Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBGCUGHOUSPKBA
|
7.5 | IC50 | 2 | — | |
ABEPADPRAQLNSN
|
7.5 | IC50 | 3 | — | |
BLQYVHBZHAISJM
|
7.5 | Ki | 54 | — | |
FVRYPYDPKSZGNS
|
7.5 | IC50 | 2 | — | |
GAIBPGQSYNAFNN
|
7.5 | IC50 | 3 | — | |
HZFKGEGMOFIQKL
|
7.5 | IC50 | 2 | — | |
NZDLTZYLNOKWBF
|
7.5 | IC50 | 2 | — | |
VXWZZARWLSAHEX
|
7.5 | IC50 | 2 | — | |
RUBWYYYEDDAWLB
|
7.5 | IC50 | 5 | — | |
FAOGJKJCGFIFLI
|
7.5 | IC50 | 6 | — | |
NTZZVPFINNIFIF
|
7.5 | IC50 | 2 | — | |
XBGQOGKKOFCYQD
|
7.5 | IC50 | 2 | — | |
ABOWQJUFRKXEIL
|
7.5 | IC50 | 2 | — | |
NNGJBTGAVCLGTM
|
7.5 | IC50 | 2 | — | |
YTUZELSDHUVEFM
|
7.5 | IC50 | 4 | — | |
CJLMANFTWLNAKC
|
7.5 | IC50 | 5 | — | |
ZOMQASFZVQEKHR
|
7.5 | IC50 | 3 | — | |
FFLJVBPCONQSQW
|
7.4 | IC50 | 8 | — | |
JRWJZLHBSKAXJW
|
7.4 | IC50 | 2 | — | |
NSVCYZBCJCPLDO
|
7.4 | IC50 | 2 | — | |
VDXGLZJPQRGNLY
|
7.4 | IC50 | 10 | — | |
CCKKGJFQFLRASM
|
7.4 | IC50 | 2 | — | |
DPDIGSURNQRYQS
|
7.4 | IC50 | 3 | — | |
JUUFLLKHNYWHKP
|
7.4 | Kd | 12 | — | |
TVLFEDKEAOXRCZ
|
7.4 | Ki | 22 | — | |
FVCQZDADSCVUOD
|
7.4 | IC50 | 2 | — | |
HXVUNNJZNBHKIA
|
7.4 | IC50 | 2 | — | |
WLXBZZLKNLKRKJ
|
7.4 | IC50 | 3 | — | |
JDYMCSKANXEKMK
|
7.4 | IC50 | 3 | — | |
DXLXRNZCYAYUED
|
7.4 | IC50 | 2 | — | |
QDSBPGDYULDNNW
|
7.4 | IC50 | 2 | — | |
ROCFHKYAFOQDHC
|
7.4 | IC50 | 5 | — | |
RVRSJCNFHLBUKI
|
7.4 | IC50 | 2 | — | |
WMTXIPYJYDISKM
|
7.4 | IC50 | 8 | — | |
SRPLSQLPBCVKSL
|
7.4 | IC50 | 2 | — | |
UAHBMBZHEHEEAW
|
7.4 | IC50 | 4 | — | |
ABOWQJUFRKXEIL
|
7.3 | IC50 | 2 | — | |
ZCFRPQTXMMLPFH
|
7.3 | IC50 | 2 | — | |
QDSMDFVMOMUBDR
|
7.3 | IC50 | 2 | — | |
WSNLCMQIUFLQBS
|
7.3 | IC50 | 3 | — | |
GNLAGGCSJGJECE
|
7.3 | Ki | 19 | Yes | |
KUNZDWIFPOMUOX
|
7.3 | Ki | 36 | — | |
SLEWGGZPOQNVSU
|
7.3 | Kd | 22 | — | |
WCDLCPLAAKUJNY
|
7.3 | IC50 | 8 | — | |
BKJSJLXWFRXVNO
|
7.3 | IC50 | 2 | — | |
PBPRYPLWJIJEMD
|
7.3 | IC50 | 2 | — | |
UFBDDUGKCAERNV
|
7.3 | IC50 | 2 | — | |
JUACWTBEXKUOOV
|
7.2 | IC50 | 2 | — | |
KPONRYYSJPIILR
|
7.2 | IC50 | 2 | — | |
LMNXBEZQGBWMMY
|
7.2 | IC50 | 3 | — |