Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GNDTWZQOAXPKCV
|
7.9 | IC50 | 3 | — | |
GPLMXGSESNBQQL
|
7.9 | IC50 | 2 | — | |
JDAFKLSYNCTYHC
|
7.9 | IC50 | 3 | — | |
MOTRKLJWPDOTBN
|
7.9 | IC50 | 2 | — | |
RIGIHWPKCOSNDD
|
7.9 | IC50 | 3 | — | |
XCQPASNBVLQPAI
|
7.9 | IC50 | 2 | — | |
JFDSOYMKCLUKEJ
|
7.9 | IC50 | 2 | — | |
RKBYYWVZFBATHQ
|
7.9 | IC50 | 12 | — | |
SMMLJZCTRMSMMI
|
7.9 | IC50 | 3 | — | |
YPRRJKORYBKLRH
|
7.9 | IC50 | 2 | — | |
DONRBWYKHKBNAQ
|
7.8 | IC50 | 2 | — | |
JHBVJUXBKKKJGW
|
7.8 | IC50 | 2 | — | |
JHBVJUXBKKKJGW
|
7.8 | IC50 | 2 | — | |
JHBVJUXBKKKJGW
|
7.8 | IC50 | 2 | — | |
MEDZXCCPJFWNLJ
|
7.8 | IC50 | 3 | — | |
PBPRYPLWJIJEMD
|
7.8 | IC50 | 2 | — | |
QNXUBBYNLLCNPH
|
7.8 | IC50 | 2 | — | |
WCTODNJGIAJWJX
|
7.8 | IC50 | 2 | — | |
ZRCZZPPDWCVIOL
|
7.8 | IC50 | 2 | — | |
ZYBANBICDUFKMJ
|
7.8 | IC50 | 2 | — | |
AKSKEXPIRSTUBP
|
7.8 | IC50 | 2 | — | |
KVLSZJPFQDRDPI
|
7.8 | IC50 | 4 | — | |
LYZXDNCSIHIAMI
|
7.8 | IC50 | 3 | — | |
WBRIXUZLHYMBMA
|
7.8 | IC50 | 2 | — | |
WFZZPLAPENBNIY
|
7.8 | IC50 | 3 | — | |
DBAUTMSTTOYZCH
|
7.8 | IC50 | 2 | — | |
IONTZIKRBZYYLS
|
7.8 | IC50 | 2 | — | |
KDJGCVHPUMHUOL
|
7.8 | Ki | 11 | — | |
QCXBJMRMYRQRCV
|
7.8 | IC50 | 4 | — | |
GVKXHJBRWOYLAK
|
7.8 | IC50 | 3 | — | |
CDOVNWNANFFLFJ
|
7.8 | IC50 | 10 | — | |
CGAOZJWPBAWCGJ
|
7.8 | IC50 | 2 | — | |
FTSHNQVAJPKPPY
|
7.8 | IC50 | 2 | — | |
MEDZXCCPJFWNLJ
|
7.8 | IC50 | 3 | — | |
WTEJOBNHOMFLQN
|
7.8 | IC50 | 2 | — | |
AOFHPWKDAJCJHE
|
7.7 | IC50 | 2 | — | |
JRWJZLHBSKAXJW
|
7.7 | IC50 | 2 | — | |
JXPPULPLYFLFJI
|
7.7 | IC50 | 3 | — | |
MKKQYAXMQPGYNY
|
7.7 | IC50 | 3 | — | |
NJSRQYMTTJJEJH
|
7.7 | IC50 | 2 | — | |
RCORIFCNLQIMKN
|
7.7 | IC50 | 2 | — | |
RQXROVVCXFAAOM
|
7.7 | IC50 | 3 | — | |
VPAYUAUNRWCJTE
|
7.7 | IC50 | 2 | — | |
WUEJFDOJIBRVBJ
|
7.7 | IC50 | 3 | — | |
ZNGBDCDUILRYET
|
7.7 | IC50 | 3 | — | |
BBWFHMVFMVFXJP
|
7.7 | IC50 | 3 | — | |
TUFWPHNCGNFLJQ
|
7.7 | IC50 | 3 | — | |
XJRNYUDHNXZYCF
|
7.7 | IC50 | 3 | — | |
AJRCHNXNYNADRQ
|
7.7 | IC50 | 3 | — | |
MKKQYAXMQPGYNY
|
7.7 | IC50 | 2 | — |