Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GDEWTWLRSSWVEX
|
8.0 | IC50 | 3 | Yes | |
UHIFMIXIMAHXIB
|
8.0 | IC50 | 6 | — | |
CDXNZQYZADSNCP
|
8.0 | IC50 | 12 | Yes | |
DSXXEELGXBCYNQ
|
8.0 | IC50 | 28 | Yes | |
FFKRSNGYONHGEV
|
8.0 | IC50 | 12 | Yes | |
GJIHZDZOVHMYJS
|
8.0 | IC50 | 3 | Yes | |
MODWLWDUUDGOEB
|
8.0 | IC50 | 5 | Yes | |
OPQUGNXQOSDRMT
|
8.0 | IC50 | 12 | Yes | |
PGWBJRRPIUVOAD
|
8.0 | IC50 | 12 | Yes | |
PXRPXQKBRGMQJJ
|
8.0 | Ki | 2 | — | |
ZJTHRAYTYMYRHI
|
8.0 | IC50 | 2 | — | |
ZKMXMSATAIWGAR
|
8.0 | IC50 | 2 | — | |
SHNAOUAXXNYCRS
|
8.0 | IC50 | 2 | — | |
SZUVPYWZPMECBT
|
8.0 | IC50 | 2 | — | |
FDFNBRWULOMEEQ
|
8.0 | IC50 | 3 | — | |
ZEGIXAPFKAAIOT
|
8.0 | IC50 | 3 | Yes | |
DMTWTBBJQAQFID
|
8.0 | IC50 | 3 | Yes | |
FLWBAZOREVFEAD
|
8.0 | IC50 | 3 | Yes | |
HAYBNIARWRGYIC
|
8.0 | IC50 | 3 | Yes | |
LCLDOTQNYVMPRQ
|
8.0 | IC50 | 3 | Yes | |
OOLJOHRMOKSYKO
|
8.0 | IC50 | 2 | Yes | |
VCVVTOKATIJIQL
|
8.0 | IC50 | 2 | — | |
KOYAHXZNMXHPNA
|
7.9 | IC50 | 2 | — | |
AWKZERSILQVXCP
|
7.9 | IC50 | 3 | Yes | |
BPNUQXPIQBZCMR
|
7.9 | Kd | 83 | Yes | |
GZRXZIIXJPGKRW
|
7.9 | Ki | 2 | — | |
JRKIWLCZVXSNKH
|
7.9 | IC50 | 2 | — | |
MVPSDKPPZLPMBB
|
7.9 | Ki | 7 | Yes | |
MXZMNMJBRPSOOG
|
7.9 | IC50 | 3 | Yes | |
RETKZRRHASOPND
|
7.9 | IC50 | 2 | — | |
RTRUTBCNJSOKHT
|
7.9 | IC50 | 2 | — | |
SUMGTNPLBQXBDN
|
7.9 | IC50 | 3 | Yes | |
ZBGKNKIERAXNKR
|
7.9 | IC50 | 3 | Yes | |
ZQTCWRKVJWJCMV
|
7.9 | IC50 | 3 | Yes | |
GJOXRIYWDHESDF
|
7.9 | Ki | 27 | — | |
KGPGFQWBCSZGEL
|
7.9 | Kd | 59 | Yes | |
XWKJUHBICAMYNW
|
7.9 | IC50 | 6 | — | |
ALLMHFJXFWBPDH
|
7.9 | IC50 | 3 | Yes | |
DDVKURVSLBGSOS
|
7.9 | IC50 | 3 | Yes | |
DNYURFSSJKXPTF
|
7.9 | IC50 | 3 | Yes | |
FAQJIZKBJRQPIA
|
7.9 | IC50 | 3 | Yes | |
GTWLYEVXNCSGBU
|
7.9 | IC50 | 3 | Yes | |
HETWGNHMXYNQPB
|
7.9 | IC50 | 2 | — | |
PBCZSGKMGDDXIJ
|
7.9 | IC50 | 14 | Yes | |
SWZXKBUPFISEFY
|
7.9 | IC50 | 3 | Yes | |
VEMLCWMDXJGJLI
|
7.9 | Ki | 8 | Yes | |
AGJAPEBQOOHERM
|
7.8 | IC50 | 4 | Yes | |
FQUIZYRWNTVYLN
|
7.8 | IC50 | 3 | Yes | |
GPGZMTPPOHCJRE
|
7.8 | IC50 | 16 | Yes | |
IELYDRFCDPGZGF
|
7.8 | Ki | 6 | — |