Target Details
| UniProt AC | Q04912 |
|---|---|
| Gene Symbol | MST1R |
| Protein Name | Macrophage-stimulating protein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG) |
Summary
- Multi-target molecules 158
- Clinical molecules 28
- Avg pChEMBL 7.04
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.6 | Ki | 118 | — | |
SBLMCLDRWJNEJK
|
9.0 | Ki | 17 | — | |
UVNDVSUMHWZESZ
|
8.9 | Ki | 8 | Yes | |
NWMPVMMGSHXANZ
|
8.8 | Ki | 58 | — | |
VNBRGSXVFBYQNN
|
8.7 | IC50 | 22 | Yes | |
XHIQDQUOOKVPRP
|
8.7 | IC50 | 4 | — | |
HVCCYRAHPMMFKT
|
8.7 | IC50 | 2 | — | |
CTSDMCNSBRVZGJ
|
8.7 | IC50 | 2 | — | |
CTSDMCNSBRVZGJ
|
8.6 | IC50 | 7 | — | |
GZVQZLVAKXRTHU
|
8.5 | IC50 | 7 | — | |
SEJGTFPOEJWEGG
|
8.5 | Kd | 149 | — | |
FQIRYXKZWMEKES
|
8.5 | IC50 | 8 | — | |
CXQHYVUVSFXTMY
|
8.5 | IC50 | 154 | — | |
QHADVLVFMKEIIP
|
8.4 | IC50 | 9 | — | |
KEDANNMRCOENMZ
|
8.4 | IC50 | 7 | — | |
CTSDMCNSBRVZGJ
|
8.2 | IC50 | 2 | — | |
AYNVIPPTDMPZRW
|
8.2 | IC50 | 2 | — | |
JGEBLDKNWBUGRZ
|
8.2 | IC50 | 20 | Yes | |
VMJFTOSOFDEKTM
|
8.2 | IC50 | 2 | — | |
OWRXHGAFWZFFCW
|
8.1 | Ki | 113 | — | |
UYMSIPINLJNNOU
|
8.1 | IC50 | 4 | — | |
GLBZSOQDAOLMGC
|
8.0 | IC50 | 23 | Yes | |
WPHKIQPVPYJNAX
|
8.0 | Ki | 81 | — | |
CXWRJKJKIGCZER
|
7.8 | IC50 | 2 | — | |
JPWGMNSPCZZICA
|
7.8 | IC50 | 4 | — | |
AEXYDYPBGQQOMN
|
7.8 | IC50 | 2 | — | |
PSTHAQGLUUIJDB
|
7.7 | IC50 | 6 | — | |
DVRMYRDLCLUXQP
|
7.7 | IC50 | 2 | — | |
FVPYEAORCOKOLV
|
7.7 | IC50 | 6 | — | |
PSTHAQGLUUIJDB
|
7.7 | IC50 | 4 | — | |
RYYNGWLOYLRZLK
|
7.7 | Ki | 104 | — | |
LVVUVXCYFVJIIX
|
7.6 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
7.6 | Ki | 137 | Yes | |
PROLIXHVRCJEFH
|
7.6 | Ki | 46 | — | |
UQRCJCNVNUFYDX
|
7.6 | Kd | 27 | — | |
WINHZLLDWRZWRT
|
7.6 | Ki | 66 | — | |
HBFSOOUBBFCSKA
|
7.6 | IC50 | 2 | — | |
ONSZEUCTVQJHOZ
|
7.5 | Ki | 9 | — | |
DQVUCDBOFDTXMU
|
7.5 | IC50 | 5 | — | |
UKRFXUSHZYFIGR
|
7.5 | IC50 | 2 | Yes | |
WLWPMTAGPLBRJQ
|
7.5 | IC50 | 2 | Yes | |
ZRZMXDFMUVZMFF
|
7.5 | IC50 | 2 | — | |
VCFDMLBPASGZTP
|
7.5 | Ki | 38 | — | |
VKBFHTIUXUCYRQ
|
7.5 | Ki | 66 | — | |
VNDWQCSOSCCWIP
|
7.5 | Ki | 39 | Yes | |
BXBIAORMFZJTAV
|
7.5 | IC50 | 2 | — | |
XVUGJMRSDJSHFU
|
7.5 | IC50 | 2 | — | |
UOVCGJXDGOGOCZ
|
7.4 | Ki | 59 | — | |
ZWQGPGURLYBTGX
|
7.4 | IC50 | 2 | Yes | |
LQVXSNNAFNGRAH
|
7.4 | IC50 | 33 | Yes |