Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RTYJMUXLFRYRBU
|
7.0 | Ki | 35 | — | |
VCFDMLBPASGZTP
|
7.0 | Ki | 38 | — | |
XHBVYDAKJHETMP
|
7.0 | IC50 | 24 | Yes | |
MDGXLOFLFFEXSH
|
7.0 | IC50 | 2 | — | |
SQRAKIQIMGAALF
|
7.0 | IC50 | 2 | — | |
UOAHJPVGHFVHGE
|
7.0 | IC50 | 4 | — | |
OFEFRENRYAYAGU
|
7.0 | IC50 | 2 | — | |
AWYCHWICAWWJPC
|
7.0 | IC50 | 2 | — | |
FAAFMTXOUNMIAO
|
7.0 | IC50 | 2 | — | |
GIAGHNVPQYZDIK
|
7.0 | IC50 | 3 | — | |
JMIFGARJSWXZSH
|
7.0 | IC50 | 3 | — | |
GGQCWUKLPMFTDA
|
7.0 | IC50 | 5 | — | |
GHUBYLSYFHNRLX
|
7.0 | IC50 | 2 | — | |
IIYOBXCNRFSCBH
|
7.0 | IC50 | 8 | — | |
WJSYQJFCHPTVCI
|
6.9 | IC50 | 3 | — | |
QIGLCSOIUAUGES
|
6.9 | IC50 | 2 | — | |
CXZJXVJPISUKMR
|
6.9 | IC50 | 6 | — | |
JWSRLZGLCYGKSQ
|
6.9 | IC50 | 2 | — | |
LCVIRAZGMYMNNT
|
6.9 | Kd | 20 | — | |
MPUAEAFJNJDWLV
|
6.9 | IC50 | 3 | — | |
SLPKIKLAGAHKDI
|
6.9 | IC50 | 2 | — | |
ZAMFNZGKRRMOFE
|
6.9 | IC50 | 2 | — | |
AXHZUYXKPFPWMO
|
6.9 | IC50 | 2 | — | |
FPLAQCFCGCSDRB
|
6.9 | Ki | 4 | — | |
QKQYCTJIQVLCOH
|
6.9 | Ki | 2 | — | |
QYTUSJSFZCPMSV
|
6.9 | IC50 | 2 | — | |
RGNHKJWHFIPHIM
|
6.9 | Ki | 66 | — | |
WRZNQKSBJJKEBD
|
6.9 | Ki | 6 | — | |
XKFTZKGMDDZMJI
|
6.9 | Ki | 56 | — | |
ICKRRSVRNGVVPJ
|
6.9 | IC50 | 2 | — | |
LDBDZEBZXYQPTJ
|
6.9 | IC50 | 2 | — | |
UOTRHTRIIAWPIM
|
6.9 | IC50 | 3 | — | |
JTWDQFJHOKLOHG
|
6.9 | IC50 | 3 | — | |
GVISBDZSDFJHJS
|
6.8 | IC50 | 3 | — | |
HGJYCMLNAQLZFL
|
6.8 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
6.8 | Kd | 191 | — | |
FGLKZAVLKCAKGX
|
6.8 | IC50 | 2 | — | |
UPGITVUUJFWGDH
|
6.8 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.8 | Kd | 139 | — | |
LCNMZQCSKWYNQF
|
6.8 | IC50 | 2 | — | |
UHTHHESEBZOYNR
|
6.8 | Kd | 66 | Yes | |
ILUYOBAWAMCPBZ
|
6.8 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
6.8 | Ki | 48 | — | |
NMHMCXTYPRADBA
|
6.8 | Ki | 20 | — | |
OWRXHGAFWZFFCW
|
6.8 | Ki | 113 | — | |
TVUWQDLBEOZVOU
|
6.8 | Ki | 41 | — | |
UKJHXNZUFMVJFI
|
6.8 | IC50 | 3 | — | |
ULQWBLKUEAKIFZ
|
6.8 | IC50 | 2 | — | |
URUAVMYQAQXGRF
|
6.8 | IC50 | 2 | — | |
VAARYSWULJUGST
|
6.8 | Kd | 119 | Yes |