Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CNEUJSQUCXSRDD
|
6.8 | IC50 | 7 | — | |
SGIKWGLEUPAMLM
|
6.8 | IC50 | 3 | — | |
BNRSWMLKHCENGN
|
6.8 | IC50 | 2 | — | |
NEBJGJOGYMUDIV
|
6.7 | IC50 | 3 | — | |
QCEHAYINFMPPPM
|
6.7 | IC50 | 3 | — | |
XRONIIQINPKHFL
|
6.7 | IC50 | 2 | — | |
NBSJZWFDNFWQDN
|
6.7 | IC50 | 29 | — | |
ADLPKFFMGIJZIM
|
6.7 | Ki | 44 | — | |
CSEOMSQIOBWXNZ
|
6.7 | IC50 | 3 | — | |
SDTHQOXRWZXTJF
|
6.7 | Ki | 16 | — | |
YNUMBZPWLHDVEX
|
6.7 | Ki | 6 | — | |
ZCCJKVBTHCOISJ
|
6.7 | Ki | 46 | — | |
ZGDYBJXDIXVTLV
|
6.7 | Ki | 54 | — | |
OIDBPSOIVPMQGT
|
6.7 | IC50 | 2 | — | |
QPIFMCLNACVAAT
|
6.7 | IC50 | 7 | — | |
RXPZOSHFGJWSLQ
|
6.7 | IC50 | 6 | — | |
DKZYXHCYPUVGAF
|
6.7 | Kd | 112 | — | |
QWRZWSKROKOPNQ
|
6.6 | IC50 | 2 | — | |
UVOJVOHBYLNVCM
|
6.6 | IC50 | 2 | — | |
MCKKWYKONXTPFI
|
6.6 | IC50 | 3 | — | |
BSVRVRYBQFKTMV
|
6.6 | IC50 | 3 | — | |
BXMKDTWGFLBPKB
|
6.6 | IC50 | 2 | — | |
UOVCGJXDGOGOCZ
|
6.6 | Ki | 59 | — | |
VKBFHTIUXUCYRQ
|
6.6 | Ki | 66 | — | |
WKDACQVEJIVHMZ
|
6.6 | Kd | 46 | — | |
ITRDMWUZJMBHJF
|
6.6 | IC50 | 2 | — | |
PISUPWGJJGVRQG
|
6.6 | IC50 | 2 | — | |
XGUIEYMNFRMLPV
|
6.5 | IC50 | 6 | — | |
AKOPMGQQNOSEED
|
6.5 | IC50 | 4 | — | |
BJVDFBKBRZLKCF
|
6.5 | IC50 | 2 | — | |
FVAUWSNXHKYZKA
|
6.5 | IC50 | 4 | — | |
GTJCBPZCSZZPQO
|
6.5 | IC50 | 3 | — | |
IAXXRGACLVIRBH
|
6.5 | IC50 | 3 | — | |
OJGOVIODTPNPDG
|
6.5 | IC50 | 3 | — | |
OKNNCKJQXLUIJK
|
6.5 | IC50 | 3 | — | |
OXJWXQVCCWDQJS
|
6.5 | IC50 | 3 | — | |
OZCYACNGDDKBEX
|
6.5 | IC50 | 3 | — | |
PGRJFPIBHFUXKF
|
6.5 | IC50 | 3 | — | |
AJIRLUWVMCLWFU
|
6.5 | IC50 | 2 | — | |
JWLJDRWZFALRKE
|
6.5 | Ki | 3 | — | |
YEKVTSRZMPLPFK
|
6.5 | Ki | 17 | — | |
AMLGBGSXVKQKOZ
|
6.5 | IC50 | 3 | — | |
OGJHYZPOJBSQJC
|
6.5 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
RVYNOQUUDOREOT
|
6.4 | IC50 | 2 | — | |
HXHAJRMTJXHJJZ
|
6.4 | Ki | 52 | Yes | |
RYYNGWLOYLRZLK
|
6.4 | Ki | 104 | — | |
WPHKIQPVPYJNAX
|
6.4 | Ki | 81 | — | |
XAVIPIHNPPAYAJ
|
6.4 | IC50 | 3 | — | |
KTEIFNKAUNYNJU
|
6.4 | Kd | 114 | — |