Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IFPPYSWJNWHOLQ
|
7.7 | IC50 | 52 | Yes | |
KPRPFTOLWQQUAV
|
7.7 | IC50 | 3 | — | |
MNCBGNHYCLQCSA
|
7.7 | IC50 | 2 | — | |
OBLCGNSTBZOGIQ
|
7.7 | IC50 | 3 | — | |
BAGWVDYVFGYURF
|
7.7 | IC50 | 2 | — | |
DBAUTMSTTOYZCH
|
7.7 | IC50 | 2 | — | |
HWXVIOGONBBTBY
|
7.7 | Kd | 27 | — | |
NYYYLFUSXWJOML
|
7.7 | IC50 | 3 | — | |
OVXMCCQKIOSDGE
|
7.7 | IC50 | 3 | — | |
QQYOZULVMVWDFQ
|
7.7 | IC50 | 3 | — | |
RZYYJEYQNNJBMD
|
7.7 | IC50 | 3 | — | |
WMBPMDQTARNBNK
|
7.7 | IC50 | 2 | — | |
HZFKGEGMOFIQKL
|
7.6 | IC50 | 2 | — | |
IOEZZOIIFUBFFP
|
7.6 | IC50 | 2 | — | |
OVAAGWFAUDJCKW
|
7.6 | IC50 | 2 | — | |
PAHLIVNOHVHPBG
|
7.6 | IC50 | 6 | — | |
UPBPVAZUFAXUAC
|
7.6 | IC50 | 6 | — | |
WBRIXUZLHYMBMA
|
7.6 | IC50 | 2 | — | |
AWERICKZHUFDGO
|
7.6 | IC50 | 3 | — | |
BHUXVRVMMYAXKN
|
7.6 | IC50 | 3 | — | |
DUGKWSLUPDXHDO
|
7.6 | IC50 | 3 | — | |
HSAUZUYGDAHMLS
|
7.6 | IC50 | 2 | — | |
UTCHZVUDAGSGMY
|
7.6 | IC50 | 3 | — | |
XYIZJZFZXCURDK
|
7.6 | IC50 | 5 | — | |
DONRBWYKHKBNAQ
|
7.6 | IC50 | 2 | — | |
PRKWSDOLROTYLX
|
7.6 | IC50 | 3 | — | |
SRIVDECCESIDAQ
|
7.6 | IC50 | 3 | — | |
ZROZDTQXWWJRDP
|
7.6 | IC50 | 2 | — | |
ZNGBDCDUILRYET
|
7.6 | IC50 | 2 | — | |
BBDGBGOVJPEFBT
|
7.6 | IC50 | 6 | — | |
FJHJLNXCFAIWOY
|
7.6 | IC50 | 2 | — | |
QPRFLHHDQOLCJS
|
7.6 | IC50 | 2 | — | |
UXVFRKCJRULCNV
|
7.6 | IC50 | 4 | — | |
BZXHYPDAQAEAKY
|
7.6 | IC50 | 5 | — | |
LDFGETAUTXIODG
|
7.6 | IC50 | 2 | — | |
MZIQJPGLZXVJCP
|
7.6 | IC50 | 2 | — | |
GLJHPFGWEFTXKS
|
7.5 | IC50 | 2 | — | |
GAIBPGQSYNAFNN
|
7.5 | IC50 | 3 | — | |
GMVCGHNKICTUFJ
|
7.5 | IC50 | 2 | — | |
IIXWYSCJSQVBQM
|
7.5 | IC50 | 18 | — | |
KPRPFTOLWQQUAV
|
7.5 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
7.5 | Kd | 231 | Yes | |
UIIXJLLQKFFGKU
|
7.5 | IC50 | 3 | — | |
DDVZCQMFWBEKAW
|
7.5 | IC50 | 2 | — | |
IFZOMAMCUJXLIP
|
7.5 | IC50 | 2 | — | |
MHRAFUWHUFJCFB
|
7.5 | IC50 | 2 | — | |
XASOXDFSRMCVGS
|
7.5 | IC50 | 2 | — | |
XQLHGVZYEZLJEG
|
7.5 | IC50 | 3 | — | |
BLKUTJODYRMUJL
|
7.5 | IC50 | 4 | — | |
RJCVCOCSWGHLMV
|
7.5 | IC50 | 2 | — |