Target Details
| UniProt AC | Q04771 |
|---|---|
| Gene Symbol | ACVR1 |
| Protein Name | Activin receptor type-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 394
- Clinical molecules 19
- Avg pChEMBL 7.24
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (394)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HULQVTAEMIYULR
|
9.3 | IC50 | 2 | — | |
WJASKODGMHBDFO
|
8.9 | IC50 | 5 | — | |
ZCCPLJOKGAACRT
|
8.8 | Kd | 599 | — | |
ORRRLMFZEDPMSZ
|
8.6 | IC50 | 2 | — | |
DERIBTSHHPNLEG
|
8.5 | IC50 | 2 | — | |
VWACUNWBMWWMPJ
|
8.5 | Ki | 18 | — | |
QFFKJPJEWNRMHC
|
8.5 | IC50 | 2 | — | |
FHTCHCUICJOIGJ
|
8.4 | IC50 | 7 | — | |
CUAUTGRQMYJPFC
|
8.4 | IC50 | 5 | — | |
MFAQYJIYDMLAIM
|
8.4 | Kd | 130 | Yes | |
OUKYUETWWIPKQR
|
8.4 | Kd | 31 | Yes | |
NIOZQSIYXGTSOO
|
8.3 | IC50 | 2 | — | |
KIAKJNRDKPGTQR
|
8.3 | IC50 | 6 | — | |
ALKJNCZNEOTEMP
|
8.3 | Kd | 55 | — | |
JBTJGPURAPMJSS
|
8.3 | IC50 | 3 | — | |
WTNLXMJMLHJDKF
|
8.3 | IC50 | 3 | — | |
MMQQLUARMBFVKE
|
8.3 | IC50 | 2 | — | |
RIWTUJFFSTVYPW
|
8.2 | IC50 | 6 | — | |
ZPKLGSLFCKFOCY
|
8.2 | IC50 | 3 | — | |
YPTIRJISDXITNF
|
8.2 | IC50 | 3 | — | |
WOAXRKYXUKTLEM
|
8.2 | IC50 | 7 | — | |
GPLMXGSESNBQQL
|
8.2 | IC50 | 3 | — | |
NSVCYZBCJCPLDO
|
8.2 | IC50 | 2 | — | |
PTHVKCSYXICMAR
|
8.2 | IC50 | 14 | — | |
MQFUFNHTCJRLKW
|
8.1 | IC50 | 6 | — | |
MXDCACLUETVZNL
|
8.1 | IC50 | 8 | — | |
BBWFHMVFMVFXJP
|
8.1 | IC50 | 3 | — | |
KVDFCDPSKGACEZ
|
8.1 | IC50 | 4 | — | |
KWZMLARYZJWIGD
|
8.1 | IC50 | 3 | — | |
PVDWNOWJXDXMDH
|
8.1 | IC50 | 5 | — | |
SCHRCCHASZMVAB
|
8.1 | IC50 | 7 | — | |
ZBOSAPQCJDMZCV
|
8.1 | IC50 | 6 | — | |
XIAQAOWQYMNJJB
|
8.1 | IC50 | 2 | — | |
GFEAXKZXFORDDU
|
8.1 | IC50 | 2 | — | |
IPESYYFOXATSFJ
|
8.1 | IC50 | 3 | — | |
WAOTXMYGOSUFGX
|
8.1 | IC50 | 3 | — | |
YBDMDASOVBUGSC
|
8.1 | IC50 | 3 | — | |
LRSOQWKCWLRMRR
|
8.0 | IC50 | 2 | — | |
SHWKNOUREYUNBF
|
8.0 | IC50 | 6 | — | |
FCURQEMLQWEPFI
|
8.0 | IC50 | 2 | — | |
ODVUZZFWFOPOAH
|
8.0 | IC50 | 5 | — | |
OTMZESJOOWWVGH
|
8.0 | IC50 | 2 | — | |
SJOCBUINMBQCTH
|
8.0 | IC50 | 2 | — | |
AGBKRFXLWIHJQH
|
8.0 | IC50 | 3 | — | |
AGMGRCAUAZCHPG
|
8.0 | IC50 | 5 | — | |
HZFKGEGMOFIQKL
|
8.0 | IC50 | 2 | — | |
JFDSOYMKCLUKEJ
|
8.0 | IC50 | 2 | — | |
MOTRKLJWPDOTBN
|
8.0 | IC50 | 3 | — | |
NJSRQYMTTJJEJH
|
8.0 | IC50 | 2 | — | |
WCTODNJGIAJWJX
|
8.0 | IC50 | 2 | — |