Target Details
| UniProt AC | Q04912 |
|---|---|
| Gene Symbol | MST1R |
| Protein Name | Macrophage-stimulating protein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 158
- Clinical molecules 28
- Avg pChEMBL 7.04
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BULVKSWQYNUHHB
|
7.3 | IC50 | 2 | — | |
JSDFIHRUQVWHKK
|
7.3 | IC50 | 2 | — | |
ABXAHAOCSWBNBG
|
7.2 | IC50 | 2 | Yes | |
GUGPWGWLXMBBBT
|
7.2 | IC50 | 2 | Yes | |
SDBOIBYRBWPIEL
|
7.2 | Ki | 31 | — | |
WDARYLSSWBWVCU
|
7.2 | Ki | 49 | — | |
XKFTZKGMDDZMJI
|
7.2 | Ki | 56 | — | |
OYONTEXKYJZFHA
|
7.2 | IC50 | 69 | Yes | |
ONIQOQHATWINJY
|
7.2 | IC50 | 25 | — | |
ZCCPLJOKGAACRT
|
7.2 | Kd | 599 | — | |
LVYXERPKYAQGKM
|
7.2 | IC50 | 4 | — | |
KTEIFNKAUNYNJU
|
7.1 | IC50 | 114 | — | |
CIGNUCKEHATOKY
|
7.1 | IC50 | 2 | Yes | |
DUTNABYDBFVZOA
|
7.1 | Ki | 3 | — | |
KOSDHWQYVDNUML
|
7.1 | Ki | 3 | Yes | |
XUFLBSMTYMFOQH
|
7.1 | Ki | 43 | — | |
QODZCSPDZVDCSD
|
7.1 | IC50 | 7 | — | |
JWQRJKUZDUQDNX
|
7.0 | IC50 | 3 | — | |
XTBHHEIOMKZKGA
|
7.0 | IC50 | 2 | Yes | |
QOMGQLZYIUPQLG
|
7.0 | IC50 | 7 | — | |
VWCZORWQNKCYGE
|
7.0 | IC50 | 17 | — | |
FUMCKNCUEAQHCV
|
7.0 | Ki | 103 | — | |
KDKUVYLMPJIGKA
|
7.0 | Ki | 91 | Yes | |
LJKJYKWDLJUZHA
|
7.0 | Ki | 24 | — | |
LOYACYJWFBZPCW
|
7.0 | IC50 | 3 | — | |
RGNHKJWHFIPHIM
|
7.0 | Ki | 66 | — | |
UJBJWYNPUOLFIZ
|
7.0 | Ki | 49 | — | |
WAKGEHXTOOFEAE
|
7.0 | Ki | 27 | — | |
BDTVSYMIPDPQBV
|
6.9 | IC50 | 5 | — | |
NVRXTLZYXZNATH
|
6.9 | Ki | 47 | Yes | |
RFKWZWJQRQCLJF
|
6.9 | IC50 | 2 | — | |
RFKWZWJQRQCLJF
|
6.9 | IC50 | 2 | — | |
WDAHGVLBPINGHW
|
6.8 | IC50 | 6 | — | |
LKHSVIZPSAOZJI
|
6.8 | IC50 | 2 | — | |
DPEXRCOBPACFOO
|
6.8 | Ki | 36 | — | |
HZPACYSNLOCDLW
|
6.8 | Ki | 48 | — | |
OAVGBZOFDPFGPJ
|
6.8 | Ki | 42 | Yes | |
SEZFNTZQMWJIAI
|
6.8 | Ki | 22 | — | |
OEUQPIPNLAICFE
|
6.8 | IC50 | 3 | Yes | |
PEGWVOKOYYAQEV
|
6.7 | Ki | 9 | — | |
CGLQYOUHMNTUAK
|
6.7 | IC50 | 2 | — | |
JZTOUVBEZONDKA
|
6.7 | Ki | 80 | — | |
LBVKEEFIPBQIMD
|
6.7 | Ki | 27 | — | |
ZCBUQCWBWNUWSU
|
6.7 | Ki | 11 | — | |
ZCCJKVBTHCOISJ
|
6.7 | Ki | 46 | — | |
HKSZLNNOFSGOKW
|
6.7 | IC50 | 408 | — | |
UVABKUWKYDJFPD
|
6.7 | IC50 | 2 | — | |
QACCVOJRKKIYFM
|
6.6 | IC50 | 3 | — | |
BRTHUECZMVKNMQ
|
6.6 | Ki | 31 | — | |
HAYYBYPASCDWEQ
|
6.6 | Ki | 47 | — |