Target Details
UniProt ACQ04912
Gene SymbolMST1R
Protein NameMacrophage-stimulating protein receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF07714 (PK_Tyr_Ser-Thr) PF01437 (PSI) PF01403 (Sema) PF01833 (TIG)
Summary
  • Multi-target molecules 158
  • Clinical molecules 28
  • Avg pChEMBL 7.04
KEGG Pathways (1)
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (158)
InChIKey pChEMBL Type Targets Clinical
HKSZLNNOFSGOKW 9.6 Ki 118
SBLMCLDRWJNEJK 9.0 Ki 17
UVNDVSUMHWZESZ 8.9 Ki 8 Yes
NWMPVMMGSHXANZ 8.8 Ki 58
VNBRGSXVFBYQNN 8.7 IC50 22 Yes
XHIQDQUOOKVPRP 8.7 IC50 4
HVCCYRAHPMMFKT 8.7 IC50 2
CTSDMCNSBRVZGJ 8.7 IC50 2
CTSDMCNSBRVZGJ 8.6 IC50 7
GZVQZLVAKXRTHU 8.5 IC50 7
SEJGTFPOEJWEGG 8.5 Kd 149
FQIRYXKZWMEKES 8.5 IC50 8
CXQHYVUVSFXTMY 8.5 IC50 154
QHADVLVFMKEIIP 8.4 IC50 9
KEDANNMRCOENMZ 8.4 IC50 7
CTSDMCNSBRVZGJ 8.2 IC50 2
AYNVIPPTDMPZRW 8.2 IC50 2
JGEBLDKNWBUGRZ 8.2 IC50 20 Yes
VMJFTOSOFDEKTM 8.2 IC50 2
OWRXHGAFWZFFCW 8.1 Ki 113
UYMSIPINLJNNOU 8.1 IC50 4
GLBZSOQDAOLMGC 8.0 IC50 23 Yes
WPHKIQPVPYJNAX 8.0 Ki 81
CXWRJKJKIGCZER 7.8 IC50 2
JPWGMNSPCZZICA 7.8 IC50 4
AEXYDYPBGQQOMN 7.8 IC50 2
PSTHAQGLUUIJDB 7.7 IC50 6
DVRMYRDLCLUXQP 7.7 IC50 2
FVPYEAORCOKOLV 7.7 IC50 6
PSTHAQGLUUIJDB 7.7 IC50 4
RYYNGWLOYLRZLK 7.7 Ki 104
LVVUVXCYFVJIIX 7.6 IC50 2
PIQCTGMSNWUMAF 7.6 Ki 137 Yes
PROLIXHVRCJEFH 7.6 Ki 46
UQRCJCNVNUFYDX 7.6 Kd 27
WINHZLLDWRZWRT 7.6 Ki 66
HBFSOOUBBFCSKA 7.6 IC50 2
ONSZEUCTVQJHOZ 7.5 Ki 9
DQVUCDBOFDTXMU 7.5 IC50 5
UKRFXUSHZYFIGR 7.5 IC50 2 Yes
WLWPMTAGPLBRJQ 7.5 IC50 2 Yes
ZRZMXDFMUVZMFF 7.5 IC50 2
VCFDMLBPASGZTP 7.5 Ki 38
VKBFHTIUXUCYRQ 7.5 Ki 66
VNDWQCSOSCCWIP 7.5 Ki 39 Yes
BXBIAORMFZJTAV 7.5 IC50 2
XVUGJMRSDJSHFU 7.5 IC50 2
UOVCGJXDGOGOCZ 7.4 Ki 59
ZWQGPGURLYBTGX 7.4 IC50 2 Yes
LQVXSNNAFNGRAH 7.4 IC50 33 Yes
2D structure