Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UOBWTNVFBCTTAN
|
7.2 | IC50 | 2 | — | |
GUGWAPHGUQVWRA
|
7.2 | IC50 | 3 | — | |
CWORZSMRYNSMCN
|
7.2 | IC50 | 3 | — | |
NNGJBTGAVCLGTM
|
7.2 | IC50 | 2 | — | |
HZMKNGJNPOBODV
|
7.2 | IC50 | 4 | — | |
IFSNOUHZJMGMOD
|
7.2 | IC50 | 4 | — | |
QKGNJQNQCKFAFD
|
7.2 | IC50 | 2 | — | |
SOXBHNNRUKELLI
|
7.2 | IC50 | 3 | — | |
ALEALKZBRLEOJZ
|
7.2 | IC50 | 3 | — | |
IEJPGJXAWUJROQ
|
7.2 | IC50 | 5 | — | |
KIUMBIWMXBUHDW
|
7.2 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.2 | Ki | 118 | — | |
NVRXTLZYXZNATH
|
7.2 | Ki | 47 | Yes | |
OLUKILHGKRVDCT
|
7.2 | Ki | 44 | Yes | |
PBBRWFOVCUAONR
|
7.2 | Ki | 26 | Yes | |
ZAEAGGGBPKOFMY
|
7.2 | Ki | 3 | — | |
NJDLQMXEEQORLU
|
7.2 | IC50 | 2 | — | |
HIWHLPKRUZGHRR
|
7.2 | IC50 | 4 | — | |
STQMBDHGSGMKRK
|
7.2 | IC50 | 2 | — | |
WIMYXIDFXOAJPL
|
7.2 | IC50 | 3 | — | |
FYPPBYUPMODRPA
|
7.2 | IC50 | 4 | — | |
OVNAOUBDNBHVCI
|
7.2 | IC50 | 5 | — | |
QKDBOJCTMDJVMH
|
7.2 | IC50 | 4 | — | |
QIXWNWRGNUGMRT
|
7.1 | IC50 | 2 | — | |
BCCXLOMXYXXNIU
|
7.1 | IC50 | 2 | — | |
CCKKGJFQFLRASM
|
7.1 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
LOLPPWBBNUVNQZ
|
7.1 | Kd | 97 | Yes | |
YOKGFEAEVZNOAR
|
7.1 | IC50 | 5 | — | |
LJUBHCPBQBKBHM
|
7.1 | IC50 | 5 | — | |
NTLWKKILBCETHV
|
7.1 | IC50 | 4 | — | |
TVXUSVBFYFEVJT
|
7.1 | IC50 | 2 | — | |
CLSVHDFWSGQNQH
|
7.1 | IC50 | 2 | — | |
QKIQUHJMKMTYPI
|
7.1 | IC50 | 2 | — | |
SUZKCUIXBPKMPQ
|
7.1 | IC50 | 2 | — | |
ZWIZYDKWXQTSEQ
|
7.1 | IC50 | 2 | — | |
RQXROVVCXFAAOM
|
7.1 | IC50 | 2 | — | |
XIFIYBGPRFRYNP
|
7.1 | IC50 | 4 | — | |
FZJGVHATMCAPLO
|
7.0 | IC50 | 5 | — | |
GGDVEPRDLUWBFD
|
7.0 | IC50 | 4 | — | |
KRLRRZRTVIVROZ
|
7.0 | IC50 | 3 | — | |
VUEWHTWKZUEQMF
|
7.0 | IC50 | 4 | — | |
GHUBYLSYFHNRLX
|
7.0 | IC50 | 2 | — | |
QXZQWTRSWYLAFO
|
7.0 | IC50 | 3 | — | |
FCKKBQZIGVYODN
|
7.0 | IC50 | 4 | — | |
YCFHQBMHEXTGMF
|
7.0 | IC50 | 2 | — | |
DHQCKBUTDYGTKB
|
7.0 | IC50 | 3 | — | |
DPEXRCOBPACFOO
|
7.0 | Ki | 36 | — | |
PDSJQPLUVYRPDN
|
7.0 | IC50 | 3 | — | |
QZPFUALVXZAFDD
|
7.0 | Ki | 10 | — |