Target Details
| UniProt AC | Q04912 |
|---|---|
| Gene Symbol | MST1R |
| Protein Name | Macrophage-stimulating protein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 158
- Clinical molecules 28
- Avg pChEMBL 7.04
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZDKLVOWGIOKTN
|
6.6 | Ki | 80 | — | |
RITAVMQDGBJQJZ
|
6.6 | Ki | 33 | — | |
RTYJMUXLFRYRBU
|
6.6 | Ki | 35 | — | |
UFYWONKSWCXKNY
|
6.6 | IC50 | 5 | — | |
ZJDFSKSBQBPOSK
|
6.6 | IC50 | 24 | Yes | |
DKZYXHCYPUVGAF
|
6.5 | Kd | 112 | — | |
ADLPKFFMGIJZIM
|
6.5 | Ki | 44 | — | |
AUDNGNGLLRZLDR
|
6.5 | Ki | 33 | — | |
KTEIFNKAUNYNJU
|
6.5 | Ki | 48 | — | |
KUNZDWIFPOMUOX
|
6.5 | Ki | 36 | — | |
XZWVOUQIYLZUCJ
|
6.5 | Ki | 23 | — | |
ZDPGLLQANLROFM
|
6.5 | Ki | 17 | — | |
FERXSPCVEYOEDT
|
6.5 | IC50 | 4 | — | |
HTZHPXKKPOLGTR
|
6.5 | IC50 | 9 | — | |
MJMQNGOVXMCDGQ
|
6.5 | IC50 | 2 | — | |
MVAYPHGEGDDSJN
|
6.5 | IC50 | 6 | — | |
MFYBSISLMUXOGK
|
6.4 | IC50 | 2 | — | |
OPMJBWVXRQIVBZ
|
6.4 | IC50 | 8 | — | |
AOFGEEDOUASHKV
|
6.4 | Ki | 4 | — | |
BLQYVHBZHAISJM
|
6.4 | Ki | 54 | — | |
IFPPYSWJNWHOLQ
|
6.4 | Ki | 52 | Yes | |
WRZNQKSBJJKEBD
|
6.4 | Ki | 6 | — | |
NPKHYQHLPSZNHP
|
6.4 | IC50 | 2 | — | |
UXBXTSWBNHTFRX
|
6.4 | IC50 | 3 | Yes | |
QCKKTDVCCCBGDD
|
6.4 | IC50 | 8 | — | |
OIOZTIQUNWLFQV
|
6.3 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.3 | Kd | 220 | — | |
ODPGGGTTYSGTGO
|
6.3 | Kd | 153 | — | |
WVXNSAVVKYZVOE
|
6.3 | IC50 | 92 | — | |
NKEUPUJTVALZIK
|
6.3 | Ki | 28 | — | |
ZGDYBJXDIXVTLV
|
6.3 | Ki | 54 | — | |
IKPJWGNTDNCFPS
|
6.2 | Ki | 3 | — | |
JAHNZCXMCGWZMZ
|
6.2 | IC50 | 2 | Yes | |
QQWUGDVOUVUTOY
|
6.2 | Kd | 231 | Yes | |
AEYLJTAIDDIOBA
|
6.2 | Ki | 53 | — | |
ATGVCJYHNOSZEV
|
6.2 | Ki | 23 | — | |
QLWUDWMYFSWGHK
|
6.2 | Ki | 22 | — | |
MYPQPZOTEGVVQY
|
6.2 | Ki | 3 | — | |
VLBZFDFQVGAJSP
|
6.1 | IC50 | 2 | — | |
HXHAJRMTJXHJJZ
|
6.1 | Kd | 52 | Yes | |
DFMCXVONDDGQIY
|
6.1 | Ki | 66 | — | |
GCIKSSRWRFVXBI
|
6.1 | Ki | 109 | Yes | |
JRLSUZIPUYDUKX
|
6.1 | Ki | 22 | — | |
MASJMHFQMYAPJR
|
6.1 | Ki | 41 | — | |
NECQZMQPXFYVOY
|
6.1 | Ki | 26 | — | |
UQNNJYLAPYGZBD
|
6.1 | Ki | 28 | — | |
UYJNQQDJUOUFQJ
|
6.1 | Ki | 68 | — | |
VSVWQTDDGQSGHP
|
6.1 | Ki | 51 | — | |
ZGZVRPRSFXRGCF
|
6.1 | Ki | 76 | — | |
ZLLCVOJWNDZXIO
|
6.1 | Ki | 11 | — |