Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MHXGEROHKGDZGO
|
6.3 | Kd | 10 | — | |
HKSZLNNOFSGOKW
|
6.3 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.3 | Kd | 213 | — | |
ISWRGOFCPBCOGR
|
6.3 | IC50 | 3 | — | |
OXJWXQVCCWDQJS
|
6.3 | IC50 | 6 | — | |
NKZVCOXZDFTYPG
|
6.3 | Ki | 4 | — | |
PROLIXHVRCJEFH
|
6.3 | Ki | 46 | — | |
UIRCQOKSJDLYBB
|
6.3 | Ki | 50 | — | |
QXIDSSPGGSFJDS
|
6.3 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
6.3 | Kd | 64 | Yes | |
FTIGOWUZQQHANO
|
6.3 | IC50 | 3 | — | |
DSDQKAJLESVGJN
|
6.2 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
6.2 | Kd | 165 | Yes | |
ZBNZXTGUTAYRHI
|
6.2 | Kd | 102 | Yes | |
DFMCXVONDDGQIY
|
6.2 | Ki | 66 | — | |
DJRPFIWIDKXORZ
|
6.2 | Ki | 9 | — | |
GKODJBVKKLQMEY
|
6.2 | Ki | 10 | — | |
IPTSYCYNQJITNJ
|
6.2 | Ki | 12 | — | |
QKUFEXGLTQADSA
|
6.2 | Ki | 5 | — | |
VQPBIJGXSXEOCU
|
6.2 | Ki | 24 | — | |
WDARYLSSWBWVCU
|
6.2 | Ki | 49 | — | |
WTMROIBZVGJXRP
|
6.2 | IC50 | 4 | — | |
DEVVDJCRLJUDBW
|
6.2 | IC50 | 2 | — | |
DPDGLGMFKKTTPN
|
6.2 | IC50 | 2 | — | |
ATGVCJYHNOSZEV
|
6.1 | Ki | 23 | — | |
HZPACYSNLOCDLW
|
6.1 | Ki | 48 | — | |
MHWHPWMWKYXCRJ
|
6.1 | Ki | 32 | — | |
NWMPVMMGSHXANZ
|
6.1 | Ki | 58 | — | |
ZIVDOOQUJQJBDA
|
6.1 | Ki | 4 | — | |
NRBSFHSUWBAYCI
|
6.0 | IC50 | 5 | — | |
VMLFWTDHYNRGTR
|
6.0 | IC50 | 2 | — | |
GHIRKOYLRMQNAF
|
6.0 | IC50 | 3 | — | |
AUOSKLDNVNGKRR
|
6.0 | Kd | 6 | — | |
DKXHSOUZPMHNIZ
|
6.0 | Ki | 51 | Yes | |
DWTNLZZEPSCAIH
|
6.0 | Ki | 25 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JUTMUSMWCYHBGU
|
6.0 | Ki | 3 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
PFTXFNSHFZLJNT
|
6.0 | IC50 | 17 | — | |
QFHRPRDSAHFZEG
|
6.0 | Ki | 6 | — | |
QLWUDWMYFSWGHK
|
6.0 | Ki | 22 | — | |
SLCFEJAMCRLYRG
|
6.0 | IC50 | 8 | Yes | |
ZGZVRPRSFXRGCF
|
6.0 | Ki | 76 | — |