Target Details
| UniProt AC | Q04759 |
|---|---|
| Gene Symbol | PRKCQ |
| Protein Name | Protein kinase C theta type |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF21494 (PKC_C2) PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 750
- Clinical molecules 360
- Avg pChEMBL 7.71
KEGG Pathways (12)
- Adipocytokine signaling pathway
- Autophagy - animal
- IgSF CAM signaling
- Inflammatory mediator regulation of TRP channels
- Insulin resistance
- NF-kappa B signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Shigellosis
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Vascular smooth muscle contraction
Active Molecules (750)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LPIJVXOQOOJCRR
|
8.2 | IC50 | 3 | Yes | |
XOTNYFMXYDWFEU
|
8.2 | IC50 | 3 | Yes | |
JWTNYYVEXFBGQI
|
8.2 | IC50 | 3 | Yes | |
MKBCGFUOIUKVIQ
|
8.2 | IC50 | 2 | — | |
SAYMBMAHSBYKKR
|
8.2 | IC50 | 12 | Yes | |
GGNGZCWJFMTGIR
|
8.2 | IC50 | 2 | — | |
LBDMJMNVJZNONC
|
8.2 | IC50 | 3 | Yes | |
SPKAGPPMKYJUPF
|
8.2 | IC50 | 3 | Yes | |
RSTWARDIGORXQU
|
8.2 | Ki | 7 | Yes | |
RULYSYJNGRSJSA
|
8.2 | IC50 | 2 | — | |
KAJIDAUQCMSGGN
|
8.2 | IC50 | 3 | Yes | |
GQDKNFXTRUBAEB
|
8.2 | IC50 | 3 | Yes | |
AQGHYUYFBXMRBC
|
8.2 | IC50 | 6 | — | |
JHSOAROIYKSHKX
|
8.2 | IC50 | 3 | Yes | |
VDRCTDRTPPONJY
|
8.2 | IC50 | 2 | — | |
YCFZRTPAYLSXMM
|
8.2 | IC50 | 2 | — | |
KEUYDWVTHJQHIH
|
8.1 | IC50 | 3 | Yes | |
LTGPAFCQBMWTBC
|
8.1 | IC50 | 5 | Yes | |
QFVOPUFBADFYEL
|
8.1 | IC50 | 3 | — | |
CSCOHEYTBLBQMG
|
8.1 | IC50 | 7 | Yes | |
JTUGJZFQRMCZQW
|
8.1 | IC50 | 3 | Yes | |
WYMCAIGTNRBMBV
|
8.1 | IC50 | 2 | — | |
YAHQEFRFUBPDAT
|
8.1 | IC50 | 3 | Yes | |
HTPZZARNXXDSIZ
|
8.1 | IC50 | 2 | — | |
VMRZSNDAPJYPND
|
8.1 | IC50 | 3 | Yes | |
YRYJOPMCJLSMNU
|
8.1 | IC50 | 6 | — | |
DWTNLZZEPSCAIH
|
8.1 | Ki | 25 | — | |
PHDOQFYDQFLEMJ
|
8.1 | IC50 | 3 | Yes | |
PLIDEIVUYFAECO
|
8.1 | IC50 | 2 | — | |
UXZAPNVTOAXLTD
|
8.1 | Ki | 3 | — | |
XUFLBSMTYMFOQH
|
8.1 | Ki | 43 | — | |
DQGXZJOMYLWAKM
|
8.1 | IC50 | 3 | Yes | |
MCIAOHYVDXDCLF
|
8.1 | Ki | 8 | Yes | |
DEAHYBLYNUJAIJ
|
8.1 | IC50 | 3 | Yes | |
JSBPEIYUYLNLLN
|
8.1 | IC50 | 3 | Yes | |
ZRYGSUWUNVQPFR
|
8.1 | IC50 | 6 | — | |
HKSZLNNOFSGOKW
|
8.1 | Kd | 213 | — | |
YHFWETXESAFRRE
|
8.1 | IC50 | 2 | — | |
GQKHMFJDTFXZNM
|
8.1 | IC50 | 5 | Yes | |
LUZOFMGZMUZSSK
|
8.1 | Ki | 8 | Yes | |
WIMTWVOAYCSJHC
|
8.1 | IC50 | 2 | Yes | |
WNYKGJHEQVIFGL
|
8.1 | IC50 | 2 | — | |
JTJAWKUSBMOQSN
|
8.1 | Ki | 5 | — | |
MCQPMCDEXWCMDM
|
8.1 | Ki | 2 | — | |
NDPCMXFATSKLHE
|
8.1 | IC50 | 3 | Yes | |
PJGVITFBPVCDNT
|
8.1 | IC50 | 3 | Yes | |
POTTVLREWUNNRO
|
8.1 | IC50 | 17 | Yes | |
MVYBDSJHHWQUEP
|
8.0 | IC50 | 4 | Yes | |
PEDXJGLVPJEZIK
|
8.0 | IC50 | 3 | Yes | |
BOBBYUSYHORXQS
|
8.0 | IC50 | 2 | Yes |