Target Details
| UniProt AC | Q05513 |
|---|---|
| Gene Symbol | PRKCZ |
| Protein Name | Protein kinase C zeta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00564 (PB1) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 166
- Clinical molecules 93
- Avg pChEMBL 7.14
KEGG Pathways (16)
- AGE-RAGE signaling pathway in diabetic complications
- Axon guidance
- Chemokine signaling pathway
- Diabetic cardiomyopathy
- Endocytosis
- Fluid shear stress and atherosclerosis
- Hippo signaling pathway
- Human papillomavirus infection
- Insulin resistance
- Insulin signaling pathway
- Platelet activation
- Rap1 signaling pathway
- Relaxin signaling pathway
- Sphingolipid signaling pathway
- Tight junction
- Type II diabetes mellitus
Active Molecules (166)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NTXWXFSAJRMWNA
|
6.7 | IC50 | 15 | — | |
RAOJISQDGOOXTK
|
6.7 | IC50 | 14 | Yes | |
YISMQBFJYDFMAL
|
6.7 | IC50 | 46 | — | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
GZJKVFKNTQXSQM
|
6.7 | IC50 | 12 | Yes | |
MZNUNTIEUOYNNT
|
6.6 | IC50 | 12 | Yes | |
OXEOHAXVZADDOC
|
6.6 | IC50 | 12 | Yes | |
YSVVBGPTTSJYPA
|
6.6 | IC50 | 12 | Yes | |
FUMCKNCUEAQHCV
|
6.6 | Ki | 103 | — | |
KOZFSFOOLUUIGY
|
6.6 | IC50 | 26 | — | |
QMGUOJYZJKLOLH
|
6.6 | IC50 | 21 | Yes | |
SSZFVGXDYBMVDD
|
6.6 | IC50 | 12 | Yes | |
PBCZSGKMGDDXIJ
|
6.6 | IC50 | 12 | Yes | |
LAOIBIIMKUINJL
|
6.6 | IC50 | 12 | Yes | |
IXOVKVHWGKDXKQ
|
6.6 | IC50 | 12 | Yes | |
BRZYOTMFHLERHD
|
6.5 | Ki | 17 | Yes | |
XNKIVXYFRPYKHO
|
6.5 | IC50 | 12 | Yes | |
TVIALAOHRQNPOI
|
6.5 | IC50 | 12 | Yes | |
HPCPUHOULFPBCQ
|
6.5 | IC50 | 12 | Yes | |
JDZXLEPJWLCESI
|
6.5 | IC50 | 12 | Yes | |
RHBWAFDCVFMIFK
|
6.5 | IC50 | 12 | Yes | |
RPLXVENRWORMRX
|
6.4 | IC50 | 12 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | IC50 | 147 | Yes | |
MQFYZWYYZGTHAN
|
6.4 | IC50 | 14 | — | |
UMTWTCVTRDYHQQ
|
6.4 | Ki | 56 | — | |
USHMNZBDAOGLMB
|
6.4 | Ki | 26 | — | |
YWTBGJGMTBHQTM
|
6.4 | Ki | 65 | — | |
KAJXOWFGKYKMMZ
|
6.4 | IC50 | 26 | Yes | |
ZFNQOYBHHLGQDV
|
6.3 | IC50 | 12 | Yes | |
BMBIKZHGTPMMMM
|
6.3 | IC50 | 14 | — | |
CPRVBHBRBVVLHL
|
6.3 | IC50 | 11 | — | |
ATBAETXFFCOZOY
|
6.3 | IC50 | 39 | — | |
CCRCRSXDKXZDGK
|
6.3 | IC50 | 12 | Yes | |
JSPAUBUYPPZXSG
|
6.3 | Ki | 17 | Yes | |
ORNADCNXUPZOQN
|
6.3 | IC50 | 15 | — | |
TXGUECVFNFKTBD
|
6.3 | IC50 | 2 | — | |
NEGCBIBMPAHBIM
|
6.3 | IC50 | 12 | Yes | |
BAQFZMFDZMQJAM
|
6.2 | IC50 | 12 | Yes | |
TXBFOGDMTCNBBT
|
6.2 | IC50 | 12 | Yes | |
BSFNGHCTZDCQBF
|
6.2 | Ki | 93 | — | |
DPRGOXVMSNDADU
|
6.2 | Ki | 16 | — | |
HLXIFVDYTGEUJV
|
6.2 | IC50 | 15 | Yes | |
NJPWCTYVEJIQBM
|
6.2 | Ki | 72 | — | |
OUJZYQBEFNDJQN
|
6.2 | Ki | 71 | — | |
KPJDEGAKXAUVAC
|
6.2 | Ki | 15 | Yes | |
CWFIQHQECWPWQG
|
6.2 | IC50 | 16 | Yes | |
ORNADCNXUPZOQN
|
6.2 | IC50 | 15 | — | |
AXTAPYRUEKNRBA
|
6.1 | IC50 | 24 | — | |
CHTMRWQLNNRRFJ
|
6.1 | Ki | 70 | — | |
RKUKAACYUCUJEE
|
6.1 | Ki | 58 | — |