 | — | |
JUYFHSJCSCDZBU
|
7.5 | IC50 | 2 | — | |
LDATUNFLUNWYEU
|
7.5 | IC50 | 2 | — | |
METHPDNWVRUNEU
|
7.5 | IC50 | 2 | — | |
MHGBPCHKZVKWKS
|
7.5 | IC50 | 3 | — | |
OEQSIDVSRQIXCR
|
7.5 | IC50 | 2 | — | |
QWBDJIXFGDXIAT
|
7.5 | IC50 | 3 | — |